Promising potential of new generation translocator protein tracers providing enhanced contrast of arthritis imaging by positron emission tomography in a rat model of arthritis

Arthritis Research and Therapy

Volumn 16, Issue 2, 2014, Pages

  Gent, Yoony Y J ^a   Weijers, Karin ^a   Molthoff, Carla F M ^a   Windhorst, Albert D ^a   Huisman, Marc C ^a   Kassiou, Michael ^b,c   Jansen, Gerrit ^a   Lammertsma, Adriaan A ^a   Van der Laken, Conny J ^a  

^a VU UNIVERSITY MEDICAL CENTER   (Netherlands)

^b UNIVERSITY OF SYDNEY   (Australia)

^c UNIVERSITY OF SYDNEY   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

CARRIER PROTEIN; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; N,N DIETHY 2 [2 [4 (2 FLUOROETHOXY)PHENYL] 5,7 DIMETHYLPYRAZOLO[1,5-A]PYRIMIDIN 3 YL] ACETAMIDE F 18; N,N DIETHYL 2 (4 METHOXYPHENYL) 5,7 DIMETHYLPYRAZOLO[1,5 A]PYRIMIDINE 3 ACETAMIDE C 11; TRACER; UNCLASSIFIED DRUG; ACETAMIDES; BZRP PROTEIN, RAT; CARBON RADIOISOTOPES; CARRIER PROTEINS; FLUORINE RADIOISOTOPES; N,N-DIETHYL-2-(2-(4-(2-FLUOROETHOXY)PHENYL)-5,7-DIMETHYLPYRAZOLO(1,5-A)PYRIMIDIN-3-YL)ACETAMIDE; N,N-DIETHYL-2-(2-(4-METHOXYPHENYL)-5,7-DIMETHYL-PYRAZOLO(1,5-A)PYRIMIDIN-3-YL)-ACETAMIDE; PYRAZOLES; PYRIMIDINES; RADIOPHARMACEUTICALS; RECEPTORS, GABA-A;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTHRITIS; ARTICLE; BINDING COMPETITION; BONE MARROW; CONTRAST ENHANCEMENT; CONTROLLED STUDY; DRUG UPTAKE; EX VIVO STUDY; HEART; HUMAN; HUMAN CELL; IMMUNOHISTOCHEMISTRY; IN VITRO STUDY; IN VIVO STUDY; INFLAMMATORY CELL; INTESTINE; KIDNEY; LUNG; MALE; MONOCYTE; NONHUMAN; PET SCANNER; POSITRON EMISSION TOMOGRAPHY; RAT; SPLEEN; TISSUE DISTRIBUTION; ANIMALS; ARTHRITIS, EXPERIMENTAL; ARTHRITIS, RHEUMATOID; DIAGNOSTIC USE; HUMANS; METABOLISM; METHODS; POSITRON-EMISSION TOMOGRAPHY; RADIONUCLIDE IMAGING; RATS;

ACETAMIDES; ANIMALS; ARTHRITIS, EXPERIMENTAL; ARTHRITIS, RHEUMATOID; CARBON RADIOISOTOPES; CARRIER PROTEINS; FLUORINE RADIOISOTOPES; HUMANS; POSITRON-EMISSION TOMOGRAPHY; PYRAZOLES; PYRIMIDINES; RADIOPHARMACEUTICALS; RATS; RECEPTORS, GABA-A;

EID: 84897555411     PISSN: 14786354     EISSN: 14786362     Source Type: Journal    
DOI: 10.1186/ar4509     Document Type: Article

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