Discovery of novel haloalkane dehalogenase inhibitors

Applied and Environmental Microbiology

Volumn 82, Issue 6, 2016, Pages 1958-1965

  Buryska, Tomas ^a,b   Daniel, Lukas ^a,b   Kunka, Antonin ^a   Brezovsky, Jan ^a,b   Damborsky, Jiri ^a,b   Prokop, Zbynek ^a,b  

^a MASARYK UNIVERSITY   (Czech Republic)

^b ST ANNE S UNIVERSITY HOSPITAL   (Czech Republic)

Author keywords

[No Author keywords available]

Indexed keywords

BACTERIA; ENZYMES; PATHOGENS; VIRTUAL REALITY;

HIGH SPECIFICITY; INHIBITION CONSTANTS; MOLECULAR ARCHITECTURE; MYCOBACTERIUM TUBERCULOSIS; NATURAL FUNCTIONS; POTENTIAL INHIBITORS; TARGET STRUCTURE; VIRTUAL SCREENING; MOLECULAR PROBES;

CRYSTAL STRUCTURE;

BACTERIAL DISEASE; BACTERIUM; ENZYME; INHIBITOR; MOLECULAR ANALYSIS; PATHOGEN; PATHOGENICITY; PROBE;

MYCOBACTERIUM TUBERCULOSIS; MYCOBACTERIUM TUBERCULOSIS H37RV;

ENZYME INHIBITOR; HALOALKANE DEHALOGENASE; HYDROLASE;

ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; ENZYMOLOGY; ISOLATION AND PURIFICATION; METABOLISM; MOLECULAR DYNAMICS; MOLECULAR MODEL; MYCOBACTERIUM TUBERCULOSIS; PROTEIN CONFORMATION;

ENZYME INHIBITORS; HYDROLASES; MODELS, MOLECULAR; MOLECULAR DYNAMICS SIMULATION; MOLECULAR STRUCTURE; MYCOBACTERIUM TUBERCULOSIS; PROTEIN CONFORMATION;

EID: 84961279110     PISSN: 00992240     EISSN: 10985336     Source Type: Journal    
DOI: 10.1128/AEM.03916-15     Document Type: Article

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