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Volumn 51, Issue 28, 2015, Pages 6157-6160
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Triblock peptide-linker-lipid molecular design improves potency of peptide ligands targeting family B G protein-coupled receptors
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Author keywords
[No Author keywords available]
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Indexed keywords
G PROTEIN COUPLED RECEPTOR;
PARATHYROID HORMONE RECEPTOR 1;
LIGAND;
LIPID;
PEPTIDE;
PTH1R PROTEIN, HUMAN;
AGONIST;
AMINO ACID SEQUENCE;
ARTICLE;
CELL SURFACE;
CONJUGATION;
CRITICAL MICELLE CONCENTRATION;
EC50;
KIDNEY CLEARANCE;
LIGAND BINDING;
MICELLE;
MOLECULAR MODEL;
MOLECULAR WEIGHT;
PROTEIN DEGRADATION;
PROTEIN LIPID INTERACTION;
STEREOSPECIFICITY;
SURFACE TENSION;
BIOSYNTHESIS;
CHEMICAL STRUCTURE;
CHEMISTRY;
DOSE RESPONSE;
GENETICS;
HEK293 CELL LINE;
HUMAN;
STRUCTURE ACTIVITY RELATION;
DOSE-RESPONSE RELATIONSHIP, DRUG;
HEK293 CELLS;
HUMANS;
LIGANDS;
LIPIDS;
MOLECULAR STRUCTURE;
PEPTIDES;
RECEPTOR, PARATHYROID HORMONE, TYPE 1;
STRUCTURE-ACTIVITY RELATIONSHIP;
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EID: 84925583040
PISSN: 13597345
EISSN: 1364548X
Source Type: Journal
DOI: 10.1039/c5cc00301f Document Type: Article |
Times cited : (8)
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References (32)
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