Synthesis, antioxidant activities and urease inhibition of some new 1,2,4-triazole and 1,3,4-thiadiazole derivatives

European Journal of Medicinal Chemistry

Volumn 45, Issue 11, 2010, Pages 5200-5207

  Khan, Imtiaz ^a   Ali, Sajid ^a   Hameed, Shahid ^a   Rama, Nasim Hasan ^a   Hussain, Muhammad Tahir ^b   Wadood, Abdul ^c   Uddin, Reaz ^c   Ul Haq, Zaheer ^c   Khan, Ajmal ^c   Ali, Sajjad ^c   Choudhary, M Iqbal ^c  

^a QUAID I AZAM UNIVERSITY   (Pakistan)

^b NATIONAL TEXTILE UNIVERSITY   (Pakistan)

^c UNIVERSITY OF KARACHI   (Pakistan)

Author keywords

1,2,4 Triazoles; 1,3,4 Thiadiazoles; Antioxidant activities; Urease inhibition

Indexed keywords

4 (2,3 DIMETHYLPHENYL) 5 (2 METHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 4 (2,3 DIMETHYLPHENYL) 5 PHENYL 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 4 (2,4 DIMETHYLPHENYL) 5 (3 NITROPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 4 (2,6 DIMETHYLPHENYL) 5 (4 METHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (2 CHLOROPHENYL) 4 (2,6 DIMETHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (2 CHLOROPHENYL) N (2,6 DIMETHYLPHENYL) 1,3,4 THIADIAZOL 2 AMINE; 5 (3 CHLOROPHENYL) 4 (2,4 DIMETHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (3 CHLOROPHENYL) 4 (2,6 DIMETHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (3 CHLOROPHENYL) N (2,4 DIMETHYLPHENYL) 1,3,4 THIADIAZOL 2 AMINE; 5 (4 CHLOROPHENYL) 4 (2,3 DIMETHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (4 CHLOROPHENYL) 4 (2,4 DIMETHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (4 CHLOROPHENYL) 4 (2,6 DIMETHYLPHENYL) 2,4 DIHYDRO 3H 1,2,4 TRIAZOLE 3 THIONE; 5 (4 CHLOROPHENYL) N (2,3 DIMETHYLPHENYL) 1,3,4 THIADIAZOL 2 AMINE; 5 (4 CHLOROPHENYL) N (2,6 DIMETHYLPHENYL) 1,3,4 THIADIAZOL 2 AMINE; GALLIC ACID PROPYL ESTER; N (2,3 DIMETHYLPHENYL) 5 PHENYL 1,3,4 THIADIAZOL 2 AMINE; N (2,4 DIMETHYLPHENYL) 5 (3 METHYLPHENYL) 1,3,4 THIADIAZOL 2 AMINE; N (2,4 DIMETHYLPHENYL) 5 (4 NITROPHENYL) 1,3,4 THIADIAZOL 2 AMINE; N (2,6 DIMETHYLPHENYL) 5 (4 METHYLPHENYL) 1,3,4 THIADIAZOL 2 AMINE; THIADIAZOLE DERIVATIVE; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG; UREASE;

ANTIOXIDANT ACTIVITY; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; CYCLIZATION; DRUG INHIBITION; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; IC 50; IRRADIATION; MASS SPECTROMETRY; PROTON NUCLEAR MAGNETIC RESONANCE;

ANTIOXIDANTS; INHIBITORY CONCENTRATION 50; MAGNETIC RESONANCE SPECTROSCOPY; SPECTROMETRY, MASS, ELECTROSPRAY IONIZATION; THIADIAZOLES; TRIAZOLES; UREASE;

EID: 77957856848     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2010.08.034     Document Type: Article

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