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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 16, 2015, Pages 3285-3289

Synthesis of novel derivatives of oxindole, their urease inhibition and molecular docking studies

(10) Taha, Muhammad a,b Ismail, Nor Hadiani a,b Khan, Ajmal c Shah, Syed Adnan Ali a Anwar, Ammarah d Halim, Sobia Ahsan e Fatmi, M Qaiser d Imran, Syahrul a,b Rahim, Fazal f Khan, Khalid Mohammed g

a UNIVERSITI TEKNOLOGI MARA (Malaysia)

b Faculty of Civil Engineering (UiTM) (Malaysia)

c COMSATS Institute of Information Technology ^* (Pakistan)

d Universiti Teknologi MARA Puncak Alam ^* (Pakistan)

e UNIVERSITY OF THE PUNJAB (Pakistan)

f HAZARA UNIVERSITY (Pakistan)

g UNIVERSITY OF KARACHI (Pakistan)

Author keywords

Docking studies; Novel derivatives; Oxindole; Urease activity

Indexed keywords

6 CHLOROOXINDOLE; ACETOHYDROXAMIC ACID; ACETOPHENONE DERIVATIVE; ALDEHYDE DERIVATIVE; CARBON 13; INDOLE DERIVATIVE; OXINDOLE; OXINDOLE DERIVATIVE; PROTON; THIOUREA; UNCLASSIFIED DRUG; UREASE; UREASE INHIBITOR; BENZAMIDE DERIVATIVE; HYDRAZINE DERIVATIVE;

ARTICLE; BINDING SITE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; ELECTROSPRAY MASS SPECTROMETRY; HYDROGEN BOND; IC50; INFRARED SPECTROSCOPY; MOLECULAR DOCKING; MOLECULAR INTERACTION; PROTON NUCLEAR MAGNETIC RESONANCE; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECTS; ENZYME ACTIVATION; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SYNTHESIS;

BENZAMIDES; ENZYME ACTIVATION; HYDRAZINES; HYDROGEN BONDING; INDOLES; INHIBITORY CONCENTRATION 50; MAGNETIC RESONANCE SPECTROSCOPY; MOLECULAR DOCKING SIMULATION; MOLECULAR STRUCTURE; UREASE;

EID: 84934830620 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2015.05.069 Document Type: Article

Times cited : (77)

References (46)

1
- 0037377325
- A. Dermatakis, K.C. Luk, and W. DePinto Bioorg. Med. Chem. 13 2003 1873
- (2003) Bioorg. Med. Chem. , vol.13 , pp. 1873
- Dermatakis, A.¹ Luk, K.C.² DePinto, W.³

2
- 0035924185
- T. Tokunaga, W.E. Hume, T. Umezome, K. Okazaki, Y. Ueki, K. Kumagai, S. Hourai, J. Nagamine, H. Seki, M. Taiji, H. Noguchi, and R. Nagata J. Med. Chem. 44 2001 4641
- (2001) J. Med. Chem. , vol.44 , pp. 4641
- Tokunaga, T.¹ Hume, W.E.² Umezome, T.³ Okazaki, K.⁴ Ueki, Y.⁵ Kumagai, K.⁶ Hourai, S.⁷ Nagamine, J.⁸ Seki, H.⁹ Taiji, M.¹⁰ Noguchi, H.¹¹ Nagata, R.¹²

3
- 33845445111
- T. Kagata, S. Saito, H. Shigemori, A. Ohsaki, H. Ishiyama, T. Kubota, and J. Kobayashi J. Nat. Prod. 69 2006 1517
- (2006) J. Nat. Prod. , vol.69 , pp. 1517
- Kagata, T.¹ Saito, S.² Shigemori, H.³ Ohsaki, A.⁴ Ishiyama, H.⁵ Kubota, T.⁶ Kobayashi, J.⁷

4
- 0034105791
- Y. Koguchi, J. Kohno, M. Nishio, K. Takahashi, T. Okuda, T. Ohnuki, and S. Komatsubara J. Antibiot. 53 2000 105
- (2000) J. Antibiot. , vol.53 , pp. 105
- Koguchi, Y.¹ Kohno, J.² Nishio, M.³ Takahashi, K.⁴ Okuda, T.⁵ Ohnuki, T.⁶ Komatsubara, S.⁷

5
- 2542609191
- N.T. Zaveri, F. Jiang, C.M. Olsen, J.R. Deschamps, D. Parrish, W. Polgar, and L. Toll J. Med. Chem. 47 2004 2973
- (2004) J. Med. Chem. , vol.47 , pp. 2973
- Zaveri, N.T.¹ Jiang, F.² Olsen, C.M.³ Deschamps, J.R.⁴ Parrish, D.⁵ Polgar, W.⁶ Toll, L.⁷

6
- 26444521686
- M. Alcaraz, S. Atkinson, P. Cornwall, A.C. Foster, D.M. Gill, L.A. Humphries, P.S. Keegan, R. Kemp, E. Merifield, R.A. Nixon, A.J. Noble, D. O'Beirne, Z.M. Patel, J. Perkins, P. Rowa, P. Sadler, J.T. Singleton, J. Tornos, A.J. Watts, and I.A. Woodland Org. Process Res. Dev. 9 2005 555
- (2005) Org. Process Res. Dev. , vol.9 , pp. 555
- Alcaraz, M.¹ Atkinson, S.² Cornwall, P.³ Foster, A.C.⁴ Gill, D.M.⁵ Humphries, L.A.⁶ Keegan, P.S.⁷ Kemp, R.⁸ Merifield, E.⁹ Nixon, R.A.¹⁰ Noble, A.J.¹¹ O'Beirne, D.¹² Patel, Z.M.¹³ Perkins, J.¹⁴ Rowa, P.¹⁵ Sadler, P.¹⁶ Singleton, J.T.¹⁷ Tornos, J.¹⁸ Watts, A.J.¹⁹ Woodland, I.A.²⁰ more..

7
- 0037119746
- C. Kikuchi, T. Hiranuma, and M. Koyama Bioorg. Med. Chem. Lett. 12 2002 2549
- (2002) Bioorg. Med. Chem. Lett. , vol.12 , pp. 2549
- Kikuchi, C.¹ Hiranuma, T.² Koyama, M.³

8
- 0022344784
- J.R. Gregory-Gallagher, G.Lavanchy Patricia, W.Wilson James, J.Paul Hieble, and M.DeMarinis Robert J. Med. Chem. 28 1985 1533
- (1985) J. Med. Chem. , vol.28 , pp. 1533
- Gregory-Gallagher, J.R.¹ Patricia, G.L.² James, W.W.³ Hieble, J.P.⁴ Robert, M.D.⁵

9
- 0028944619
- C.D. Smith, J.T. Zilfou, K. Stratmann, G.M. Patterson, and R.E. Moore Mol. Pharmacol. 47 1995 241
- (1995) Mol. Pharmacol. , vol.47 , pp. 241
- Smith, C.D.¹ Zilfou, J.T.² Stratmann, K.³ Patterson, G.M.⁴ Moore, R.E.⁵

10
- 0020686579
- H. Pajouhesh, R. Parson, and F.D. Popp J. Pharm. Sci. 72 1983 318
- (1983) J. Pharm. Sci. , vol.72 , pp. 318
- Pajouhesh, H.¹ Parson, R.² Popp, F.D.³

11
- 0024153330
- E. Moilanen, J. Alanko, M.Z. Asmawi, H. Vapaatalo, M.Z. Asmawi, E. Moilanen, J. Alanko, and H. Vapaatalo Eicosanoids 1 1988 35
- (1988) Eicosanoids , vol.1 , pp. 35
- Moilanen, E.¹ Alanko, J.² Asmawi, M.Z.³ Vapaatalo, H.⁴ Asmawi, M.Z.⁵ Moilanen, E.⁶ Alanko, J.⁷ Vapaatalo, H.⁸

12
- 0344333471
- M.J. Mokrosz, B. Duszyńska, S. Misztal, A. Kłodzińska, E. Tatarczyńska, E. Chojnacka-Wójcik, and M. Dziedzicka-Wasylewska Arch. Pharm. 331 1998 325
- (1998) Arch. Pharm. , vol.331 , pp. 325
- Mokrosz, M.J.¹ Duszyńska, B.² Misztal, S.³ Kłodzińska, A.⁴ Tatarczyńska, E.⁵ Chojnacka-Wójcik, E.⁶ Dziedzicka-Wasylewska, M.⁷

13
- 0017079032
- J.Kornet Milton, and P.Thio Alan J. Med. Chem. 19 1976 892
- (1976) J. Med. Chem. , vol.19 , pp. 892
- Milton, J.K.¹ Alan, P.T.²

14
- 84883413388
- K.M. Khan, M. Khan, N. Ambreen, M. Taha, F. Rahim, S. Rasheed, S. Saied, H. Shafi, S. Perveen, and M.I. Choudhary Med. Chem. 9 2013 681
- (2013) Med. Chem. , vol.9 , pp. 681
- Khan, K.M.¹ Khan, M.² Ambreen, N.³ Taha, M.⁴ Rahim, F.⁵ Rasheed, S.⁶ Saied, S.⁷ Shafi, H.⁸ Perveen, S.⁹ Choudhary, M.I.¹⁰

15
- 80755125969
- K.M. Khan, Z. Shah, V.U. Ahmad, M. Khan, M. Taha, F. Rahim, H. Jahun, S. Perveen, and M.i. Choudhary Med. Chem. 7 2011 572
- (2011) Med. Chem. , vol.7 , pp. 572
- Khan, K.M.¹ Shah, Z.² Ahmad, V.U.³ Khan, M.⁴ Taha, M.⁵ Rahim, F.⁶ Jahun, H.⁷ Perveen, S.⁸ Choudhary, M.I.⁹

16
- 84874827794
- S.G. Musharraf, A. Bibi, N. Shahid, M. Najam-ul-Haq, M. Khan, M. Taha, U.R. Mughal, and K.M. Khan Am. J. Anal. Chem. 3 2012 779
- (2012) Am. J. Anal. Chem. , vol.3 , pp. 779
- Musharraf, S.G.¹ Bibi, A.² Shahid, N.³ Najam-Ul-Haq, M.⁴ Khan, M.⁵ Taha, M.⁶ Mughal, U.R.⁷ Khan, K.M.⁸

17
- 71749117357
- K.M. Khan, M. Khan, M. Ali, M. Taha, S. Rasheed, S. Perveen, and M.I. Choudhary Bioorg. Med. Chem. 17 2009 7795
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 7795
- Khan, K.M.¹ Khan, M.² Ali, M.³ Taha, M.⁴ Rasheed, S.⁵ Perveen, S.⁶ Choudhary, M.I.⁷

18
- 0028920505
- P. Mishra, P.N. Gupta, A.K. Shakya, R. Shukla, and R.C. Srimal Indian J. Physiol. Pharmacol. 39 1995 169
- (1995) Indian J. Physiol. Pharmacol. , vol.39 , pp. 169
- Mishra, P.¹ Gupta, P.N.² Shakya, A.K.³ Shukla, R.⁴ Srimal, R.C.⁵

19
- 84890856883
- E.H. Anouar, S. Raweh, I. Bayach, M. Taha, M.S. Baharudin, F.D. Meo, M.H. Hasan, A. Adam, N.H. Ismail, J.F. Weber, and P. Trouillas J. Comput. Aided Mol. Des. 27 2013 951
- (2013) J. Comput. Aided Mol. Des. , vol.27 , pp. 951
- Anouar, E.H.¹ Raweh, S.² Bayach, I.³ Taha, M.⁴ Baharudin, M.S.⁵ Meo, F.D.⁶ Hasan, M.H.⁷ Adam, A.⁸ Ismail, N.H.⁹ Weber, J.F.¹⁰ Trouillas, P.¹¹

20
- 84885126789
- M. Taha, N.H. Ismail, W. Jamil, S. Yousuf, F.M. Jaafar, M.I. Ali, S.M. Kashif, and E. Hussain Molecules 18 2013 10912
- (2013) Molecules , vol.18 , pp. 10912
- Taha, M.¹ Ismail, N.H.² Jamil, W.³ Yousuf, S.⁴ Jaafar, F.M.⁵ Ali, M.I.⁶ Kashif, S.M.⁷ Hussain, E.⁸

21
- 84903316315
- A.N. Aziz, M. Taha, N.H. Ismail, E.H. Anouar, S. Yousuf, W. Jamil, K. Awang, N. Ahmat, K.M. Khan, and S.M. Kashif Molecules 19 2014 8414
- (2014) Molecules , vol.19 , pp. 8414
- Aziz, A.N.¹ Taha, M.² Ismail, N.H.³ Anouar, E.H.⁴ Yousuf, S.⁵ Jamil, W.⁶ Awang, K.⁷ Ahmat, N.⁸ Khan, K.M.⁹ Kashif, S.M.¹⁰

22
- 84863768768
- K.M. Khan, F. Muhammad Taha, S. Naz, S.Perveen Ali, and M. Iqbal Choudhary Med. Chem. 8 2012 705
- (2012) Med. Chem. , vol.8 , pp. 705
- Khan, K.M.¹ Muhammad Taha, F.² Naz, S.³ Ali, S.P.⁴ Iqbal Choudhary, M.⁵

23
- 84905161829
- M. Taha, N.H. Ismail, W. Jamil, H. Rashwan, S.M. Kashif, A.A. Sain, M.I. Adenan, E.H. Anouar, M. Ali, F. Rahim, and K.M. Khan Eur. J. Med. Chem. 84 2014 731
- (2014) Eur. J. Med. Chem. , vol.84 , pp. 731
- Taha, M.¹ Ismail, N.H.² Jamil, W.³ Rashwan, H.⁴ Kashif, S.M.⁵ Sain, A.A.⁶ Adenan, M.I.⁷ Anouar, E.H.⁸ Ali, M.⁹ Rahim, F.¹⁰ Khan, K.M.¹¹

24
- 84893040474
- M. Taha, H. Naz, S. Rasheed, N.H. Ismail, A.A. Rahman, S. Yousuf, and M.I. Choudhary Molecules 19 2014 1286
- (2014) Molecules , vol.19 , pp. 1286
- Taha, M.¹ Naz, H.² Rasheed, S.³ Ismail, N.H.⁴ Rahman, A.A.⁵ Yousuf, S.⁶ Choudhary, M.I.⁷

25
- 84879727205
- K.M. Khan, M. Taha, F. Rahim, M.I. Fakhri, W. Jamil, M. Khan, S. Rasheed, A. Karim, S. Perveen, and M.I. Choudhary J. Pak. Chem Soc. 35 2013 929
- (2013) J. Pak. Chem Soc. , vol.35 , pp. 929
- Khan, K.M.¹ Taha, M.² Rahim, F.³ Fakhri, M.I.⁴ Jamil, W.⁵ Khan, M.⁶ Rasheed, S.⁷ Karim, A.⁸ Perveen, S.⁹ Choudhary, M.I.¹⁰

26
- 84920848432
- M. Taha, N.H. Ismail, S. Lalani, M.Q. Fatmi, S. Siddiqui, K.M. Khan, S. Imran, and M.I. Choudhary Eur. J. Med. Chem. 92 2015 387
- (2015) Eur. J. Med. Chem. , vol.92 , pp. 387
- Taha, M.¹ Ismail, N.H.² Lalani, S.³ Fatmi, M.Q.⁴ Siddiqui, S.⁵ Khan, K.M.⁶ Imran, S.⁷ Choudhary, M.I.⁸

27
- 84877584824
- M. Taha, M.S. Baharudin, N.H. Ismail, K.M. Khan, F.M. Jaafar, Samreen, S. Siddiqui, and M.I. Choudhary Bioorg. Med. Chem. Lett. 23 2013 3463
- (2013) Bioorg. Med. Chem. Lett. , vol.23 , pp. 3463
- Taha, M.¹ Baharudin, M.S.² Ismail, N.H.³ Khan, K.M.⁴ Jaafar, F.M.⁵ Samreen⁶ Siddiqui, S.⁷ Choudhary, M.I.⁸

28
- 84934790140
- M. Taha, N.H. Ismail, M. Ali, K.M. Khan, W. Jamil, S.M. Kashif, and M. Asraf Med. Chem. Res. 23 2014 5282
- (2014) Med. Chem. Res. , vol.23 , pp. 5282
- Taha, M.¹ Ismail, N.H.² Ali, M.³ Khan, K.M.⁴ Jamil, W.⁵ Kashif, S.M.⁶ Asraf, M.⁷

29
- 33947332625
- M.W. Weatherburn Anal. Chem. 39 1967 971
- (1967) Anal. Chem. , vol.39 , pp. 971
- Weatherburn, M.W.¹

30
- 0019451279
- A. Martelli, P. Buli, and V. Cortecchia Eur. Urol. 7 1981 291
- (1981) Eur. Urol. , vol.7 , pp. 291
- Martelli, A.¹ Buli, P.² Cortecchia, V.³

31
- 0024514293
- H.L.T. Mobley, and R.P. Hausinger J. Microbiol. Rev. 53 1989 85
- (1989) J. Microbiol. Rev. , vol.53 , pp. 85
- Mobley, H.L.T.¹ Hausinger, R.P.²

32
- 77949425914
- M. Arfan, M. Ali, H. Ahmad, I. Anis, A. Khan, M.I. Choudhary, and M.R. Shah J. Enzyme Inhib. Med. Chem. 25 2010 296
- (2010) J. Enzyme Inhib. Med. Chem. , vol.25 , pp. 296
- Arfan, M.¹ Ali, M.² Ahmad, H.³ Anis, I.⁴ Khan, A.⁵ Choudhary, M.I.⁶ Shah, M.R.⁷

33
- 80054911088
- M.A.S. Aslam, S. Mahmood, M. Shahid, A. Saeed, and J.J. Iqbal Eur. J. Med. Chem. 46 2011 5473
- (2011) Eur. J. Med. Chem. , vol.46 , pp. 5473
- Aslam, M.A.S.¹ Mahmood, S.² Shahid, M.³ Saeed, A.⁴ Iqbal, J.J.⁵

34
- 84934852218
- M. Taha, N.H. Ismail, M.S. Baharudin, S. Lalani, S. Mehboob, K.M. Khan, S. Yousuf, S. Siddiqui, F. Rahim, and M.I. Choudhary Med. Chem. Res. 24 2015 1310
- (2015) Med. Chem. Res. , vol.24 , pp. 1310
- Taha, M.¹ Ismail, N.H.² Baharudin, M.S.³ Lalani, S.⁴ Mehboob, S.⁵ Khan, K.M.⁶ Yousuf, S.⁷ Siddiqui, S.⁸ Rahim, F.⁹ Choudhary, M.I.¹⁰

35
- 84874479720
- I. Anis, M. Aslam, N. Afza, A. Hussain, F.S. Ahmad, L. Iqbal, M. Lateef, M.T. Hussain, and T.H. Bokhari Int. J. Pharm. Chem. 2 2012 73
- (2012) Int. J. Pharm. Chem. , vol.2 , pp. 73
- Anis, I.¹ Aslam, M.² Afza, N.³ Hussain, A.⁴ Ahmad, F.S.⁵ Iqbal, L.⁶ Lateef, M.⁷ Hussain, M.T.⁸ Bokhari, T.H.⁹

36
- 84973405643
- S. Shujah, U.R. Zia, N. Muhammad, A. Shah, S. Ali, N. Khalid, and A. Meetsma J. Org. Chem. 2013 741
- (2013) J. Org. Chem. , pp. 741
- Shujah, S.¹ Zia, U.R.² Muhammad, N.³ Shah, A.⁴ Ali, S.⁵ Khalid, N.⁶ Meetsma, A.⁷

37
- 33747200808
- H. Alonso, A.A. Bliznyuk, and J.E. Gready Med. Res. Rev. 5 2006 531
- (2006) Med. Res. Rev. , vol.5 , pp. 531
- Alonso, H.¹ Bliznyuk, A.A.² Gready, J.E.³

38
- 84875066762
- A.M. Vijesha, A.M. Isloorb, T. Sandeep, T. Arulmolid, and K.F. Hoong Arab. J. Chem. 6 2013 197
- (2013) Arab. J. Chem. , vol.6 , pp. 197
- Vijesha, A.M.¹ Isloorb, A.M.² Sandeep, T.³ Arulmolid, T.⁴ Hoong, K.F.⁵

39
- 0037184883
- X. Zhang, M. Breslav, J. Grimm, K. Guan, A. Huang, F. Liu, C.A. Maryanoff, D. Palmer, M. Patel, Y. Qian, C. Shaw, K. Sorgi, S. Stefanick, and D. Xu J. Org. Chem. 67 2002 9471
- (2002) J. Org. Chem. , vol.67 , pp. 9471
- Zhang, X.¹ Breslav, M.² Grimm, J.³ Guan, K.⁴ Huang, A.⁵ Liu, F.⁶ Maryanoff, C.A.⁷ Palmer, D.⁸ Patel, M.⁹ Qian, Y.¹⁰ Shaw, C.¹¹ Sorgi, K.¹² Stefanick, S.¹³ Xu, D.¹⁴

40
- 84905087111
- K.M. Khan, F. Rahim, A. Khan, M. Shabeer, S. Hussain, W. Rehman, M. Taha, M. Khan, S. Perveen, and M.I. Choudhary Bioorg. Med. Chem. 22 2014 119
- (2014) Bioorg. Med. Chem. , vol.22 , pp. 119
- Khan, K.M.¹ Rahim, F.² Khan, A.³ Shabeer, M.⁴ Hussain, S.⁵ Rehman, W.⁶ Taha, M.⁷ Khan, M.⁸ Perveen, S.⁹ Choudhary, M.I.¹⁰

41
- 84893344425
- K.M. Khan, F. Naz, M. Taha, A. Khan, S. Perveen, M.I. Choudhary, and W. Voelter Eur. J. Med. Chem. 74 2014 314
- (2014) Eur. J. Med. Chem. , vol.74 , pp. 314
- Khan, K.M.¹ Naz, F.² Taha, M.³ Khan, A.⁴ Perveen, S.⁵ Choudhary, M.I.⁶ Voelter, W.⁷

42
- 84973378870
- R.V. Koteswara, R.V. Jhansi, W.D. Victor, and S.Y. Shirley J. Chem. Inf. Model. 20 2014 902
- (2014) J. Chem. Inf. Model. , vol.20 , pp. 902
- Koteswara, R.V.¹ Jhansi, R.V.² Victor, W.D.³ Shirley, S.Y.⁴

43
- 84870249445
- C.A. Lipinski, F. Lombardo, B.W. Dominy, and P.J. Feeney Adv. Drug Delivery Rev. 64 2012 4
- (2012) Adv. Drug Delivery Rev. , vol.64 , pp. 4
- Lipinski, C.A.¹ Lombardo, F.² Dominy, B.W.³ Feeney, P.J.⁴

44
- 13244266921
- C.A. Lipinski Drug Disc. Today Technol. 1 2004 337
- (2004) Drug Disc. Today Technol. , vol.1 , pp. 337
- Lipinski, C.A.¹

45
- 76549123580
- H. Azizian, H. Bahrami, P. Pasalar, and M. Amanlou J. Mol. Graphics Modell. 28 2010 626
- (2010) J. Mol. Graphics Modell. , vol.28 , pp. 626
- Azizian, H.¹ Bahrami, H.² Pasalar, P.³ Amanlou, M.⁴

46
- 0035991974
- H. Mishra, A.L. Parrill, and J.S. Williamson Antimicrob. Agents Chemother. 46 2002 2613
- (2002) Antimicrob. Agents Chemother. , vol.46 , pp. 2613
- Mishra, H.¹ Parrill, A.L.² Williamson, J.S.³

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