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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 16, 2015, Pages 3189-3193

Discovery of potent, selective small molecule inhibitors of α-subtype of type III phosphatidylinositol-4-kinase (PI4KIIIα)

(7) Raubo, Piotr a Andrews, David M a McKelvie, Jennifer C b Robb, Graeme R a Smith, James M a,c Swarbrick, Martin E c Waring, Michael J a

a ASTRAZENECA (United Kingdom)

b ROYAL VETERINARY COLLEGE (United Kingdom)

c Cancer Research UK (United Kingdom)

Author keywords

In vitro tools; IP1; Oncology; PI4K

Indexed keywords

ENZYME INHIBITOR; PHOSPHATIDYLINOSITOL KINASE; PLATELET DERIVED GROWTH FACTOR; INOSITOL PHOSPHATE; MOLECULAR LIBRARY; PHOSPHATIDYLINOSITOL PHOSPHATE 4-KINASE; PHOSPHOTRANSFERASE;

ANIMAL CELL; ARTICLE; CANCER CELL LINE; CELL ACTIVITY; CELL LEVEL; DRUG POTENCY; GROWTH INHIBITION; IN VITRO STUDY; MOUSE; NONHUMAN; STRUCTURE ACTIVITY RELATION; SUZUKI REACTION; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; DRUG DESIGN; DRUG EFFECTS; HIGH THROUGHPUT SCREENING; HUMAN; METABOLISM; MOLECULAR LIBRARY; SIGNAL TRANSDUCTION; SYNTHESIS;

DRUG DESIGN; ENZYME INHIBITORS; HIGH-THROUGHPUT SCREENING ASSAYS; HUMANS; INOSITOL PHOSPHATES; MODELS, MOLECULAR; PHOSPHOTRANSFERASES (ALCOHOL GROUP ACCEPTOR); PLATELET-DERIVED GROWTH FACTOR; SIGNAL TRANSDUCTION; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84934872663 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2015.05.093 Document Type: Article

Times cited : (11)

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