Mucoadhesive beads of gliclazide: Design, development, and evaluation

ScienceAsia

Volumn 36, Issue 4, 2010, Pages 319-325

  Nayak, Amit Kumar ^a   Hasnain, M Saquib ^a   Beg, Sarwar ^a   Alam, M Intakhab ^b  

^a SEEMANTA INSTITUTE OF PHARMACEUTICAL SCIENCES   (India)

^b HAMDARD UNIVERSITY   (India)

Author keywords

Alginate ispaghula; Bioadhesion; Cross linking; Mucoadhesion

Indexed keywords

EID: 79251482762     PISSN: 15131874     EISSN: None     Source Type: Journal    
DOI: 10.2306/scienceasia1513-1874.2010.36.319     Document Type: Article

References (38)

1. Chowdary KPR, Srinivas L (2000) Mucoadhesive drug delivery systems: a status of current review. Indian Drugs 37, 400-6.
2. Garg S, Vasir JK, Tambweker K (2003) Bioadhesive microspheres as a controlled drug delivery system. Int J Pharm 255, 13-32. (Pubitemid 36369587)
3. Roldo M, Barbu E, Brown JF, Laight DW, Smart JD, Tsibouklis J (2006) Orally administered, colon-specific mucoadhesive azopolymer particles for the treatment of inflammatory bowel disease: An in vivo study. J Biomed Mater Res A 79, 706-15.
4. Cashman J, Burt HM, Springate C, Gleave J, Jackson JK (2004) Camptothecin-loaded films for the prevention of postsurgical adhesions. Inflamm Res 53, 355-62. (Pubitemid 39141749)
5. Chang JY, Oh YK, Kong HS, Kim EJ, Jang DD, Nam KT, Kim CK (2002) Prolonged antifungal effects of clotrimazole-containing mucoadhesive thermosensitive gels on vaginitis. J Contr Release 82, 39-50.
6. Malaekeh-Nikouei B, Sajadi TSA, Jaafari MR (2008) Preparation, characterization, and mucoadhesive properties of chitosan-coated microspheres encapsulated with cyclosporine A. Drug Dev Ind Pharm 34, 492-8.
7. Ikeda K, Murata K, Kobayashi M, Noda K (1992) Enhancement of bioavailability of dopamine via nasal route in beagle dogs. Chem Pharmaceut Bull 40, 2155-8.
8. Nagai T, Nishimoto Y, Nambu N, Suzuki Y, Sekine K (1984) Powder dosage form of insulin for nasal administration. J Contr Release 1, 15-22. (Pubitemid 15175635)
9. Shinde JV, Mali KK, Dias RJ, Havaldar VD, Mahajan NS (2008) Insitu mucoadhesive nasal gels of metoclopramide hydrochloride: preformulation and formulation studies. J Pharm Res 1, 88-96.
10. Kumar M, Misra A, Mishra AK, Mishra P, Pathak K (2008) Mucoadhesive nanoemulsion-based intranasal drug delivery system of olanzapine for brain targeting. J Drug Target 16, 806-14.
11. Wu C, Qi H, Chen W, Huang C, Su C, Li W, Hou S (2007) Preparation and evaluation of a carbopol/HPMC-based in situ gelling ophthalmic syatem for puerarin. Yakugaku Zasshi 127, 183-91.
12. Sakagami M, Kinoshita W, Sakon K, Sato JI, Makino Y (2002) Mucoadhesive beclomethasone microspheres for powder inhalation: their pharmacokinetics and pharmacodynamics evaluation. J Contr Release 80, 207-18.
13. Jasti DB, Xiaoling LI, Cleary G (2003) Recent advances in mucoadhesive drug delivery system. Business Briefing Pharmatech 194-6.
14. Thorat YS, Modi VS, Dhavale SC (2009) Use of carbomers to design mucoadhesive microspheres for an anti- H. pylori drug, clarithromycin. Int J PharmTech Res 1, 1421-8.
15. Chowdary KPR, Rao YS (2003) Design and in vitro and in vivo evaluation of mucoadhesive microcapsules of glipizide for oral controlled release: A technical note. AAPS PharmSciTech 4, 87-92.
16. Cuna M, Alonso MJ, Torres D (2001) Preparation and in vivo evaluation of mucoadhesive microparticles containing amoxicillin-resin complexes for drug delivery to the gastric mucosa. Eur J Pharm Biopharm 51, 199-205.
17. Nagahara N, Akiyama Y, Nakao M, Tada M, Kitano M, Ogawa Y (1998) Mucoadhesive microspheres containing amoxicillin for clearance of H. pylori. Antimicrob Agents Chemother 42, 2492-4.
18. Liu Z, Lu W, Qian L (2005) In vitro and in vivo studies on mucoadhesive microspheres of amoxicillin. J Contr Release 102, 135-44. (Pubitemid 40093780)
19. Takishima J, Onishi H, Machida Y (2002) Prolonged intestinal absorption of Cephradine with chitosancoated ethylcellulose microparticles in rats. Biol Pharmaceut Bull 25, 1498-502.
20. Sharma HK, Sarangi B, Pradhan SP (2009) Preparation and in-vitro evaluation of mucoadhesive microbeads containing Timolol Maléate using mucoadhesive substances of Dillenia indica L. Arch Pharmaceut Sci Res 1, 181-8.
21. Harrower A (1994) Comparison of efficacy, secondary failure rate and complication of sulfonylureas. J Diabetes Complications 8, 201-3.
22. Palmer K, Brogde R (1993) Gliclazide- an update of its pharmacological properties and therapeutic efficacy in non-insulin dependent diabetes mellitus. Drugs 46, 92-125. (Pubitemid 23232408)
23. Mailhot J (1993) Efficacy and safety of gliclazide in the treatment of non-insulin dependent diabetes mellitus: a Canadian multicenter study. Clin Therapeut 15, 1060-8.
24. Young JF, Wei GL, Lu R, Liu CX, Zheng BZ, Feng P (2006) Bioavailability of gliclazide sustained release tablet in healthy volunteers. Asian J Pharmacodyn Pharmacokin 2, 150-60.
25. Hong S, Lee S, Lee Y, Chung S, Lee M, Shim C (1998) Accelerated oral absorption of gliclazide in human subjects from a soft gelatin capsule containing a PEG 400 suspension of gliclazide. J Contr Release 51, 85-92.
26. Al-Kassas RS, Al-Gohary OMN, Al-Faadhel MM (2007) Controlling of systemic absorption of gliclazide through incorporation into alginate beads. Int J Pharm 341, 230-7.
27. Bhardwaj TR, Kanwar M, Lal R, Gupta A (2000) Natural gums and modified natural gums as sustainedrelease carriers. Drug Dev Ind Pharm 26, 1025-38.
28. El-Kamel AH, Al-Gohary MN, Hosny EA (2003) Alginate-diltiazem hydrochloride beads: Optimization of formulation factors, in vitro and in vivo availability. J Microencapsul 20, 211-25.
29. Smidsrod O, Draget KI (1996) Chemistry and physical properties of alginates. Carbohydr Eur 14, 6-13.
30. Prajapati SK, Tripathi P, Ubaidulla U, Anand V (2008) Design and development of gliclazide mucoadhesive microcapsules: in vitro and in vivo evaluation. AAPS PharmSciTech 9, 224-30.
31. Sharma VK, Bhattacharya A (2008) Release of metformin hydrochloride from ispaghula-sodium alginate beads adhered on cock intestinal mucosa. Indian J Pharmaceut Educ Res 42, 365-72.
32. Kikuci A, Kawabuchi M, Sugihara M, Sakurai Y (1997) Pulsed dextran release from calcium-alginate beads. J Contr Release 47, 21-9. (Pubitemid 27154397)
33. Hudson A, Mitchell J, Davies M, Melia C (1995) Structure behavior of hydrophilic matrix sustained-release dosage form 3. The influence of pH on the sustained release performance and internal gel structure of sodium alginate matrices. J Contr Release 33, 143-52.
34. George M, Abraham TE (2006) Polyionic hydrocolloids for the intestinal delivery of protein drugs: alginate and chitosan- a review. J Contr Release 114, 1-14.
35. Sandhu JS, Hudson J, Kennedy JF (1981) The gel nature and structure of the carbohydrate of Ispaghula husk (ex Plantago ovatd) Forsk. Carbohydr Res 93, 247-50.
36. Yotsuyangi T, Ohkubo T, Ohaasi T, Kedak I (1987) Calcium-induced gelation of alginic acid and pH sensitive reswelling of dried gels. Chem Pharmaceut Bull 34, 1555-63.
37. Andreopoulos AG (1985) Stability of some soluble alginate solutions. Biomaterials 6, 68-9.
38. Sanap GS (2009) Formulation and evaluation of mucoadhesive beads of glipizide using 23 factorial design. J Pharm Res 2, 934-8.