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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 15, 2015, Pages 2913-2917

Design, synthesis and biological evaluation of 4-(alkyloxy)-6-methyl-2H-pyran-2-one derivatives as quorum sensing inhibitors

(6) Park, Suzie a Kim, Han Shin a Ok, Kiwon a Kim, Yunhye a Park, Hee Deung a Byun, Youngjoo a,b

a Korea University (South Korea)

b Korea University College of Medicine (South Korea)

Author keywords

Biofilm inhibition; Pseudomonas aeruginosa; Pyrone; Quorum sensing

Indexed keywords

2 PYRONE DERIVATIVE; LIGAND; N (3 OXODODECANOYL)HOMOSERINE LACTONE; ANTIINFECTIVE AGENT; BACTERIAL PROTEIN; GAMMA BUTYROLACTONE; HOMOSERINE; LASR PROTEIN, PSEUDOMONAS AERUGINOSA; N-(3-OXODODECANOYL)HOMOSERINE LACTONE; PYRONE DERIVATIVE; TRANSACTIVATOR PROTEIN;

ARTICLE; BACTERIAL GENE; BIOFILM; CONTROLLED STUDY; CRYSTAL STRUCTURE; DOWN REGULATION; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; IN VITRO STUDY; MOLECULAR MODEL; NONHUMAN; PSEUDOMONAS AERUGINOSA; QUORUM SENSING; STRUCTURE ACTIVITY RELATION; ANALOGS AND DERIVATIVES; CHEMISTRY; DRUG EFFECTS; HUMAN; METABOLISM; MICROBIOLOGY; MOLECULAR DOCKING; PHYSIOLOGY; PSEUDOMONAS INFECTIONS;

PSEUDOMONAS AERUGINOSA;

4-BUTYROLACTONE; ANTI-BACTERIAL AGENTS; BACTERIAL PROTEINS; BIOFILMS; HOMOSERINE; HUMANS; MOLECULAR DOCKING SIMULATION; PSEUDOMONAS AERUGINOSA; PSEUDOMONAS INFECTIONS; PYRONES; QUORUM SENSING; STRUCTURE-ACTIVITY RELATIONSHIP; TRANS-ACTIVATORS;

EID: 84930924160 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2015.05.054 Document Type: Article

Times cited : (40)

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