-
1
-
-
15744393640
-
Regulation of signal transduction pathways by estrogen and progesterone
-
Edwards DP, (2005) Regulation of signal transduction pathways by estrogen and progesterone. Annu Rev Physiol 67: 335-376.
-
(2005)
Annu Rev Physiol
, vol.67
, pp. 335-376
-
-
Edwards, D.P.1
-
2
-
-
82155173499
-
The G protein-coupled estrogen receptor GPER in health and disease
-
Prossnitz ER, Barton M, (2011) The G protein-coupled estrogen receptor GPER in health and disease. Nature Reviews Endocrinology 7 (12): 715-726.
-
(2011)
Nature Reviews Endocrinology
, vol.7
, Issue.12
, pp. 715-726
-
-
Prossnitz, E.R.1
Barton, M.2
-
3
-
-
33947401482
-
Integration of rapid signaling events with steroid hormone receptor action in breast and prostate cancer
-
Lange CA, Goalie D, Hammes SR, Marker PC, (2007) Integration of rapid signaling events with steroid hormone receptor action in breast and prostate cancer. Annu Rev Physiol 69: 171-199.
-
(2007)
Annu Rev Physiol
, vol.69
, pp. 171-199
-
-
Lange, C.A.1
Goalie, D.2
Hammes, S.R.3
Marker, P.C.4
-
4
-
-
52949111533
-
Minireview:nuclear receptors and breast cancer
-
Conzen SD, (2008) Minireview:nuclear receptors and breast cancer. Mol Endocrinol 22 (10): 2215-28.
-
(2008)
Mol Endocrinol
, vol.22
, Issue.10
, pp. 2215-2228
-
-
Conzen, S.D.1
-
5
-
-
43549095238
-
Estrogen signaling through the transmembrane G protein-coupled receptor GPR30
-
Prossnitz ER, Arterburn JB, Smith HO, Oprea TI, Sklar LA, et al. (2008) Estrogen signaling through the transmembrane G protein-coupled receptor GPR30. Annu Rev Physiol 70: 165-190.
-
(2008)
Annu Rev Physiol
, vol.70
, pp. 165-190
-
-
Prossnitz, E.R.1
Arterburn, J.B.2
Smith, H.O.3
Oprea, T.I.4
Sklar, L.A.5
-
6
-
-
33751272253
-
Distribution of GPR30, a seven membrane-spanning estrogen receptor, in primary breast cancer and its association with clinicopathologic determinants of tumor progression
-
Filardo EJ, Graeber CT, Quinn JA, Resnic MB, Giri D, et al. (2006) Distribution of GPR30, a seven membrane-spanning estrogen receptor, in primary breast cancer and its association with clinicopathologic determinants of tumor progression. Clin Cancer Res 12: 6359-6366.
-
(2006)
Clin Cancer Res
, vol.12
, pp. 6359-6366
-
-
Filardo, E.J.1
Graeber, C.T.2
Quinn, J.A.3
Resnic, M.B.4
Giri, D.5
-
7
-
-
33947697810
-
GPR30: a novel indicator of poor survival for endometrial carcinoma
-
386.e1-11
-
Smith HO, Leslie KK, Singh M, Qualls CR, Revankar CM, et al. (2007) GPR30: a novel indicator of poor survival for endometrial carcinoma. Am J Obstet Gynecol 196: 386.e1-11.
-
(2007)
Am J Obstet Gynecol
, vol.196
-
-
Smith, H.O.1
Leslie, K.K.2
Singh, M.3
Qualls, C.R.4
Revankar, C.M.5
-
8
-
-
67749119671
-
GPR30 predicts poor survival for ovarian cancer
-
Smith HO, Arias-Pulido H, Kuo DY, Howard T, Qualls CR, et al. (2009) GPR30 predicts poor survival for ovarian cancer. Gynecol Oncol 114 (3): 465-71.
-
(2009)
Gynecol Oncol
, vol.114
, Issue.3
, pp. 465-471
-
-
Smith, H.O.1
Arias-Pulido, H.2
Kuo, D.Y.3
Howard, T.4
Qualls, C.R.5
-
9
-
-
77955774697
-
GPR30 and estrogen receptor expression: new insights into hormone dependence of inflammatory breast cancer
-
Arias-Pulido H, Royce M, Gong Y, Joste N, Lomo L, et al. (2010) GPR30 and estrogen receptor expression: new insights into hormone dependence of inflammatory breast cancer. Breast Cancer Res Treat 123 (1): 51-8.
-
(2010)
Breast Cancer Res Treat
, vol.123
, Issue.1
, pp. 51-58
-
-
Arias-Pulido, H.1
Royce, M.2
Gong, Y.3
Joste, N.4
Lomo, L.5
-
10
-
-
33646366423
-
Virtual and biomolecular screening converge on a selective agonist for GPR30
-
Bologa CG, Revankar CM, Young SM, Edwards BS, Arterburn JB, et al. (2006) Virtual and biomolecular screening converge on a selective agonist for GPR30. Nat Chem Biol 2: 207-212.
-
(2006)
Nat Chem Biol
, vol.2
, pp. 207-212
-
-
Bologa, C.G.1
Revankar, C.M.2
Young, S.M.3
Edwards, B.S.4
Arterburn, J.B.5
-
11
-
-
67349140294
-
In vivo effects of a GPR30 antagonist
-
Dennis MK, Burai R, Ramesh C, Petrie WK, Alcon SN, et al. (2009) In vivo effects of a GPR30 antagonist. Nat Chem Biol 5: 421-427.
-
(2009)
Nat Chem Biol
, vol.5
, pp. 421-427
-
-
Dennis, M.K.1
Burai, R.2
Ramesh, C.3
Petrie, W.K.4
Alcon, S.N.5
-
12
-
-
81255160989
-
Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity
-
Dennis MK, Field AS, Burai R, Ramesh C, Petrie WK, et al. (2011) Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity. J Steroid Biochem Mol Biol 127: 358-366.
-
(2011)
J Steroid Biochem Mol Biol
, vol.127
, pp. 358-366
-
-
Dennis, M.K.1
Field, A.S.2
Burai, R.3
Ramesh, C.4
Petrie, W.K.5
-
13
-
-
67650308267
-
A crowdsourcing evaluation of the NIH chemical probes
-
Oprea TI, Bologa CG, Boyer S, Curpan RF, Glen RC, et al. (2009) A crowdsourcing evaluation of the NIH chemical probes. Nature Chem Biol 5: 441-447.
-
(2009)
Nature Chem Biol
, vol.5
, pp. 441-447
-
-
Oprea, T.I.1
Bologa, C.G.2
Boyer, S.3
Curpan, R.F.4
Glen, R.C.5
-
14
-
-
77249119272
-
Synthesis and characterization of iodinated tetrahydroquinolines targeting the G protein-coupled estrogen receptor GPR30
-
Ramesh C, Nayak TK, Burai R, Dennis MK, Hathaway HJ, et al. (2010) Synthesis and characterization of iodinated tetrahydroquinolines targeting the G protein-coupled estrogen receptor GPR30. J Med Chem 53: 1004-14.
-
(2010)
J Med Chem
, vol.53
, pp. 1004-1014
-
-
Ramesh, C.1
Nayak, T.K.2
Burai, R.3
Dennis, M.K.4
Hathaway, H.J.5
-
15
-
-
77955014125
-
Influence of charge on cell permeability and tumor imaging of GPR30-targeted 111In-labeled non-steroidal imaging agents
-
Nayak TK, Dennis MK, Ramesh C, Burai R, Atcher RW, et al. (2010) Influence of charge on cell permeability and tumor imaging of GPR30-targeted 111In-labeled non-steroidal imaging agents. ACS Chem Biol 5: 681-90.
-
(2010)
ACS Chem Biol
, vol.5
, pp. 681-690
-
-
Nayak, T.K.1
Dennis, M.K.2
Ramesh, C.3
Burai, R.4
Atcher, R.W.5
-
16
-
-
35348857513
-
Synthetic estrogen derivatives demonstrate the functionality of intracellular GPR30
-
Revankar CM, Mitchell HD, Field AS, Burai R, Corona C, et al. (2007) Synthetic estrogen derivatives demonstrate the functionality of intracellular GPR30. ACS Chem Biol 2: 536-44.
-
(2007)
ACS Chem Biol
, vol.2
, pp. 536-544
-
-
Revankar, C.M.1
Mitchell, H.D.2
Field, A.S.3
Burai, R.4
Corona, C.5
-
17
-
-
79959347634
-
Down-modulation of the G-protein-coupled estrogen receptor, GPER, from the cell surface occurs via a trans-golgi-proteasome pathway
-
Chen SB, Quinn JA, Graeber CT, Filardo EJ, (2011) Down-modulation of the G-protein-coupled estrogen receptor, GPER, from the cell surface occurs via a trans-golgi-proteasome pathway. J Biol Chem 286 (25): 22441-22455.
-
(2011)
J Biol Chem
, vol.286
, Issue.25
, pp. 22441-22455
-
-
Chen, S.B.1
Quinn, J.A.2
Graeber, C.T.3
Filardo, E.J.4
-
18
-
-
77952482481
-
Technetium and gallium derived radiopharmaceuticals: comparing and contrasting the chemistry of two important radiometals for the molecular imaging era
-
Bartholomä MD, Louie AS, Valliant JF, Zubieta J, (2010) Technetium and gallium derived radiopharmaceuticals: comparing and contrasting the chemistry of two important radiometals for the molecular imaging era. Chem Rev 110 (5): 2903-20.
-
(2010)
Chem Rev
, vol.110
, Issue.5
, pp. 2903-2920
-
-
Bartholomä, M.D.1
Louie, A.S.2
Valliant, J.F.3
Zubieta, J.4
-
19
-
-
0034836075
-
Synthesis and properties of boranocarbonate: a convenient in situ CO source for the aqueous preparation of [99mTc(OH2)3(CO)3]-
-
Alberto R, Ortner K, Wheatley N, Schibli R, Schubiger AP, (2001) Synthesis and properties of boranocarbonate: a convenient in situ CO source for the aqueous preparation of [99mTc(OH2)3(CO)3]-. J Am Chem Soc 123 (13): 3135-3136.
-
(2001)
J Am Chem Soc
, vol.123
, Issue.13
, pp. 3135-3136
-
-
Alberto, R.1
Ortner, K.2
Wheatley, N.3
Schibli, R.4
Schubiger, A.P.5
-
20
-
-
77951119518
-
Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs
-
Burai R, Ramesh C, Shorty M, Curpan R, Bologa C, et al. (2010) Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs. Org Biomol Chem 8: 2252-9.
-
(2010)
Org Biomol Chem
, vol.8
, pp. 2252-2259
-
-
Burai, R.1
Ramesh, C.2
Shorty, M.3
Curpan, R.4
Bologa, C.5
-
21
-
-
33751004697
-
Linkage effects on binding affinity and activation of GPR30 and estrogen receptors ERalpha/beta with tridentate pyridin-2-yl hydrazine tricarbonyl-Re/(99m)Tc(I) chelates
-
Ramesh C, Bryant BJ, Nayak TK, Revankar CM, Anderson T, et al. (2006) Linkage effects on binding affinity and activation of GPR30 and estrogen receptors ERalpha/beta with tridentate pyridin-2-yl hydrazine tricarbonyl-Re/(99m)Tc(I) chelates. J Am Chem Soc 128: 14476-7.
-
(2006)
J Am Chem Soc
, vol.128
, pp. 14476-14477
-
-
Ramesh, C.1
Bryant, B.J.2
Nayak, T.K.3
Revankar, C.M.4
Anderson, T.5
-
22
-
-
44849115355
-
Preclinical development of a neutral, estrogen receptor-targeted, tridentate 99mTc(I)-estradiol-pyridin-2-yl hydrazine derivative for imaging of breast and endometrial cancers
-
Nayak TK, Hathaway HJ, Ramesh C, Arterburn JB, Dai D, et al. (2008) Preclinical development of a neutral, estrogen receptor-targeted, tridentate 99mTc(I)-estradiol-pyridin-2-yl hydrazine derivative for imaging of breast and endometrial cancers. J Nucl Med 49: 978-86.
-
(2008)
J Nucl Med
, vol.49
, pp. 978-986
-
-
Nayak, T.K.1
Hathaway, H.J.2
Ramesh, C.3
Arterburn, J.B.4
Dai, D.5
-
23
-
-
58849105986
-
Single amino acid chelates (SAAC): a strategy for the diesign of technetium and rhenium radiopharmaceuticals
-
Bartholomä M, Valliant J, Maresca KP, Babich J, Zubieta J, (2009) Single amino acid chelates (SAAC): a strategy for the diesign of technetium and rhenium radiopharmaceuticals. Chem Commun 7 (5): 493-512.
-
(2009)
Chem Commun
, vol.7
, Issue.5
, pp. 493-512
-
-
Bartholomä, M.1
Valliant, J.2
Maresca, K.P.3
Babich, J.4
Zubieta, J.5
-
24
-
-
77953773495
-
Evaluation of Re and (99m)Tc complexes of 2-(4′-aminophenyl)benzothiazole as potential breast cancer radiopharmaceuticals
-
Tzanopoulou S, Sagnou M, Paravatou-Petsotas M, Gourni E, Loudos G, et al. (2010) Evaluation of Re and (99m)Tc complexes of 2-(4′-aminophenyl)benzothiazole as potential breast cancer radiopharmaceuticals. J Med Chem 53 (12): 4633-4641.
-
(2010)
J Med Chem
, vol.53
, Issue.12
, pp. 4633-4641
-
-
Tzanopoulou, S.1
Sagnou, M.2
Paravatou-Petsotas, M.3
Gourni, E.4
Loudos, G.5
-
25
-
-
33845187817
-
"Click to chelate": synthesis and installation of metal chelates into biomolecules in a single step
-
Mindt TL, Struthers H, Brans L, Anguelov T, Schweinsberg C, et al. (2006) "Click to chelate": synthesis and installation of metal chelates into biomolecules in a single step. J Am Chem Soc 128 (47): 15096-15097.
-
(2006)
J Am Chem Soc
, vol.128
, Issue.47
, pp. 15096-15097
-
-
Mindt, T.L.1
Struthers, H.2
Brans, L.3
Anguelov, T.4
Schweinsberg, C.5
-
26
-
-
52449087056
-
"Click-to-Chelate": Design and Incorporation of Triazole-Containing Metal-Chelating Systems into Biomolecules of Diagnostic and Therapeutic Interest
-
Struthers H, Spingler B, Mindt TL, Schibli R, (2008) "Click-to-Chelate": Design and Incorporation of Triazole-Containing Metal-Chelating Systems into Biomolecules of Diagnostic and Therapeutic Interest. Chem Eur J 14 (20): 6173-83.
-
(2008)
Chem Eur J
, vol.14
, Issue.20
, pp. 6173-6183
-
-
Struthers, H.1
Spingler, B.2
Mindt, T.L.3
Schibli, R.4
-
27
-
-
33745262314
-
Rapid microwave assisted hydration of internal arylalkynes in the presence of PTSA: an efficient regioselective access to carbonyl compounds
-
Le Bras G, Provot O, Peyrat J-F, Alami M, Brion J-D, (2006) Rapid microwave assisted hydration of internal arylalkynes in the presence of PTSA: an efficient regioselective access to carbonyl compounds. Tetrahedron Lett 47 (31): 5497-5501.
-
(2006)
Tetrahedron Lett
, vol.47
, Issue.31
, pp. 5497-5501
-
-
Le Bras, G.1
Provot, O.2
Peyrat, J.-F.3
Alami, M.4
Brion, J.-D.5
-
28
-
-
0037047536
-
Highly Active Oxime-Derived Palladacycle Complexes for Suzuki-Miyaura and Ullmann-Type Coupling Reactions
-
Alonso DA, Najera C, Pacheco MC, (2002) Highly Active Oxime-Derived Palladacycle Complexes for Suzuki-Miyaura and Ullmann-Type Coupling Reactions. J Org Chem 2002 67: 5588-5594.
-
(2002)
J Org Chem 2002
, vol.67
, pp. 5588-5594
-
-
Alonso, D.A.1
Najera, C.2
Pacheco, M.C.3
-
29
-
-
1942436087
-
Synthesis of aryl azides and vinyl azides via proline-promoted CuI-catalyzed coupling reactions
-
Zhu W, Ma D, (2004) Synthesis of aryl azides and vinyl azides via proline-promoted CuI-catalyzed coupling reactions. Chem Commun (7) pp. 888-889.
-
(2004)
Chem Commun
, Issue.7
, pp. 888-889
-
-
Zhu, W.1
Ma, D.2
-
30
-
-
14844343093
-
A transmembrane intracellular estrogen receptor mediates rapid cell signaling
-
Revankar CM, Cimino DF, Sklar LA, Arterburn JB, Prossnitz ER, (2005) A transmembrane intracellular estrogen receptor mediates rapid cell signaling. Science 11 (3): 1625-1630.
-
(2005)
Science
, vol.11
, Issue.3
, pp. 1625-1630
-
-
Revankar, C.M.1
Cimino, D.F.2
Sklar, L.A.3
Arterburn, J.B.4
Prossnitz, E.R.5
|