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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 1, 2015, Pages 70-74

α-Ketoamino acid ester derivatives as promising MAO inhibitors

(6) El Faham, Ayman a,b Al Marhoon, Zainab a Abdel Megeed, Ahmed a,c Khattab, Sherine N b Bekhit, Adnan A d Albericio, Fernando a,e,f,g,h

a KING SAUD UNIVERSITY (Saudi Arabia)

b Alexandria University Faculty Of Science (Egypt)

c ALEXANDRIA UNIVERSITY (Egypt)

d Alexandria University Faculty of Pharmacy (Egypt)

e INSTITUTE FOR RESEARCH IN BIOMEDICINE (Spain)

f UNIVERSITY OF BARCELONA (Spain)

g UNIVERSITY OF KWAZULU NATAL (South Africa)

h YACHAY TECH UNIVERSITY (Ecuador)

Author keywords

Monoamine oxidase inhibitors; N Acetylisatin; OxymaPure; p Aminobenzoic acid; Ketoamino acid ester

Indexed keywords

CLORGYLINE; ESTER DERIVATIVE; MONOAMINE OXIDASE INHIBITOR; AMINO ACID; ESTER; KETONE; PROTEIN BINDING;

ACUTE TOXICITY; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG DESIGN; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; DRUG TOLERABILITY; ENZYME INHIBITION; HYDROGEN BOND; MALE; MOLECULAR DOCKING; MOLECULAR INTERACTION; MOLECULAR MODEL; MOUSE; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; ANIMAL; HUMAN; METABOLISM; PHYSIOLOGY; SYNTHESIS;

AMINO ACIDS; ANIMALS; ESTERS; HUMANS; KETONES; MALE; MICE; MONOAMINE OXIDASE INHIBITORS; PROTEIN BINDING;

EID: 84913582484 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.11.007 Document Type: Article

Times cited : (12)

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