Atovaquone and quinine anti-malarials inhibit ATP binding cassette transporter activity

Malaria Journal

Volumn 13, Issue 1, 2014, Pages

  Rijpma, Sanna R ^a   Van Den Heuvel, Jeroen J M W ^a   Van Der Velden, Maarten ^a   Sauerwein, Robert W ^a   Russel, Frans G M ^a   Koenderink, Jan B ^a  

^a RADBOUD UNIVERSITY MEDICAL CENTER   (Netherlands)

Author keywords

ABC transporter; Anti malarial; BCRP; BSEP; MRP; P glycoprotein; Transport; Vesicle

Indexed keywords

ABC TRANSPORTER; ARTEMISININ; ATOVAQUONE; BENFLUMETOL; BILE SALT EXPORT PUMP; BREAST CANCER RESISTANCE PROTEIN; CHLOROQUINE; DIHYDROARTEMISININ; MEFLOQUINE; MULTIDRUG RESISTANCE PROTEIN; MULTIDRUG RESISTANCE PROTEIN 1; MULTIDRUG RESISTANCE PROTEIN 2; MULTIDRUG RESISTANCE PROTEIN 3; MULTIDRUG RESISTANCE PROTEIN 4; PROGUANIL; QUININE; ANTIMALARIAL AGENT;

ARTICLE; CELL ISOLATION; CONTROLLED STUDY; DRUG BLOOD LEVEL; DRUG EFFECT; DRUG SCREENING; HEK293 CELL LINE; IC50; ISOTOPE LABELING; MEMBRANE VESICLE; NONHUMAN; NUCLEOTIDE SEQUENCE; PROTEIN ANALYSIS; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN INTERACTION; PROTEIN TRANSPORT; ANTAGONISTS AND INHIBITORS; HUMAN;

ANTIMALARIALS; ATOVAQUONE; ATP-BINDING CASSETTE TRANSPORTERS; HEK293 CELLS; HUMANS; P-GLYCOPROTEIN; QUININE;

EID: 84908457958     PISSN: None     EISSN: 14752875     Source Type: Journal    
DOI: 10.1186/1475-2875-13-359     Document Type: Article

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