Identification and characterization of an anti-pseudomonal dichlorocarbazol derivative displaying anti-biofilm activity

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 23, 2014, Pages 5404-5408

  Liebens, Veerle ^a   Gerits, Evelien ^a   Knapen, Wouter J ^a   Swings, Toon ^a   Beullens, Serge ^a   Steenackers, Hans P ^a   Robijns, Stijn ^a   Lippell, Anna ^b   O'Neill, Alex J ^b   Veber, Matija ^c   Fröhlich, Mirjam ^c,d   Krona, Annika ^e   Lövenklev, Maria ^e   Corbau, Romu ^f,h   Marchand, Arnaud ^f   Chaltin, Patrick ^a,f   De Brucker, Katrijn ^a   Thevissen, Karin ^a   Cammue, Bruno P ^a,g   Fauvart, Maarten ^a   Verstraeten, Natalie ^a   Michiels, Jan ^a   more..

^a UNIVERSITY OF LEUVEN   (Belgium)

^b UNIVERSITY OF LEEDS   (United Kingdom)

^c Educell   (Slovenia)

^d JO EF STEFAN INSTITUTE   (Slovenia)

^e SIK THE SWEDISH INSTITUTE FOR FOOD AND BIOTECHNOLOGY   (Sweden)

^f CISTIM Leuven Vzw   (Belgium)

^g DEPARTMENT OF PLANT SYSTEMS BIOLOGY   (Belgium)

^h CHILDREN S HOSPITAL OF PHILADELPHIA   (United States)

Author keywords

Biofilm; Carbazoles; Escherichia coli; Porphyromonas gingivalis; Pseudomonas aeruginosa; Staphylococcus aureus; Staphylococcus epidermidis

Indexed keywords

3,6 DIHALOGENOCARBAZOL 1 (SEC BUTYLAMINO) 3 (3,6 DICHLORO 9H CARBAZOL 9 YL)PROPAN 2 OL; ANTIBIOTIC AGENT; CARBAZOLE DERIVATIVE; CEFEPIME; CEFTAZIDIME; CIPROFLOXACIN; GENTAMICIN; OFLOXACIN; PIPERACILLIN; TICARCILLIN; UNCLASSIFIED DRUG; ANTIINFECTIVE AGENT;

ANTIBACTERIAL ACTIVITY; ANTIBIOTIC SENSITIVITY; ANTIBIOTIC THERAPY; ARTICLE; BACTERIOSTASIS; BIOFILM; CONTROLLED STUDY; CYTOTOXICITY; DRUG IDENTIFICATION; ENDOTHELIUM CELL; ESCHERICHIA COLI; HUMAN; HUMAN CELL; MESENCHYMAL STEM CELL; MINIMUM INHIBITORY CONCENTRATION; OSTEOBLAST; PERIODONTITIS; PORPHYROMONAS GINGIVALIS; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS; WILD TYPE; CHEMISTRY; ISOLATION AND PURIFICATION; MICROBIAL SENSITIVITY TEST;

ANTI-BACTERIAL AGENTS; BIOFILMS; CARBAZOLES; HUMANS; MICROBIAL SENSITIVITY TESTS; PSEUDOMONAS AERUGINOSA;

EID: 84910148161     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2014.10.039     Document Type: Article

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