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Angewandte Chemie - International Edition

Volumn 54, Issue 16, 2015, Pages 4758-4763

Nanomolar Inhibitors of the Transcription Factor STAT5b with High Selectivity over STAT5a

(5) Elumalai, Nagarajan a Berg, Angela a Natarajan, Kalaiselvi a Scharow, Andrej a Berg, Thorsten a

a UNIVERSITY OF LEIPZIG (Germany)

Author keywords

inhibitors; natural products; protein protein interactions; STAT5; transcription factors

Indexed keywords

CORROSION INHIBITORS; MOLECULES; PROTEINS; SIGNAL TRANSDUCTION; TRANSCRIPTION; AMINO ACIDS; TRANSCRIPTION FACTORS;

NANOMOLAR INHIBITORS; NATURAL PRODUCTS; NATURALLY OCCURRING; PROTEIN-PROTEIN INTERACTIONS; SMALL ORGANIC MOLECULES; SRC HOMOLOGY 2 DOMAINS; STAT5; STRUCTURAL SIMILARITY;

TRANSCRIPTION FACTORS; TRANSCRIPTION;

BIOLOGICAL PRODUCT; CATECHOL; CATECHOL DERIVATIVE; PEPTIDE; PROTEIN BINDING; STAT5 PROTEIN; STAT5A PROTEIN, HUMAN; STAT5B PROTEIN, HUMAN; TUMOR SUPPRESSOR PROTEIN;

AMINO ACID SEQUENCE; ANTAGONISTS AND INHIBITORS; BINDING SITE; CHEMISTRY; HUMAN; METABOLISM; MOLECULAR DOCKING; PHOSPHORYLATION; PROTEIN DOMAIN; SRC HOMOLOGY DOMAIN; STRUCTURE ACTIVITY RELATION;

AMINO ACID SEQUENCE; BINDING SITES; BIOLOGICAL PRODUCTS; CATECHOLS; HUMANS; MOLECULAR DOCKING SIMULATION; PEPTIDES; PHOSPHORYLATION; PROTEIN BINDING; PROTEIN INTERACTION DOMAINS AND MOTIFS; SRC HOMOLOGY DOMAINS; STAT5 TRANSCRIPTION FACTOR; STRUCTURE-ACTIVITY RELATIONSHIP; TUMOR SUPPRESSOR PROTEINS;

EID: 84923376898 PISSN: 14337851 EISSN: 15213773 Source Type: Journal
DOI: 10.1002/anie.201410672 Document Type: Article

Times cited : (51)

References (28)

1
- 0842346438
- T. Pawson, Cell 2004, 116, 191–203.
- (2004) Cell , vol.116 , pp. 191-203
- Pawson, T.¹

2
- 0034008847
- R
- J. E. Ladbury, S. Arold, Chem. Biol. 2000, 7, R3–8;
- (2000) Chem. Biol. , vol.7 , pp. 3-8
- Ladbury, J.E.¹ Arold, S.²

3
- 84883353803
- D. Kraskouskaya, E. Duodu, C. C. Arpin, P. T. Gunning, Chem. Soc. Rev. 2013, 42, 3337–3370.
- (2013) Chem. Soc. Rev. , vol.42 , pp. 3337-3370
- Kraskouskaya, D.¹ Duodu, E.² Arpin, C.C.³ Gunning, P.T.⁴

4
- 41149149301
- L. Hennighausen, G. W. Robinson, Genes Dev. 2008, 22, 711–721.
- (2008) Genes Dev. , vol.22 , pp. 711-721
- Hennighausen, L.¹ Robinson, G.W.²

5
- 0030607257
- P. May, C. Gerhartz, B. Heesel, T. Welte, W. Doppler, L. Graeve, F. Horn, P. C. Heinrich, FEBS Lett. 1996, 394, 221–226.
- (1996) FEBS Lett. , vol.394 , pp. 221-226
- May, P.¹ Gerhartz, C.² Heesel, B.³ Welte, T.⁴ Doppler, W.⁵ Graeve, L.⁶ Horn, F.⁷ Heinrich, P.C.⁸

6
- 79952528759
- V. Hwa, K. Nadeau, J. M. Wit, R. G. Rosenfeld, Best. Pract. Res. Clin. Endocrinol. Metab. 2011, 25, 61–75;
- (2011) Best. Pract. Res. Clin. Endocrinol. Metab. , vol.25 , pp. 61-75
- Hwa, V.¹ Nadeau, K.² Wit, J.M.³ Rosenfeld, R.G.⁴

7
- 46349102713
- B. Basham, M. Sathe, J. Grein, T. McClanahan, A. D’Andrea, E. Lees, A. Rascle, Nucleic Acids Res. 2008, 36, 3802–3818.
- (2008) Nucleic Acids Res. , vol.36 , pp. 3802-3818
- Basham, B.¹ Sathe, M.² Grein, J.³ McClanahan, T.⁴ D’Andrea, A.⁵ Lees, E.⁶ Rascle, A.⁷

8
- 0142219889
- S. Xi, Q. Zhang, W. E. Gooding, T. E. Smithgall, J. R. Grandis, Cancer Res. 2003, 63, 6763–6771.
- (2003) Cancer Res. , vol.63 , pp. 6763-6771
- Xi, S.¹ Zhang, Q.² Gooding, W.E.³ Smithgall, T.E.⁴ Grandis, J.R.⁵

9
- 84901290824
- e
- M. Schaller-Schönitz, D. Barzan, A. J. Williamson, J. R. Griffiths, I. Dallmann, K. Battmer, A. Ganser, A. D. Whetton, M. Scherr, M. Eder, PLoS One 2014, 9, e97243.
- (2014) PLoS One , vol.9
- Schaller-Schönitz, M.¹ Barzan, D.² Williamson, A.J.³ Griffiths, J.R.⁴ Dallmann, I.⁵ Battmer, K.⁶ Ganser, A.⁷ Whetton, A.D.⁸ Scherr, M.⁹ Eder, M.¹⁰

10
- 43149095374
- J. Müller, B. Sperl, W. Reindl, A. Kiessling, T. Berg, ChemBioChem 2008, 9, 723–727;
- (2008) ChemBioChem , vol.9 , pp. 723-727
- Müller, J.¹ Sperl, B.² Reindl, W.³ Kiessling, A.⁴ Berg, T.⁵

11
- 77952362757
- S. Wetzel, W. Wilk, S. Chammaa, B. Sperl, A. G. Roth, A. Yektaoglu, S. Renner, T. Berg, C. Arenz, A. Giannis, T. I. Oprea, D. Rauh, M. Kaiser, H. Waldmann, Angew. Chem. Int. Ed. 2010, 49, 3666–3670;
- (2010) Angew. Chem. Int. Ed. , vol.49 , pp. 3666-3670
- Wetzel, S.¹ Wilk, W.² Chammaa, S.³ Sperl, B.⁴ Roth, A.G.⁵ Yektaoglu, A.⁶ Renner, S.⁷ Berg, T.⁸ Arenz, C.⁹ Giannis, A.¹⁰ Oprea, T.I.¹¹ Rauh, D.¹² Kaiser, M.¹³ Waldmann, H.¹⁴

12
- 79952176565
- Angew. Chem. 2010, 122, 3748–3752;
- (2010) Angew. Chem. , vol.122 , pp. 3748-3752

13
- 84856845674
- B. D. Page, H. Khoury, R. C. Laister, S. Fletcher, M. Vellozo, A. Manzoli, P. Yue, J. Turkson, M. D. Minden, P. T. Gunning, J. Med. Chem. 2012, 55, 1047–1055;
- (2012) J. Med. Chem. , vol.55 , pp. 1047-1055
- Page, B.D.¹ Khoury, H.² Laister, R.C.³ Fletcher, S.⁴ Vellozo, M.⁵ Manzoli, A.⁶ Yue, P.⁷ Turkson, J.⁸ Minden, M.D.⁹ Gunning, P.T.¹⁰

14
- 84926465672
- A. A. Cumaraswamy, A. M. Lewis, M. Geletu, A. Todic, D. B. Diaz, X. R. Cheng, C. E. Brown, R. C. Laister, D. Muench, K. Kerman, H. L. Grimes, M. D. Minden, P. T. Gunning, ACS Med. Chem. Lett. 2014, 5, 1202–1206.
- (2014) ACS Med. Chem. Lett. , vol.5 , pp. 1202-1206
- Cumaraswamy, A.A.¹ Lewis, A.M.² Geletu, M.³ Todic, A.⁴ Diaz, D.B.⁵ Cheng, X.R.⁶ Brown, C.E.⁷ Laister, R.C.⁸ Muench, D.⁹ Kerman, K.¹⁰ Grimes, H.L.¹¹ Minden, M.D.¹² Gunning, P.T.¹³

15
- 80054999462
- M. Gräber, W. Janczyk, B. Sperl, N. Elumalai, C. Kozany, F. Hausch, T. A. Holak, T. Berg, ACS Chem. Biol. 2011, 6, 1008–1014.
- (2011) ACS Chem. Biol. , vol.6 , pp. 1008-1014
- Gräber, M.¹ Janczyk, W.² Sperl, B.³ Elumalai, N.⁴ Kozany, C.⁵ Hausch, F.⁶ Holak, T.A.⁷ Berg, T.⁸

16
- 65749095573
- B. Sperl, M. H. Seifert, T. Berg, Bioorg. Med. Chem. Lett. 2009, 19, 3305–3309.
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 3305-3309
- Sperl, B.¹ Seifert, M.H.² Berg, T.³

17
- 76149120388
- O. Trott, A. J. Olson, J. Comput. Chem. 2010, 31, 455–461.
- (2010) J. Comput. Chem. , vol.31 , pp. 455-461
- Trott, O.¹ Olson, A.J.²

18
- 28844472292
- D. Neculai, A. M. Neculai, S. Verrier, K. Straub, K. Klumpp, E. Pfitzner, S. Becker, J. Biol. Chem. 2005, 280, 40782–40787.
- (2005) J. Biol. Chem. , vol.280 , pp. 40782-40787
- Neculai, D.¹ Neculai, A.M.² Verrier, S.³ Straub, K.⁴ Klumpp, K.⁵ Pfitzner, E.⁶ Becker, S.⁷

19
- 0030950608
- J. Kuriyan, D. Cowburn, Annu. Rev. Biophys. Biomol. Struct. 1997, 26, 259–288.
- (1997) Annu. Rev. Biophys. Biomol. Struct. , vol.26 , pp. 259-288
- Kuriyan, J.¹ Cowburn, D.²

20
- 0030047044
- L. J. Silverberg, J. L. Dillon, P. Vemishetti, Tetrahedron Lett. 1996, 37, 771–774.
- (1996) Tetrahedron Lett. , vol.37 , pp. 771-774
- Silverberg, L.J.¹ Dillon, J.L.² Vemishetti, P.³

21
- 7444262377
- Z. Nikolovska-Coleska, R. Wang, X. Fang, H. Pan, Y. Tomita, P. Li, P. P. Roller, K. Krajewski, N. G. Saito, J. A. Stuckey, S. Wang, Anal. Biochem. 2004, 332, 261–273.
- (2004) Anal. Biochem. , vol.332 , pp. 261-273
- Nikolovska-Coleska, Z.¹ Wang, R.² Fang, X.³ Pan, H.⁴ Tomita, Y.⁵ Li, P.⁶ Roller, P.P.⁷ Krajewski, K.⁸ Saito, N.G.⁹ Stuckey, J.A.¹⁰ Wang, S.¹¹

22
- 0029866781
- F. W. Quelle, D. Wang, T. Nosaka, W. E. Thierfelder, D. Stravopodis, Y. Weinstein, J. N. Ihle, Mol. Cell. Biol. 1996, 16, 1622–1631.
- (1996) Mol. Cell. Biol. , vol.16 , pp. 1622-1631
- Quelle, F.W.¹ Wang, D.² Nosaka, T.³ Thierfelder, W.E.⁴ Stravopodis, D.⁵ Weinstein, Y.⁶ Ihle, J.N.⁷

23
- 40649097012
- J. Müller, J. Schust, T. Berg, Anal. Biochem. 2008, 375, 249–254.
- (2008) Anal. Biochem. , vol.375 , pp. 249-254
- Müller, J.¹ Schust, J.² Berg, T.³

24
- 0036782706
- J. E. Darnell, Jr., Nat. Rev. Cancer 2002, 2, 740–749;
- (2002) Nat. Rev. Cancer , vol.2 , pp. 740-749
- Darnell, J.E.¹

25
- 1042302005
- H. Yu, R. Jove, Nat. Rev. Cancer 2004, 4, 97–105;
- (2004) Nat. Rev. Cancer , vol.4 , pp. 97-105
- Yu, H.¹ Jove, R.²

26
- 50449096662
- T. Berg, ChemBioChem 2008, 9, 2039–2044.
- (2008) ChemBioChem , vol.9 , pp. 2039-2044
- Berg, T.¹

27
- 79957742210
- P. K. Mandal, F. Gao, Z. Lu, Z. Ren, R. Ramesh, J. S. Birtwistle, K. K. Kaluarachchi, X. Chen, R. C. Bast, W. S. Liao, J. S. McMurray, J. Med. Chem. 2011, 54, 3549–3563.
- (2011) J. Med. Chem. , vol.54 , pp. 3549-3563
- Mandal, P.K.¹ Gao, F.² Lu, Z.³ Ren, Z.⁴ Ramesh, R.⁵ Birtwistle, J.S.⁶ Kaluarachchi, K.K.⁷ Chen, X.⁸ Bast, R.C.⁹ Liao, W.S.¹⁰ McMurray, J.S.¹¹

28
- 33750982120
- J. Schust, B. Sperl, A. Hollis, T. U. Mayer, T. Berg, Chem. Biol. 2006, 13, 1235–1242.
- (2006) Chem. Biol. , vol.13 , pp. 1235-1242
- Schust, J.¹ Sperl, B.² Hollis, A.³ Mayer, T.U.⁴ Berg, T.⁵

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