메뉴 건너뛰기




Volumn 9, Issue 4, 2014, Pages 293-300

Synthesis, characterization and pharmacological studies of sulphur containing 1,2,4-triazole derivatives

Author keywords

1,2,4 triazole derivatives; Antimicrobial activity; Drug like characteristics; Spectral analysis; Synthesis

Indexed keywords

1 [2 (4 CHLOROPHENOXY)ACETYL] THIOSEMICARBAZIDE; 1,2,4 TRIAZOLE DERIVATIVE; 2 (4 CHLOROPHENOXY)ACETOHYDRAZIDE; 3 BENZYLSULFANYL 5 (4 CHLORO PHENOXYMETHYL) 4H 1,2,4 TRIAZOLE; 4 [3 BENZYLSULFANYL 5 (4 CHLOROPHENOXYMETHYL) 1,2,4 TRIAZOLE 4 YLMETHYL] MORPHOLINE; 4 [[3 (4 CHLORO PHENOXYMETHYL) 5 (4 SUBSTITUTED BENZYLSULFONYL) 1,2,4 TRIAZOL 4 YL]METHYL] MORPHOLINE; 5 (4 CHLOROPHENOXYMETHYL) 2,4 DIHYDRO 1,2,4TRIAZOLE 3 THIONE; ETHYL 2 (4 CHLOROPHENOXY)ACETATE; SULFUR; UNCLASSIFIED DRUG;

EID: 84919843565     PISSN: 16583612     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jtumed.2014.06.002     Document Type: Article
Times cited : (13)

References (23)
  • 2
    • 33746492059 scopus 로고
    • US patent, 3, 849434, (1974)
    • Coffen DL, Fryer RI. US patent, 3, 849434, (1974). Chem Abstr 1975; 82: 730044v.
    • (1975) Chem Abstr , vol.82 , pp. 730044v
    • Coffen, D.L.1    Fryer, R.I.2
  • 3
    • 77952431201 scopus 로고
    • Antibiotiki Moscow, 18, 71, (1973)
    • F.E. Povelista, and A.G. Gural Antibiotiki Moscow, 18, 71, (1973) Chem Abstr 78 1973 93044
    • (1973) Chem Abstr , vol.78 , pp. 93044
    • Povelista, F.E.1    Gural, A.G.2
  • 4
    • 84874112919 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity of some new 1,3-thiazoles, 1,3,4-thiadiazoles, 1,2,4-triazoles and 1,3-thiazines incorporating acridine and 1,2,3,4-tetrahydroacridine moieties
    • Tarik El-Sayed Ali, and Azza Mohammed El-Kazak Synthesis and antimicrobial activity of some new 1,3-thiazoles, 1,3,4-thiadiazoles, 1,2,4-triazoles and 1,3-thiazines incorporating acridine and 1,2,3,4-tetrahydroacridine moieties Eur J Chem 1 2010 6 11
    • (2010) Eur J Chem , vol.1 , pp. 6-11
    • El-Sayed Ali, T.1    El-Kazak, A.M.2
  • 5
    • 84863292054 scopus 로고    scopus 로고
    • Novel biotransformation process of podophyllotoxin to 4 β-sulfur-substituted podophyllum derivates with anti-tumor activity by penicillium purpurogenum
    • J.K. Bai, W. Zhao, H.M. Li, and Y.J. Tang Novel biotransformation process of podophyllotoxin to 4 β-sulfur-substituted podophyllum derivates with anti-tumor activity by penicillium purpurogenum Curr Med Chem 19 2012 927 936
    • (2012) Curr Med Chem , vol.19 , pp. 927-936
    • Bai, J.K.1    Zhao, W.2    Li, H.M.3    Tang, Y.J.4
  • 6
    • 33748462990 scopus 로고    scopus 로고
    • Heterocyclic system containing bridgehead nitrogen atom: Synthesis and pharmacological activities of some substituted 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles
    • V. Mathew, J. Keshavayya, and V.P. Vaidya Heterocyclic system containing bridgehead nitrogen atom: synthesis and pharmacological activities of some substituted 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles Eur J Med Chem 41 2006 1048 1058
    • (2006) Eur J Med Chem , vol.41 , pp. 1048-1058
    • Mathew, V.1    Keshavayya, J.2    Vaidya, V.P.3
  • 8
    • 38949192856 scopus 로고    scopus 로고
    • Synthesis, determination of the lipophilicity, anticancer and antimicrobial properties of some fused 1,2,4 triazolederivatives
    • K. Sztanke, T. Tomasz, R. Jolanta, P. Kazimierz, and K. Martyna Synthesis, determination of the lipophilicity, anticancer and antimicrobial properties of some fused 1,2,4 triazolederivatives Eur J Med Chem 43 2008 404 419
    • (2008) Eur J Med Chem , vol.43 , pp. 404-419
    • Sztanke, K.1    Tomasz, T.2    Jolanta, R.3    Kazimierz, P.4    Martyna, K.5
  • 9
    • 77957856848 scopus 로고    scopus 로고
    • Synthesis, antioxidant activities and urease inhibition of some 1,2,4-triazole and 1,3,4-thiadiazole derivaties
    • I. Khan, Shajid Ali, Shahid Hameed, Naseem Hasan Rama, Muhammed Tahir Hussain, Abdul Wabood, Reazuddin, Zaheer Ul-Haq, Ajmal Khan, and M.C. Iqbal Synthesis, antioxidant activities and urease inhibition of some 1,2,4-triazole and 1,3,4-thiadiazole derivaties Eur J Med Chem 45 2010 5200 5207
    • (2010) Eur J Med Chem , vol.45 , pp. 5200-5207
    • Khan, I.1    Ali, S.2    Hameed, S.3    Rama, N.H.4    Hussain, M.T.5    Wabood, A.6    Reazuddin7    Ul-Haq, Z.8    Khan, A.9    Iqbal, M.C.10
  • 10
    • 80054914442 scopus 로고    scopus 로고
    • Synthesis and biological activity of triazole derivatives as inhibitors of InhA and anti tuberculosis agents
    • M. Christophe, G. Sylvain, L. Christian, R.P. Maria, F. Frederic, I. Cyril, and B. Michel Synthesis and biological activity of triazole derivatives as inhibitors of InhA and anti tuberculosis agents Eur J Med Chem 46 2011 5524 5531
    • (2011) Eur J Med Chem , vol.46 , pp. 5524-5531
    • Christophe, M.1    Sylvain, G.2    Christian, L.3    Maria, R.P.4    Frederic, F.5    Cyril, I.6    Michel, B.7
  • 11
    • 0043158805 scopus 로고    scopus 로고
    • Synthesis characterization and anticancer activity studies on some mannich bases derived from 1,2,4-triazoles
    • B.S. Holla, B. Veerendra, M.K. Shivananda, and B. Poojary Synthesis characterization and anticancer activity studies on some mannich bases derived from 1,2,4-triazoles Eur J Med Chem 38 2003 759 767
    • (2003) Eur J Med Chem , vol.38 , pp. 759-767
    • Holla, B.S.1    Veerendra, B.2    Shivananda, M.K.3    Poojary, B.4
  • 12
    • 34249660531 scopus 로고    scopus 로고
    • Studies on synthesis and pharmacological activities of 3,6-disubstituted-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and their dihydro analogues
    • V. Mathew, J. Keshavayya, V.P. Vaidya, and D. Giles Studies on synthesis and pharmacological activities of 3,6-disubstituted-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and their dihydro analogues Eur J Med Chem 42 2007 823 840
    • (2007) Eur J Med Chem , vol.42 , pp. 823-840
    • Mathew, V.1    Keshavayya, J.2    Vaidya, V.P.3    Giles, D.4
  • 13
    • 0036176817 scopus 로고    scopus 로고
    • Synthesis and anti-inflammatory activity of 1-acylthiosemi-carbazides, 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazole-3-thiones
    • E. Palaska, G. Sahin, P. Kelicen, N.T. Durlu, and G. AltInok Synthesis and anti-inflammatory activity of 1-acylthiosemi-carbazides, 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazole-3-thiones Farmaco 57 2002 101 107
    • (2002) Farmaco , vol.57 , pp. 101-107
    • Palaska, E.1    Sahin, G.2    Kelicen, P.3    Durlu, N.T.4    Altinok, G.5
  • 14
    • 29644434205 scopus 로고    scopus 로고
    • Synthesis and preliminary anticancer activity of new 1H-4,5-dihydro-3-(3-hydroxy-2-naphthyl)-4-substituted-1,2,4-triazoline-5-thiones
    • H.N. Dogan, A. Duran, and S. Rollas Synthesis and preliminary anticancer activity of new 1H-4,5-dihydro-3-(3-hydroxy-2-naphthyl)-4-substituted-1,2,4-triazoline-5-thiones Indian J Chem 44B 2005 2301 2307
    • (2005) Indian J Chem , vol.44 B , pp. 2301-2307
    • Dogan, H.N.1    Duran, A.2    Rollas, S.3
  • 15
    • 84901660465 scopus 로고    scopus 로고
    • Novel compounds containing 1,3,4-oxadiazole and pyrazole-3-one nuclei - Synthesis and antimicrobial evaluation
    • E. Krishna Naik, A. Raghavendra Guru Prasad, Y.N. Spoorthy, and L.K. Ravindranath Novel compounds containing 1,3,4-oxadiazole and pyrazole-3-one nuclei - synthesis and antimicrobial evaluation An R Acad Nac Farm 80 2014 201 213
    • (2014) An R Acad Nac Farm , vol.80 , pp. 201-213
    • Krishna Naik, E.1    Raghavendra Guru Prasad, A.2    Spoorthy, Y.N.3    Ravindranath, L.K.4
  • 18
    • 33947339418 scopus 로고
    • The micro estimation of halogens in organic compounds
    • A. Elek, and D.W. Hill The micro estimation of halogens in organic compounds J Am Chem Soc 55 1933 2550 2554
    • (1933) J Am Chem Soc , vol.55 , pp. 2550-2554
    • Elek, A.1    Hill, D.W.2
  • 19
    • 0034130689 scopus 로고    scopus 로고
    • Comparative evaluation of PASCO and National Committee for Clinical Laboratory Standards M27-A broth micro dilution methods for antifungal drug susceptibility testing of yeasts
    • B.A. Arthington-Skaggs, M. Motley, D.W. Warnock, and C.J. Morrison Comparative evaluation of PASCO and National Committee for Clinical Laboratory Standards M27-A broth micro dilution methods for antifungal drug susceptibility testing of yeasts J Clin Microbiol 38 2000 2254 2260
    • (2000) J Clin Microbiol , vol.38 , pp. 2254-2260
    • Arthington-Skaggs, B.A.1    Motley, M.2    Warnock, D.W.3    Morrison, C.J.4
  • 20
    • 39449086721 scopus 로고    scopus 로고
    • Agar and broth dilution methods to determine the minimal inhibitory concentration (MIC) of antimicrobial substances
    • I. Wiegand, K. Hilpert, and R.E. Hancock Agar and broth dilution methods to determine the minimal inhibitory concentration (MIC) of antimicrobial substances Nat Protoc 3 2008 163 175
    • (2008) Nat Protoc , vol.3 , pp. 163-175
    • Wiegand, I.1    Hilpert, K.2    Hancock, R.E.3
  • 21
    • 84893680300 scopus 로고    scopus 로고
    • Synthesis, evaluation and docking studies on steroidal pyrazolones as anticancer and antimicrobial agents
    • A. Shamsuzzaman, Mashrai, A. Ahmad, A.M. Dar, H. Khanam, M. Danishuddin, and A.U. Khan Synthesis, evaluation and docking studies on steroidal pyrazolones as anticancer and antimicrobial agents Med Chem Res 23 2014 348 362
    • (2014) Med Chem Res , vol.23 , pp. 348-362
    • Shamsuzzaman, A.1    Mashrai2    Ahmad, A.3    Dar, A.M.4    Khanam, H.5    Danishuddin, M.6    Khan, A.U.7
  • 22
    • 0031024171 scopus 로고    scopus 로고
    • Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
    • C.A. Lipinski, F. Lombardo, B.W. Dominy, and P.J. Feeney Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings Adv Drug Deliv Rev 23 1997 3 25
    • (1997) Adv Drug Deliv Rev , vol.23 , pp. 3-25
    • Lipinski, C.A.1    Lombardo, F.2    Dominy, B.W.3    Feeney, P.J.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.