2-(Thienothiazolylimino)-1,3-thiazolidin-4-ones inhibit cell division cycle 25 A phosphatase

Bioorganic and Medicinal Chemistry

Volumn 24, Issue 13, 2016, Pages 2920-2928

  Huber Villaume, Sophie ^a   Revelant, Germain ^a   Sibille, Estelle ^b   Philippot, Stéphanie ^a   Morabito, Angelica ^a   Dunand, Sandrine ^a   Chaimbault, Patrick ^b   Bagrel, Denyse ^a   Kirsch, Gilbert ^a   Hesse, Stéphanie ^a   Schohn, Hervé ^a  

^a UNIVERSITÉ DE LORRAINE   (France)

^b UNIVERSITÉ DE LORRAINE   (France)

Author keywords

Antiproliferative activities; Breast cancer; CDC25 phosphatases inhibition; Cell cycle arrest; Thiazolyliminothiazolidin 4 ones

Indexed keywords

2 (THIENOTHIAZOLYLIMINO) 1,3 THIAZOLIDIN 4 ONE DERIVATIVE; 4 THIAZOLIDINONE DERIVATIVE; CDC25A; CDC25B; CDC25C; ISOENZYME; NAPHTHOQUINONE; PROTEIN TYROSINE PHOSPHATASE; PROTEIN TYROSINE PHOSPHATASE INHIBITOR; UNCLASSIFIED DRUG; CDC25A PROTEIN, HUMAN; THIAZOLIDINE DERIVATIVE;

ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BACTERICIDAL ACTIVITY; CELL CYCLE PROGRESSION; CELL GROWTH; CONTROLLED STUDY; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; GROWTH INHIBITION; HUMAN; HUMAN CELL; IC50; INFLAMMATION; MCF 7 CELL LINE; PROTEIN EXPRESSION; ANTAGONISTS AND INHIBITORS; BREAST NEOPLASMS; CELL PROLIFERATION; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECTS; FEMALE; MCF-7 CELL LINE; SYNTHESIS;

BREAST NEOPLASMS; CDC25 PHOSPHATASES; CELL PROLIFERATION; FEMALE; HUMANS; INHIBITORY CONCENTRATION 50; MCF-7 CELLS; MOLECULAR STRUCTURE; THIAZOLIDINES;

EID: 84971634890     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2016.04.063     Document Type: Article

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