Electronic sculpting of ligand-GPCR subtype selectivity: The case of angiotensin II

ACS Chemical Biology

Volumn 9, Issue 7, 2014, Pages 1420-1425

  Magnani, Francesca ^a,h   Pappas, Charalampos G ^b   Crook, Tim ^c   Magafa, Vassiliki ^d   Cordopatis, Paul ^d   Ishiguro, Susumu ^e   Ohta, Naomi ^e   Selent, Jana ^f   Bosnyak, Sanja ^g   Jones, Emma S ^g   Gerothanassis, Ioannis P ^b   Tamura, Masaaki ^c   Widdop, Robert E ^g   Tzakos, Andreas G ^b  

^a MRC LABORATORY OF MOLECULAR BIOLOGY   (United Kingdom)

^b UNIVERSITY OF IOANNINA   (Greece)

^c UNIVERSITY OF DUNDEE   (United Kingdom)

^d UNIVERSITY OF PATRAS   (Greece)

^e KANSAS STATE UNIVERSITY   (United States)

^f UNIVERSITAT POMPEU FABRA   (Spain)

^g MONASH UNIVERSITY   (Australia)

^h UNIVERSITY OF PAVIA   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

ANGIOTENSIN 1 RECEPTOR; ANGIOTENSIN 2 RECEPTOR; ANGIOTENSIN II; G PROTEIN COUPLED RECEPTOR; ANTINEOPLASTIC AGENT; LIGAND;

ARTICLE; BREAST CARCINOMA; CELL PROLIFERATION; CONFORMATION; CONTROLLED STUDY; DRUG SELECTIVITY; IC 50; ISOMERIZATION; LIGAND BINDING; NERVE FIBER GROWTH; PHENOTYPE; PRIORITY JOURNAL; PROTEIN DATABASE; SEQUENCE ALIGNMENT; SIGNAL TRANSDUCTION; AGONISTS; ANALOGS AND DERIVATIVES; BREAST NEOPLASMS; CHEMISTRY; DRUG DESIGN; DRUG EFFECTS; FEMALE; HUMAN; METABOLISM; MOLECULAR DOCKING; TUMOR CELL LINE;

ANGIOTENSIN II; ANTINEOPLASTIC AGENTS; BREAST NEOPLASMS; CELL LINE, TUMOR; CELL PROLIFERATION; DRUG DESIGN; FEMALE; HUMANS; LIGANDS; MOLECULAR DOCKING SIMULATION; RECEPTOR, ANGIOTENSIN, TYPE 1; RECEPTOR, ANGIOTENSIN, TYPE 2;

EID: 84904577699     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb500063y     Document Type: Article

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