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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 2, 2014, Pages 586-590

Synthesis, anticancer activity and DNA-binding properties of novel 4-pyrazolyl-1,8-naphthalimide derivatives

(9) Li, Shenghui a Xu, Shengjie a Tang, Yonghe a Ding, Shan a Zhang, Jinchao a Wang, Shuxiang a Zhou, Guoqiang a Zhou, Chuanqi a Li, Xiaoliu a

a HEBEI UNIVERSITY (China)

Author keywords

Anticancer; DNA binding; Naphthalimides; Pyrazole

Indexed keywords

4 PYRAZOLYL 1,8 NAPHTHALIMIDE DERIVATIVE; AMONAFIDE; NAPHTHALIMIDE DERIVATIVE; UNCLASSIFIED DRUG; ANTINEOPLASTIC AGENT;

ANTINEOPLASTIC ACTIVITY; ARTICLE; BINDING AFFINITY; CANCER CELL; CIRCULAR DICHROISM; CONTROLLED STUDY; CYTOTOXICITY; DENATURATION; DNA BINDING; DRUG SYNTHESIS; FLUORESCENCE SPECTROSCOPY; HUMAN; HUMAN CELL; LUNG CANCER; ULTRAVIOLET SPECTROSCOPY; UTERINE CERVIX CARCINOMA; BREAST CANCER; DRUG STRUCTURE; FLUORESCENCE; IC50; IN VITRO STUDY;

ANTICANCER; DNA-BINDING; NAPHTHALIMIDES; PYRAZOLE;

ANIMALS; ANTINEOPLASTIC AGENTS; CATTLE; DNA; DRUG SCREENING ASSAYS, ANTITUMOR; HELA CELLS; HUMANS; INTERCALATING AGENTS; MCF-7 CELLS; NAPHTHALIMIDES; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84891887724 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.12.014 Document Type: Article

Times cited : (39)

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