메뉴 건너뛰기




Volumn 83, Issue , 2016, Pages 19-27

Fundamental understanding of drug absorption from a parenteral oil depot

Author keywords

Absorbance; Benzyl alcohol; Nandrolone; Oil depots; Pharmacokinetics

Indexed keywords

BENZYL ALCOHOL; HALOPERIDOL DECANOATE; NANDROLONE DECANOATE; NANDROLONE PHENPROPIONATE; OIL; PRODRUG; ANDROGEN; DRUG DOSAGE FORM; NANDROLONE; SESAME SEED OIL;

EID: 84950258562     PISSN: 09280987     EISSN: 18790720     Source Type: Journal    
DOI: 10.1016/j.ejps.2015.12.011     Document Type: Article
Times cited : (22)

References (38)
  • 1
    • 84929309802 scopus 로고    scopus 로고
    • Setup and validation of shake-flask procedures for the determination of partition coefficients (logD) from low drug amounts
    • A. Andrés, M. Rosés, C. Ràfols, E. Bosch, S. Espinosa, V. Segarra, and J.M. Huerta Setup and validation of shake-flask procedures for the determination of partition coefficients (logD) from low drug amounts Eur. J. Pharm. Sci. 76 2015 181 191 10.1016/j.ejps.2015.05.008
    • (2015) Eur. J. Pharm. Sci. , vol.76 , pp. 181-191
    • Andrés, A.1    Rosés, M.2    Ràfols, C.3    Bosch, E.4    Espinosa, S.5    Segarra, V.6    Huerta, J.M.7
  • 2
    • 0015868690 scopus 로고
    • Lymph flow and lymph protein concentration in the skin and muscle of the rabbit hind limb
    • C. Bach, and G.P. Lewis Lymph flow and lymph protein concentration in the skin and muscle of the rabbit hind limb J. Physiol. 235 1973 477 492
    • (1973) J. Physiol. , vol.235 , pp. 477-492
    • Bach, C.1    Lewis, G.P.2
  • 3
    • 18844391997 scopus 로고    scopus 로고
    • Pharmacokinetic evaluation of three different intramuscular doses of nandrolone decanoate: Analysis of serum and urine samples in healthy men
    • W.M. Bagchus, J.M.W. Smeets, H.A.M. Verheul, S.M. De Jager-Van Der Veen, A. Port, and T.B.P. Geurts Pharmacokinetic evaluation of three different intramuscular doses of nandrolone decanoate: analysis of serum and urine samples in healthy men J. Clin. Endocrinol. Metab. 90 2005 2624 2630 10.1210/jc.2004-1526
    • (2005) J. Clin. Endocrinol. Metab. , vol.90 , pp. 2624-2630
    • Bagchus, W.M.1    Smeets, J.M.W.2    Verheul, H.A.M.3    De Jager-Van Der Veen, S.M.4    Port, A.5    Geurts, T.B.P.6
  • 6
    • 0030697177 scopus 로고    scopus 로고
    • Lymph flow dynamics in exercising human skeletal muscle as detected by scintography
    • E. Havas, T. Parviainen, J. Vuorela, J. Toivanen, T. Nikula, and V. Vihko Lymph flow dynamics in exercising human skeletal muscle as detected by scintography J. Physiol. 504 1997 233 239 10.1111/j.1469-7793.1997.233bf.x
    • (1997) J. Physiol. , vol.504 , pp. 233-239
    • Havas, E.1    Parviainen, T.2    Vuorela, J.3    Toivanen, J.4    Nikula, T.5    Vihko, V.6
  • 8
    • 0021843298 scopus 로고
    • Clinical pharmacokinetics of the depot antipsychotics
    • M.W. Jann, L. Ereshefsky, and S.R. Saklad Clinical pharmacokinetics of the depot antipsychotics Clin. Pharmacokinet. 10 1985 315 333 10.2165/00003088-198510040-00003
    • (1985) Clin. Pharmacokinet. , vol.10 , pp. 315-333
    • Jann, M.W.1    Ereshefsky, L.2    Saklad, S.R.3
  • 9
    • 0026537290 scopus 로고
    • Influence of the injection volume on the release pattern of intramuscularly administered propranolol to rats
    • F. Kadir, C.B.J. Seijsener, and J. Zuidema Influence of the injection volume on the release pattern of intramuscularly administered propranolol to rats Int. J. Pharm. 81 1992 193 198 10.1016/0378-5173(92)90011-P
    • (1992) Int. J. Pharm. , vol.81 , pp. 193-198
    • Kadir, F.1    Seijsener, C.B.J.2    Zuidema, J.3
  • 10
    • 0025200456 scopus 로고
    • Drug lipophilicity and release pattern of some β-blocking agents after intra-adipose injection in pigs
    • F. Kadir, J. Zuidema, A. Pijpers, A. Vulto, and J.H.M. Verheijden Drug lipophilicity and release pattern of some β-blocking agents after intra-adipose injection in pigs Int. J. Pharm. 64 1990 171 180 10.1016/0378-5173(90)90266-7
    • (1990) Int. J. Pharm. , vol.64 , pp. 171-180
    • Kadir, F.1    Zuidema, J.2    Pijpers, A.3    Vulto, A.4    Verheijden, J.H.M.5
  • 11
    • 0033392246 scopus 로고    scopus 로고
    • Pharmacokinetics of haloperidol: An update
    • S. Kudo, and T. Ishizaki Pharmacokinetics of haloperidol: an update Clin. Pharmacokinet. 37 1999 435 456
    • (1999) Clin. Pharmacokinet. , vol.37 , pp. 435-456
    • Kudo, S.1    Ishizaki, T.2
  • 12
    • 33750694953 scopus 로고    scopus 로고
    • In vitro assessment of drug release rates from oil depot formulations intended for intra-articular administration
    • S.W. Larsen, J. Østergaard, H. Friberg-Johansen, M.N.B. Jessen, and C. Larsen In vitro assessment of drug release rates from oil depot formulations intended for intra-articular administration Eur. J. Pharm. Sci. 29 2006 348 354 10.1016/j.ejps.2006.07.002
    • (2006) Eur. J. Pharm. Sci. , vol.29 , pp. 348-354
    • Larsen, S.W.1    Østergaard, J.2    Friberg-Johansen, H.3    Jessen, M.N.B.4    Larsen, C.5
  • 13
    • 0030924263 scopus 로고    scopus 로고
    • Pharmacokinetics and pharmacodynamics of nandrolone esters in oil vehicle: Effects of ester, injection site and injection volume
    • C.F. Minto, C. Howe, S. Wishart, A.J. Conway, and D.J. Handelsman Pharmacokinetics and pharmacodynamics of nandrolone esters in oil vehicle: effects of ester, injection site and injection volume J. Pharmacol. Exp. Ther. 281 1997 93 102
    • (1997) J. Pharmacol. Exp. Ther. , vol.281 , pp. 93-102
    • Minto, C.F.1    Howe, C.2    Wishart, S.3    Conway, A.J.4    Handelsman, D.J.5
  • 15
    • 55549147133 scopus 로고    scopus 로고
    • Long acting testosterone undecanoate therapy in men with hypogonadism: Results of a pharmacokinetic clinical study
    • A. Morgentaler, A.S. Dobs, J.M. Kaufman, M.M. Miner, R. Shabsigh, R.S. Swerdloff, and C. Wang Long acting testosterone undecanoate therapy in men with hypogonadism: results of a pharmacokinetic clinical study J. Urol. 180 2008 2307 2313 10.1016/j.juro.2008.08.126
    • (2008) J. Urol. , vol.180 , pp. 2307-2313
    • Morgentaler, A.1    Dobs, A.S.2    Kaufman, J.M.3    Miner, M.M.4    Shabsigh, R.5    Swerdloff, R.S.6    Wang, C.7
  • 18
    • 0019247209 scopus 로고
    • Intrinsic contractility of prenodal lymph vessels and lymph flow in human leg
    • W.L. Olszewski, and A. Engeset Intrinsic contractility of prenodal lymph vessels and lymph flow in human leg Am. J. Physiol. 239 1980 H775 H783
    • (1980) Am. J. Physiol. , vol.239 , pp. H775-H783
    • Olszewski, W.L.1    Engeset, A.2
  • 20
    • 0034020054 scopus 로고    scopus 로고
    • Lymphatic transport of proteins after subcutaneous administration
    • C.J.H. Porter, and S.A. Charman Lymphatic transport of proteins after subcutaneous administration J. Pharm. Sci. 89 2000 297 310 10.1002/(SICI)1520-6017(200003)89:3<297::AID-JPS2>3.0.CO;2-P
    • (2000) J. Pharm. Sci. , vol.89 , pp. 297-310
    • Porter, C.J.H.1    Charman, S.A.2
  • 21
    • 33847394968 scopus 로고    scopus 로고
    • Lipids and lipid-based formulations: Optimizing the oral delivery of lipophilic drugs
    • C.J.H. Porter, N.L. Trevaskis, and W.N. Charman Lipids and lipid-based formulations: optimizing the oral delivery of lipophilic drugs Nat. Rev. Drug Discov. 6 2007 231 248 10.1038/nrd2197
    • (2007) Nat. Rev. Drug Discov. , vol.6 , pp. 231-248
    • Porter, C.J.H.1    Trevaskis, N.L.2    Charman, W.N.3
  • 22
    • 0028246255 scopus 로고
    • Limits to steady-state lymph flow rates derived from plasma-to-tissue uptake measurements
    • E. Renkin, and H. Wiig Limits to steady-state lymph flow rates derived from plasma-to-tissue uptake measurements Microvasc. Res. 47 1994 318 328
    • (1994) Microvasc. Res. , vol.47 , pp. 318-328
    • Renkin, E.1    Wiig, H.2
  • 23
    • 0027474901 scopus 로고
    • Subarachnoid local anesthetic block does not affect morphine absorption from paired intramuscular and subcutaneous injection sites in the elderly patient
    • A. Ronald, D. Docherty, J. Broom, and W. Chambers Subarachnoid local anesthetic block does not affect morphine absorption from paired intramuscular and subcutaneous injection sites in the elderly patient Anesth. Analg. 76 1993 778 782 10.1213/00000539-199304000-00016
    • (1993) Anesth. Analg. , vol.76 , pp. 778-782
    • Ronald, A.1    Docherty, D.2    Broom, J.3    Chambers, W.4
  • 25
    • 0023786760 scopus 로고
    • Plasma levels of fluphenazine decanoate: Effects of site of injection, massage and muscle activity
    • S.M. Soni, D. Wiles, A.A. Schiff, and J.S. Bamrah Plasma levels of fluphenazine decanoate: effects of site of injection, massage and muscle activity Br. J. Psychiatry 153 1988 382 384 10.1192/bjp.153.3.382
    • (1988) Br. J. Psychiatry , vol.153 , pp. 382-384
    • Soni, S.M.1    Wiles, D.2    Schiff, A.A.3    Bamrah, J.S.4
  • 26
    • 35148812430 scopus 로고    scopus 로고
    • Interstitial flow and its effects in soft tissues
    • M.A. Swartz, and M.E. Fleury Interstitial flow and its effects in soft tissues Annu. Rev. Biomed. Eng. 9 2007 229 256 10.1146/annurev.bioeng.9.060906.151850
    • (2007) Annu. Rev. Biomed. Eng. , vol.9 , pp. 229-256
    • Swartz, M.A.1    Fleury, M.E.2
  • 28
    • 84855795838 scopus 로고    scopus 로고
    • In vitro release from oil injectables for intra-articular administration: Importance of interfacial area, diffusivity and partitioning
    • M. Thing, C. Larsen, J. Østergaard, H. Jensen, and S.W. Larsen In vitro release from oil injectables for intra-articular administration: importance of interfacial area, diffusivity and partitioning Eur. J. Pharm. Sci. 45 2012 351 357 10.1016/j.ejps.2011.12.006
    • (2012) Eur. J. Pharm. Sci. , vol.45 , pp. 351-357
    • Thing, M.1    Larsen, C.2    Østergaard, J.3    Jensen, H.4    Larsen, S.W.5
  • 29
    • 0014837290 scopus 로고
    • Model studies in vitro with long-acting hormonal preparations
    • J. Van Der Vies Model studies in vitro with long-acting hormonal preparations Acta Endocrinol. (Copenh) 64 1970 656 669 10.1530/acta.0.0640656
    • (1970) Acta Endocrinol. (Copenh) , vol.64 , pp. 656-669
    • Van Der Vies, J.1
  • 30
    • 34249768667 scopus 로고
    • Comparative bioavailability study of two haloperidol decanoate containing products
    • G. Van Weringh, B.J. Komen, R.E. Thieme, R.T.M. van der Hoeven, and T. Vos Comparative bioavailability study of two haloperidol decanoate containing products Pharm. World Sci. 16 1994 343 347 10.1007/BF02178564
    • (1994) Pharm. World Sci. , vol.16 , pp. 343-347
    • Van Weringh, G.1    Komen, B.J.2    Thieme, R.E.3    Van Der Hoeven, R.T.M.4    Vos, T.5
  • 31
    • 0016713944 scopus 로고
    • Sex differences in the intramuscular absorption and bioavailability of cephradine
    • R.A. Vukovich, L.J. Brannick, A.A. Sugerman, and E.S. Neiss Sex differences in the intramuscular absorption and bioavailability of cephradine Clin. Pharmacol. Ther. 18 1975 215 220
    • (1975) Clin. Pharmacol. Ther. , vol.18 , pp. 215-220
    • Vukovich, R.A.1    Brannick, L.J.2    Sugerman, A.A.3    Neiss, E.S.4
  • 32
    • 0016356405 scopus 로고
    • Application of the Wagner-Nelson absorption method to the two-compartment open model
    • J.G. Wagner Application of the Wagner-Nelson absorption method to the two-compartment open model J. Pharmacokinet. Biopharm. 2 1974 469 486 10.1007/BF01070942
    • (1974) J. Pharmacokinet. Biopharm. , vol.2 , pp. 469-486
    • Wagner, J.G.1
  • 33
    • 72949121224 scopus 로고    scopus 로고
    • Critical factors influencing the in vivo performance of long-acting lipophilic solutions - Impact on in vitro release method design
    • S. Weng Larsen, and C. Larsen Critical factors influencing the in vivo performance of long-acting lipophilic solutions - impact on in vitro release method design AAPS J. 11 2009 762 770 10.1208/s12248-009-9153-9
    • (2009) AAPS J. , vol.11 , pp. 762-770
    • Weng Larsen, S.1    Larsen, C.2
  • 34
    • 0033306851 scopus 로고    scopus 로고
    • The effect of pharmacokinetically guided acute intravenous testosterone administration on electrocardiographic and blood pressure variables
    • C.M. White, M.J. Ferraro-Borgida, N.M. Moyna, C.C. McGill, A.W. Ahlberg, P.D. Thompson, and G.V. Heller The effect of pharmacokinetically guided acute intravenous testosterone administration on electrocardiographic and blood pressure variables J. Clin. Pharmacol. 39 1999 1038 1043 10.1177/00912709922011809
    • (1999) J. Clin. Pharmacol. , vol.39 , pp. 1038-1043
    • White, C.M.1    Ferraro-Borgida, M.J.2    Moyna, N.M.3    McGill, C.C.4    Ahlberg, A.W.5    Thompson, P.D.6    Heller, G.V.7
  • 35
    • 0022203791 scopus 로고
    • Pharmacokinetic parameters of nandrolone (19-nortestosterone) after intramuscular administration of nandrolone decanoate (Deca-Durabolin) to healthy volunteers
    • H.P. Wijnand, A.M. Bosch, and C.W. Donker Pharmacokinetic parameters of nandrolone (19-nortestosterone) after intramuscular administration of nandrolone decanoate (Deca-Durabolin) to healthy volunteers Acta Endocrinol. Suppl. (Copenh) 271 1985 19 30 10.1530/acta.0.109S00019
    • (1985) Acta Endocrinol. Suppl. (Copenh) , vol.271 , pp. 19-30
    • Wijnand, H.P.1    Bosch, A.M.2    Donker, C.W.3
  • 36
    • 79956119127 scopus 로고    scopus 로고
    • Flip-flop pharmacokinetics - Delivering a reversal of disposition: Challenges and opportunities during drug development
    • J.A. Yáñez, C.M. Remsberg, C.L. Sayre, M.L. Forrest, and N.M. Davies Flip-flop pharmacokinetics - delivering a reversal of disposition: challenges and opportunities during drug development Ther. Deliv. 2 2011 643 672 10.4155/tde.11.19
    • (2011) Ther. Deliv. , vol.2 , pp. 643-672
    • Yáñez, J.A.1    Remsberg, C.M.2    Sayre, C.L.3    Forrest, M.L.4    Davies, N.M.5
  • 37
    • 0028299106 scopus 로고
    • Release and absorption rates of intramuscularly and subcutaneously injected pharmaceuticals (II)
    • J. Zuidema, F. Kadir, H.A.C. Titulaer, and C. Oussoren Release and absorption rates of intramuscularly and subcutaneously injected pharmaceuticals (II) Int. J. Pharm. 105 1994 189 207 10.1016/0378-5173(94)90103-1
    • (1994) Int. J. Pharm. , vol.105 , pp. 189-207
    • Zuidema, J.1    Kadir, F.2    Titulaer, H.A.C.3    Oussoren, C.4
  • 38
    • 0023804439 scopus 로고
    • Release and absorption rate aspects of intramuscularly injected pharmaceuticals
    • J. Zuidema, F.A.J.M. Pieters, and G.S.M.J.E. Duchateau Release and absorption rate aspects of intramuscularly injected pharmaceuticals Int. J. Pharm. 47 1988 1 12 10.1016/0378-5173(88)90209-8
    • (1988) Int. J. Pharm. , vol.47 , pp. 1-12
    • Zuidema, J.1    Pieters, F.A.J.M.2    Duchateau, G.S.M.J.E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.