Development of purine-derived 18F-labeled pro-drug tracers for imaging of MRP1 activity with PET

Journal of Medicinal Chemistry

Volumn 57, Issue 3, 2014, Pages 1023-1032

  Galante, Eva ^a   Okamura, Toshimitsu ^b   Sander, Kerstin ^a   Kikuchi, Tatsuya ^b   Okada, Maki ^b   Zhang, Ming Rong ^b   Robson, Mathew ^c   Badar, Adam ^c   Lythgoe, Mark ^c   Koepp, Matthias ^d   Årstad, Erik ^a  

^a UNIVERSITY COLLEGE LONDON   (United Kingdom)

^b NATIONAL INSTITUTE OF RADIOLOGICAL SCIENCES   (Japan)

^c UNIVERSITY COLLEGE LONDON   (United Kingdom)

^d UNIVERSITY COLLEGE LONDON   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

FLUORINE; MULTIDRUG RESISTANCE ASSOCIATED PROTEIN 1; MULTIDRUG RESISTANCE PROTEIN; MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 1; PRODRUG; PURINE DERIVATIVE; RADIOPHARMACEUTICAL AGENT;

ANIMAL; ARTICLE; BAGG ALBINO MOUSE; BRAIN; CHEMISTRY; GENETICS; KNOCKOUT MOUSE; METABOLISM; MOUSE; POSITRON EMISSION TOMOGRAPHY; SCINTISCANNING; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TISSUE DISTRIBUTION;

ANIMALS; BRAIN; FLUORINE RADIOISOTOPES; MICE; MICE, INBRED BALB C; MICE, KNOCKOUT; MULTIDRUG RESISTANCE-ASSOCIATED PROTEINS; POSITRON-EMISSION TOMOGRAPHY; PRODRUGS; PURINES; RADIOPHARMACEUTICALS; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE DISTRIBUTION;

EID: 84894047141     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm401764a     Document Type: Article

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