The intrinsic aqueous solubility of indomethacin

ADMET and DMPK

Volumn 2, Issue 1, 2014, Pages 18-32

  Comer, John ^a   Judge, Sam ^a   Matthews, Darren ^a   Towes, Louise ^a   Falcone, Bruno ^b   Goodman, Jonathan ^b   Dearden, John ^c  

^a Sirius Analytical Ltd   (United Kingdom)

^b UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^c LIVERPOOL JOHN MOORES UNIVERSITY   (United Kingdom)

Author keywords

CheqSol; Decomposition; Indomethacin; P chlorobenzoic acid; Solubility

Indexed keywords

EID: 84905509019     PISSN: None     EISSN: 18487718     Source Type: Journal    
DOI: 10.5599/admet.2.1.33     Document Type: Article

References (44)

1. H. Yamamoto. Chem. Pharm. Bull. 16(1) (1968) 17-19.
2. L. Borka. Acta Pharm. Suecica. 11(3) (1974) 295-303.
3. S-Y Lin. J Pharm Sci. 81(6) (1992) 572-576.
4. N. Kaneniwa, M. Otsuka, T. Hayashi. Chem. Pharm. Bull. 33(8) (1985) 3447-3455.
5. V. Andronis, G. Zografi. J. Non-Cryst. Solids. 271(3) (2000) 236-248.
6. J.M. Aceves-Hernandez, I. Nicolás-Vázquez, F.J. Aceves, J. Hinojosa-Torres, M. Paz, V.M. Castaño. J. Pharm. Sci. 98(7) (2009) 2448-2463.
7. C. Aubrey-Medendorp, M.J. Swadley, T. Li. Pharm. Res. 25(4) (2008) 953-959.
8. N. Hamdi, Y. Feutelais, N. Yagoubi, D. de Girolamo, B. Legendre. J. Therm. Anal. Cal. 76 (2004) 985-1001.
9. B.C. Hancock, M. Parks. Pharm. Res. 17(4) (2000) 397-403.
10. S.B. Murdande, M.J. Pikal, R.M. Shanker, R.H. Bogner. J. Pharm. Sci. 99(3) (2010) 1254-1264.
11. D. Iohara, F. Hirayama, T. Ishiguro, H. Arima, K. Uekama. Int. J. Pharm. 354(1-2) (2008) 70-76.
12. M. Otsuka, T. Matsumoto, N. Kaneniwa. Chem. Pharm. Bull. 34(4) (1986) 1784-1793.
13. A. Rezaei Mokarram, A. Kebriaee Zadeh, M. Keshavarz, A. Ahmadi, B. Mohtat. DARU J. Pharm Sci. 18(3) (2010) 185-192.
14. T. Ito, T. Sugafuji, M. Maruyama, Y. Ohwa, T. Takahashi. J. Supramol. Chem. 1(4-6) (2001) 217-219.
15. O.A. Deshpande, V.B. Yadav. Int. J. Chem.Tech. Res. 1(4) (2009) 1312-1317.
16. S.H. Yalkowsky, R.M. Dannenfelser. AQUASOL Database of Aqueous Solubility, version 5, College of Pharmacy, University of Arizona, Tucson, AZ, USA, 1992.
17. F. Martínez, M.A. Peña, P. Bustamante. Fluid Phase Equilib. 308(1-2) (2011) 98-106.
18. A. Nokhodchi. J. Pharm. Pharmaceu.t Sci. 8(1) (2005) 18-25.
19. C.A.S. Bergström, M. Strafford, L. Lazorova, A. Avdeef, K. Luthman, P. Artursson. J. Med. Chem. 46(4) (2003) 558-570.
20. S. Muchtar, M. Abdulrazik, J. Frucht-Pery, S. Benita. J. Control. Release 44(1) (1997) 55-64.
21. S. Jambhekar, R. Casella, T. Maher. Int. J. Pharm. 270(1-2) (2004) 149-166.
22. R. Bodmeier, H. Chen. J. Control. Release. 12(3) (1990) 223-233.
23. M. Hewitt, M.T. Cronin, S.J. Enoch, J.C. Madden, D.W. Roberts, J.C. Dearden. J. Chem. Inf. Model. 49(11) (2009) 2572-87.
24. A. Llinas, R.C. Glen, J.M. Goodman. J. Chem. Inf. Model. 48(7) (2008) 1289-303.
25. A.J. Hopfinger, E.X. Esposito, A. Llinàs, R.C. Glen, J.M. Goodman. J. Chem. Inf. Model. 49(1) (2009) 1-5.
26. M. Stuart, K. Box. Anal. Chem. 77(4) (2005) 983-990.
27. K.J. Box, G. Völgyi, E. Baka, M. Stuart, K. Takács-Novák, J.E.A. Comer. J. Pharm. Sci. 95(6) (2006) 1298-1307.
28. K. Box, J.E. Comer, T. Gravestock, M. Stuart. Chem. Biodiversity 6(11) (2009) 1767-1788.
29. A. Fini, G. Fazio, G. Feroci. Int. J. Pharm. 126 (1995) 95-102.
30. M. Shalaeva, J. Kenseth, F. Lombardo, A. Bastin, A. J. Pharm. Sci. 97(7) (2008) 2581-2606.
31. K.G. Mooney, M.A. Mintun, K.J. Himmelstein, V.J. Stella. J. Pharm. Sci. 70(1) (1981) 13-22.
32. B. Tsvetkova, I. Pencheva, A. Zlatkov, P. Peikov. Int. J. Pharm. Sci. 4(Supplement 3) (2012) 549.
33. S.A. Raina, G.Z. Zhang, D.E. Alonzo, J. Wu,D. Zhu,N.D. Catron, Y. Gao, L.S. Taylor. J. Pharm. Sci. 2014, DOI: 10.1002/jps.23826
34. A. Avdeef. Pharm. Pharmacol. Commun. 4 (1998) 165-178.
35. M.Z. Southard, D.W. Green, V.J. Stella, K.J. Himmelstein. Pharm. Res. 9(1) (1992) 58-69.
36. K. Okimoto, R.A. Rajewski, K. Uekama, J.A. Jona, V.J. Stella. Pharm. Res. 13(2) (1996) 256-64.
37. C.M. Wassvik, A.G. Holmen, C.A. Bergstrom, I. Zamora, P. Artursson. Eur. J. Pharm. Sci. 29(3-4) (2006) 294-305.
38. J.H. Fagerberg, O. Tsinman, N. Sun, K. Tsinman, A. Avdeef, C.A. Bergstrom. Mol. Pharm. 7(5) (2010) 1419-30.
39. Simulations Plus, Inc. 42505 10th Street West Lancaster, CA 93534, USA. http://www.simulations-plus.com/
40. StarDrop: Optibrium Ltd. 7221 Cambridge Research Park Beach Drive Cambridge CB25 9TL, UK. http://www.optibrium.com/starvue/index.php
41. CSlogWS: ChemSilico LLC, 48 Baldwin St. Tewksbury, MA 01876, USA. http://www.chemsilico.com/
42. ALOGPS: I.V. Tetko, J. Gasteiger, R. Todeschini, A. Mauri, D. Livingstone, P. Ertl, V.A. Palyulin, E.V. Radchenko, N.S. Zefirov, A.S. Makarenko, V.Y. Tanchuk, V.V. Prokopenko. J. Comput. Aid. Mol. Des 19 (2005) 453-463.
43. WSKOWWIN: http://www.epa.gov/oppt/exposure/pubs/episuite.htm
44. WATERNT: http://www.epa.gov/oppt/exposure/pubs/episuite.htm