Inhibition of GPR30 by estriol prevents growth stimulation of triple-negative breast cancer cells by 17β-estradiol

BMC Cancer

Volumn 14, Issue 1, 2014, Pages

  Girgert, Rainer ^a   Emons, Günter ^a   Gründker, Carsten ^a  

^a UNIVERSITY MEDICAL CENTER GÖTTINGEN   (Germany)

Author keywords

Estriol; GPR30; Signal transduction; Targeted therapy; Triple negative breast cancer

Indexed keywords

AROMATASE; CYCLIN D1; EPIDERMAL GROWTH FACTOR RECEPTOR; ESTRADIOL; ESTRIOL; G PROTEIN COUPLED RECEPTOR 30; PHOSPHOTRANSFERASE; PROTEIN C FOS; SRC KINASE; UNCLASSIFIED DRUG; CCND1 PROTEIN, HUMAN; CREB1 PROTEIN, HUMAN; CYCLIC AMP RESPONSIVE ELEMENT BINDING PROTEIN; ESTROGEN; ESTROGEN RECEPTOR; G PROTEIN COUPLED RECEPTOR; GPER PROTEIN, HUMAN;

ARTICLE; BREAST CANCER CELL LINE; CELL COUNT; CELL PROLIFERATION; COLORIMETRY; CONTROLLED STUDY; ENZYME ACTIVATION; ENZYME ACTIVITY; GEL MOBILITY SHIFT ASSAY; INTRACELLULAR SIGNALING; PROTEIN DETERMINATION; PROTEIN EXPRESSION; PROTEIN INDUCTION; PROTEIN PHOSPHORYLATION; PROTEIN TARGETING; REVERSE TRANSCRIPTION POLYMERASE CHAIN REACTION; TRANSACTIVATION; TRIPLE NEGATIVE BREAST CANCER; UPREGULATION; WESTERN BLOTTING; DRUG EFFECTS; GENE EXPRESSION REGULATION; GENETICS; HUMAN; METABOLISM; PATHOLOGY; PHOSPHORYLATION; TUMOR CELL LINE;

CELL LINE, TUMOR; CELL PROLIFERATION; CYCLIC AMP RESPONSE ELEMENT-BINDING PROTEIN; CYCLIN D1; ESTRADIOL; ESTRIOL; ESTROGENS; GENE EXPRESSION REGULATION, NEOPLASTIC; HUMANS; PHOSPHORYLATION; RECEPTORS, ESTROGEN; RECEPTORS, G-PROTEIN-COUPLED; TRIPLE NEGATIVE BREAST NEOPLASMS;

EID: 84965186840     PISSN: None     EISSN: 14712407     Source Type: Journal    
DOI: 10.1186/1471-2407-14-935     Document Type: Article

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