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Volumn 16, Issue 1, 2014, Pages

Estrogen receptor mutations and their role in breast cancer progression

Author keywords

[No Author keywords available]

Indexed keywords

ANASTROZOLE; ESTROGEN RECEPTOR; FULVESTRANT; LETROZOLE; TAMOXIFEN; ANTINEOPLASTIC HORMONE AGONISTS AND ANTAGONISTS; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR ALPHA, HUMAN;

EID: 84924244611     PISSN: 14655411     EISSN: 1465542X     Source Type: Journal    
DOI: 10.1186/s13058-014-0494-7     Document Type: Review
Times cited : (86)

References (42)
  • 2
    • 0031047767 scopus 로고    scopus 로고
    • Androgen receptor gene amplification in a recurrent prostate cancer after monotherapy with the nonsteroidal potent antiandrogen Casodex (bicalutamide) with a subsequent favorable response to maximal androgen blockade
    • Palmberg C, Koivisto P, Hyytinen E, Isola J, Visakorpi T, Kallioniemi OP, Tammela T: Androgen receptor gene amplification in a recurrent prostate cancer after monotherapy with the nonsteroidal potent antiandrogen Casodex (bicalutamide) with a subsequent favorable response to maximal androgen blockade. Eur Urol 1997, 31:216-219.
    • (1997) Eur Urol , vol.31 , pp. 216-219
    • Palmberg, C.1    Koivisto, P.2    Hyytinen, E.3    Isola, J.4    Visakorpi, T.5    Kallioniemi, O.P.6    Tammela, T.7
  • 3
    • 0035800507 scopus 로고    scopus 로고
    • Clinical resistance to STI-571 cancer therapy caused by BCR-ABL gene mutation or amplification
    • Gorre ME, Mohammed M, Ellwood K, Hsu N, Paquette R, Rao PN, Sawyers CL: Clinical resistance to STI-571 cancer therapy caused by BCR-ABL gene mutation or amplification. Science 2001, 293:876-880.
    • (2001) Science , vol.293 , pp. 876-880
    • Gorre, M.E.1    Mohammed, M.2    Ellwood, K.3    Hsu, N.4    Paquette, R.5    Rao, P.N.6    Sawyers, C.L.7
  • 8
    • 34247378586 scopus 로고    scopus 로고
    • Hormones and cancer
    • Shang Y: Hormones and cancer. Cell Res 2007, 17:277-279.
    • (2007) Cell Res , vol.17 , pp. 277-279
    • Shang, Y.1
  • 9
    • 33646371740 scopus 로고    scopus 로고
    • Molecular mechanisms of oestrogen and SERMs in endometrial carcinogenesis
    • Shang Y: Molecular mechanisms of oestrogen and SERMs in endometrial carcinogenesis. Nat Rev Cancer 2006, 6:360-368.
    • (2006) Nat Rev Cancer , vol.6 , pp. 360-368
    • Shang, Y.1
  • 10
    • 79958149945 scopus 로고    scopus 로고
    • The turnover of estrogen receptor alpha by the selective estrogen receptor degrader (SERD) fulvestrant is a saturable process that is not required for antagonist efficacy
    • Wardell SE, Marks JR, McDonnell DP: The turnover of estrogen receptor alpha by the selective estrogen receptor degrader (SERD) fulvestrant is a saturable process that is not required for antagonist efficacy. Biochem Pharmacol 2011, 82:122-130.
    • (2011) Biochem Pharmacol , vol.82 , pp. 122-130
    • Wardell, S.E.1    Marks, J.R.2    McDonnell, D.P.3
  • 12
    • 19344364880 scopus 로고    scopus 로고
    • Effects of chemotherapy and hormonal therapy for early breast cancer on recurrence and 15-year survival: an overview of the randomised trials
    • Early Breast Cancer Trialists' Collaborative Group: Effects of chemotherapy and hormonal therapy for early breast cancer on recurrence and 15-year survival: an overview of the randomised trials. Lancet 2005, 365:1687-1717.
    • (2005) Lancet , vol.365 , pp. 1687-1717
  • 13
    • 69249137029 scopus 로고    scopus 로고
    • Biological determinants of endocrine resistance in breast cancer
    • Musgrove EA, Sutherland RL: Biological determinants of endocrine resistance in breast cancer. Nat Rev Cancer 2009, 9:631-643.
    • (2009) Nat Rev Cancer , vol.9 , pp. 631-643
    • Musgrove, E.A.1    Sutherland, R.L.2
  • 14
    • 84858385940 scopus 로고    scopus 로고
    • Endocrine resistance in breast cancer: molecular pathways and rational development of targeted therapies
    • Roop RP, Ma CX: Endocrine resistance in breast cancer: molecular pathways and rational development of targeted therapies. Future Oncol 2012, 8:273-292.
    • (2012) Future Oncol , vol.8 , pp. 273-292
    • Roop, R.P.1    Ma, C.X.2
  • 15
    • 0022424564 scopus 로고
    • Oncogenes homologous to steroid receptors?
    • Sluyser M, Mester J: Oncogenes homologous to steroid receptors? Nature 1985, 315:546.
    • (1985) Nature , vol.315 , pp. 546
    • Sluyser, M.1    Mester, J.2
  • 17
  • 18
    • 0030940071 scopus 로고    scopus 로고
    • An estrogen receptor mutant with strong hormone-independent activity from a metastatic breast cancer
    • Zhang QX, Borg A, Wolf DM, Oesterreich S, Fuqua SA: An estrogen receptor mutant with strong hormone-independent activity from a metastatic breast cancer. Cancer Res 1997, 57:1244-1249.
    • (1997) Cancer Res , vol.57 , pp. 1244-1249
    • Zhang, Q.X.1    Borg, A.2    Wolf, D.M.3    Oesterreich, S.4    Fuqua, S.A.5
  • 20
    • 79952395270 scopus 로고    scopus 로고
    • Cancer genomics: from discovery science to personalized medicine
    • Chin L, Andersen JN, Futreal PA: Cancer genomics: from discovery science to personalized medicine. Nat Med 2011, 17:297-303.
    • (2011) Nat Med , vol.17 , pp. 297-303
    • Chin, L.1    Andersen, J.N.2    Futreal, P.A.3
  • 23
    • 84877028141 scopus 로고    scopus 로고
    • Comprehensive molecular portraits of human breast tumours
    • Network CGA: Comprehensive molecular portraits of human breast tumours. Nature 2012, 490:61-70.
    • (2012) Nature , vol.490 , pp. 61-70
    • Network, C.G.A.1
  • 26
    • 0028208456 scopus 로고
    • Endometrial cancer in tamoxifen-treated breast cancer patients: findings from the National Surgical Adjuvant Breast and Bowel Project (NSABP) B-14
    • Fisher B, Costantino JP, Redmond CK, Fisher ER, Wickerham DL, Cronin WM: Endometrial cancer in tamoxifen-treated breast cancer patients: findings from the National Surgical Adjuvant Breast and Bowel Project (NSABP) B-14. J Natl Cancer Inst 1994, 86:527-537.
    • (1994) J Natl Cancer Inst , vol.86 , pp. 527-537
    • Fisher, B.1    Costantino, J.P.2    Redmond, C.K.3    Fisher, E.R.4    Wickerham, D.L.5    Cronin, W.M.6
  • 32
    • 0030445855 scopus 로고    scopus 로고
    • Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein
    • Weis KE, Ekena K, Thomas JA, Lazennec G, Katzenellenbogen BS: Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein. Mol Endocrinol 1996, 10:1388-1398.
    • (1996) Mol Endocrinol , vol.10 , pp. 1388-1398
    • Weis, K.E.1    Ekena, K.2    Thomas, J.A.3    Lazennec, G.4    Katzenellenbogen, B.S.5
  • 33
    • 0032568527 scopus 로고    scopus 로고
    • Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains
    • Tanenbaum DM, Wang Y, Williams SP, Sigler PB: Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains. Proc Natl Acad Sci U S A 1998, 95:5998-6003.
    • (1998) Proc Natl Acad Sci U S A , vol.95 , pp. 5998-6003
    • Tanenbaum, D.M.1    Wang, Y.2    Williams, S.P.3    Sigler, P.B.4
  • 35
    • 0032446607 scopus 로고    scopus 로고
    • The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen
    • Shiau AK, Barstad D, Loria PM, Cheng L, Kushner PJ, Agard DA, Greene GL: The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen. Cell 1998, 95:927-937.
    • (1998) Cell , vol.95 , pp. 927-937
    • Shiau, A.K.1    Barstad, D.2    Loria, P.M.3    Cheng, L.4    Kushner, P.J.5    Agard, D.A.6    Greene, G.L.7
  • 36
    • 0030734795 scopus 로고    scopus 로고
    • Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: evidence that an open pocket conformation is required for ligand interaction
    • Carlson KE, Choi I, Gee A, Katzenellenbogen BS, Katzenellenbogen JA: Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: evidence that an open pocket conformation is required for ligand interaction. Biochemistry 1997, 36:14897-14905.
    • (1997) Biochemistry , vol.36 , pp. 14897-14905
    • Carlson, K.E.1    Choi, I.2    Gee, A.3    Katzenellenbogen, B.S.4    Katzenellenbogen, J.A.5
  • 37
    • 0031473542 scopus 로고    scopus 로고
    • Mechanistic aspects of estrogen receptor activation probed with constitutively active estrogen receptors: correlations with DNA and coregulator interactions and receptor conformational changes
    • Lazennec G, Ediger TR, Petz LN, Nardulli AM, Katzenellenbogen BS: Mechanistic aspects of estrogen receptor activation probed with constitutively active estrogen receptors: correlations with DNA and coregulator interactions and receptor conformational changes. Mol Endocrinol 1997, 11:1375-1386.
    • (1997) Mol Endocrinol , vol.11 , pp. 1375-1386
    • Lazennec, G.1    Ediger, T.R.2    Petz, L.N.3    Nardulli, A.M.4    Katzenellenbogen, B.S.5
  • 38
    • 0027423151 scopus 로고
    • Identification of charged residues in an N-terminal portion of the hormone-binding domain of the human estrogen receptor important in transcriptional activity of the receptor
    • Pakdel F, Reese JC, Katzenellenbogen BS: Identification of charged residues in an N-terminal portion of the hormone-binding domain of the human estrogen receptor important in transcriptional activity of the receptor. Mol Endocrinol 1993, 7:1408-1417.
    • (1993) Mol Endocrinol , vol.7 , pp. 1408-1417
    • Pakdel, F.1    Reese, J.C.2    Katzenellenbogen, B.S.3
  • 39
    • 0038711505 scopus 로고    scopus 로고
    • Mutation of Leu-536 in human estrogen receptor-alpha alters the coupling between ligand binding, transcription activation, and receptor conformation
    • Zhao C, Koide A, Abrams J, Deighton-Collins S, Martinez A, Schwartz JA, Koide S, Skafar DF: Mutation of Leu-536 in human estrogen receptor-alpha alters the coupling between ligand binding, transcription activation, and receptor conformation. J Biol Chem 2003, 278:27278-27286.
    • (2003) J Biol Chem , vol.278 , pp. 27278-27286
    • Zhao, C.1    Koide, A.2    Abrams, J.3    Deighton-Collins, S.4    Martinez, A.5    Schwartz, J.A.6    Koide, S.7    Skafar, D.F.8
  • 41
    • 33644984327 scopus 로고    scopus 로고
    • Fulvestrant in women with advanced breast cancer after progression on prior aromatase inhibitor therapy: North Central Cancer Treatment Group Trial N0032
    • Ingle JN, Suman VJ, Rowland KM, Mirchandani D, Bernath AM, Camoriano JK, Fishkin PA, Nikcevich DA, Perez EA, North Central Cancer Treatment Group Trial N0032: Fulvestrant in women with advanced breast cancer after progression on prior aromatase inhibitor therapy: North Central Cancer Treatment Group Trial N0032. J Clin Oncol 2006, 24:1052-1056.
    • (2006) J Clin Oncol , vol.24 , pp. 1052-1056


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.