Design of bilayer tablets using modified Dioscorea starches as novel excipients for immediate and sustained release of aceclofenac sodium

Frontiers in Pharmacology

Volumn 5, Issue , 2015, Pages

  Okunlola, Adenike ^a  

^a UNIVERSITY OF IBADAN   (Nigeria)

Author keywords

Aceclofenac sodium; Acid modification; Bilayer tablets; Carboxymethylation; Dioscorea starches; Excipients

Indexed keywords

ACECLOFENAC; HYDROXYPROPYLMETHYLCELLULOSE; STARCH; STARCH GLYCOLATE SODIUM;

ANGLE OF REPOSE; ARTICLE; BULK DENSITY; CARBOXYMETHYLATION; CARR INDEX; CHI SQUARE TEST; CONTROLLED DRUG RELEASE; CORRELATION COEFFICIENT; CRUSHING STRENGTH; DIFFUSION; DISSOLUTION; DRUG RELEASE; DRUG SOLUBILITY; ERROR; FLOW MEASUREMENT; HAUSNER RATIO; HIGUCHI AND HIXSON CROWELL MODEL; IMMEDIATE DRUG RELEASE; IN VITRO STUDY; INFRARED SPECTROSCOPY; MATHEMATICAL MODEL; METHYLATION; NONHUMAN; PARTICLE SIZE; PHYSICAL PARAMETERS; SUSTAINED DRUG RELEASE; SWELLING POWER; TABLET COMPRESSION; TABLET DISINTEGRATION; TABLET DISINTEGRATION TIME; TABLET FORMULATION; TABLET FRIABILITY; TAP DENSITY; YAM;

EID: 84926458856     PISSN: None     EISSN: 16639812     Source Type: Journal    
DOI: 10.3389/fphar.2015.00294     Document Type: Article

References (31)

1. Achutha, N. U., Srinivas, M., Meka, S. R., Averineni, K. R., Pralhad, K., and Nayanabhirama, U. (2008). Preparation and, in vitro, preclinical and clinical studies of aceclofenac spherical agglomerates. Euro. J. Pharm. Biopharm. 70, 674-683. doi: 10.1016/j.ejpb.2008.06.010
2. Akoroda, M. O., and Hahn, S. K. (1995). Yams in Nigeria: status and trends. Afr. J. Root Tuber Crops 1, 38-41.
3. Ansel, H. C., Allen, L. V. Jr., and Popovich, N. G. (2011). Pharmaceutical Dosage Forms and Drug Delivery Systems, 9th Edn. Philadelphia, PA: Lippincott Williams & Wilkins.
4. Atichokudomchai, N., and Varavinit, S. (2003). Characterization and utilization of acid-modified cross linked tapioca starch in pharmaceutical tablets. Carbohydr. Polym. v. 53, 263-270. doi: 10.1016/S0144-8617(03)00070-5
5. Banker, G. S., and Anderson, N. R. (1986). "Tablets," in The Theory and Practice of Industrial Pharmacy, 3rd Edn., eds L. Lachman, H. A. Lieberman, and J. L. Kanig (Philadelphia, PA: Lea and Febiger), 301-303.
6. Bowen, F. E., and Vadino, W. A. (1984). A simple method for differentiating sources. Drug Deve. Ind. Pharm. v. 10, 505-551. doi: 10.3109/03639048409041403
7. Chowdhury, S., and Das Saha, P. (2011). Comparative analysis of linear and non-linear methods of estimating the pseudo-second-order kinetic parameters for sorption of Malachite Green onto pretreated rice husk. Bioremediation J. 15, 181-188. doi: 10.1080/10889868.2011.624140
8. Costa, P., and Sousa Lobo, J. M. (2001). Modeling and comparison of dissolution profiles. Euro. J. Pharm. Sci. 13, 123-133. doi: 10.1016/S0928-0987(01)00095-1
9. Desphande, R. D., Gowda, D. V., Mohammed, N., and Mramwar, D. N. (2011). Bilayer tablets-anemerging trend: a review. Int. J. Pharm. Sci. Res. 2, 2534-2544.
10. Dey, S., Mahanti, B., Khila, S., Mazumder, B., and Gupta, S. D. (2012). Formulation development and optimization of bilayer tablets of aceclofenac. Expert Opin. Drug. Deliv. 9, 1041-1050. doi: 10.1517/17425247.2012.707187
11. Gupta, P., Vermani, K., and Garg, S. (2002). Hydrogels: from controlled release to PH responsive drug delivery. Drug Discov. Tech. 7, 569-579. doi: 10.1016/S1359-6446(02)02255-9
12. Higuchi, T. (1961). Rate of release of medicaments from ointment bases containing drugs in suspension. J. Pharm. Sci. 50, 874-875. doi: 10.1002/jps.2600501018
13. Hixson, A. W., and Crowell, J. H. (1931). Dependence of reaction velocity upon surface and agitation. Ind. Eng. Chem. 23, 923-931. doi: 10.1021/ie50260a018
14. Karna, N. (2012). Design, development and evaluation of novel sustained release bi-layer tablets of lornoxicam based on the combination of hydrophilic matrix formers and basic pH modifiers. Int. J. Pharm. Biol. Sci. 3, 392-402.
15. Karthikeyini, S. C., Jayaprakash, S., Abirami, A., and Halith, S. M. (2009). Formulation and evaluation of aceclofenac sodium bilayer sustained release tablets. Int. J. Chemtech Res. 1, 1381-1385.
16. Korsemeyer, R. W., Gurny, R., Doelker, E. M., Buri, P., and Peppas, N. A. (1983). Mechanism of solute release from porous hydrophilic polymers. Int. J. Pharm. 15, 25-35. doi: 10.1016/0378-5173(83)90064-9
17. Logidhasan, L., Suresh, S., and Mathivanan, M. (2013). Formulation and in vitro evaluation of bilayer floating tablets of Aceclofenac and Ranitidine Hcl Int. Res. J. Pharm. App. Sci. 3, 88-94.
18. Marshall, K. (2009). "Compression and consolidation of powdered solids," in The Theory and Practice of Industrial Pharmacy, eds L. Lachman and H. A. Lieberman (New Delhi: CBS Publishers and Distributors), 113-170.
19. Nayak, A. K., Hasnain, M. S., Beg, S., and Alam, M. I. (2010). Mucoadhesive beads of gliclazide: design, development and evaluation. Sci. Asia 36, 319-325. doi: 10.2306/scienceasia1513-1874.2010.36.319
20. Niwa, M. I., Hiraishi, Y., Iwasaki, N., and Terada, K. (2013). Quantitative analysis of the layer separation risk in bilayer tablets using terahertz pulsed imaging. Int. J. Pharm. 452, 249-256. doi: 10.1016/j.ijpharm.2013.05.010
21. Odeku, O. A., and Itiola, O. A. (2003). Evaluation of the effects of khaya gum on the mechanical and release properties of paracetamol tablets. Drug Dev. Ind. Pharm. 29, 311-320. doi: 10.1081/DDC-120018205
22. Odeku, O. A., and Picker-Freyer, K. M. (2009). Characterization of acid modified Dioscorea starches as direct compression excipient. Pharm. Dev. Technol. 14, 259-270. doi: 10.1080/10837450802572367
23. Okunlola, A., and Odeku, O. A. (2008). Comparative evaluation of starches from Dioscorea species as intragranular tablet disintegrant. J. Drug Deliv. Sci. Technol. 18, 444-447. doi: 10.1016/S1773-2247(08)50085-2
24. Okunlola, A., and Odeku, O. A. (2011). Evaluation of starches obtained from four Dioscorea species as binding agent in chloroquine phosphate tablet formulations. Saudi Pharm. J. 19, 95-105. doi: 10.1016/j.jsps.2011.01.002
25. Reddy, S., Panakanti, P. K., Kandaghatla, R., and Yamsani, M. R. (2010). Formulation and release characteristic of a bilayer matrix tablet containing glimepiride immediate release component and metformin hydrochloride as sustained release component. Int. J. Pharm. Sci. Nanotechnol. 3, 851-859.
26. Ritger, P. L., and Peppas, N. A. (1987). A simple equation for description of solute release II. Fickian and anomalous release from swellable devices. J. Control Rel. 5, 37-42. doi: 10.1016/0168-3659(87)90035-6
27. Sharif, A., E-Rabbani, M., Akhtar, M. F., Akhtar, B., Saleem, A., Murtaza, G., et al. (2011). Design and evaluation of modified release bilayer tablets of flurbiprofen. Adv. Clin. Exp. Med. 20, 343-349.
28. Sharma, R., Mittal, S., Kumar, D., Singla, P., Garg, V., and Arora, A. (2014). Formulation and evaluation of bi-layer tablet of Aceclofenac sodium and Tramadol hydrochloride. J. Fundam. Pharm. Res. 2, 22-34.
29. Singh, A. V., Nath, L. K., Guha, M., and Kumar, R. (2011). Microwave assisted synthesis and evaluation of cross-linked carboxymethylated Sagi starch as superdisintegrant. J. Pharm. Pharm. 2, 42-46. doi: 10.4236/pp.2011.21005
30. Stojanovic, Ž., Jeremic, K., Jovanovic, S., and Lechner, M. D. (2005). Comparison of some methods for determination of the degree of substitution of carboxymethyl starch. Starch - Stärke 57, 79-83. doi: 10.1002/star.200400342
31. Young, A. H. (1984). "Fractionation of starch," in Starch Chemistry. Technology, 2nd Edn., eds R. L. Whistler, J. N. Bemiller, and E. F. Pashall (London: Academic Press), 249-283.