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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 2, 2014, Pages 476-479

Synthesis and evaluation of isoleucine derived angiotensin II AT 2 receptor ligands

(5) Veron, Jean Baptiste a Joshi, Advait a Wallinder, Charlotta a Larhed, Mats a Odell, Luke R a

a UPPSALA UNIVERSITY (Sweden)

Author keywords

Angiotensin; AT1 receptor; AT2 receptor; Isoleucine

Indexed keywords

ANGIOTENSIN 2 RECEPTOR; ANGIOTENSIN 2 RECEPTOR ANTAGONIST; ISOLEUCINE; LEAD; ANGIOTENSIN RECEPTOR; HORMONE RECEPTOR AFFECTING AGENT; LIGAND;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG DESIGN; DRUG POTENCY; DRUG PROTEIN BINDING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HYDROPHOBICITY; NONHUMAN; SUBSTITUTION REACTION; BINDING ASSAY; BROMINATION; CARBOXY TERMINAL SEQUENCE; CYCLOADDITION; HEK293 CELL LINE; HYDROGEN BOND; HYDROLYSIS; NUCLEOPHILICITY; REDUCTION;

ANGIOTENSIN; AT(1) RECEPTOR; AT(2) RECEPTOR; ISOLEUCINE;

ANIMALS; DRUG EVALUATION, PRECLINICAL; HEK293 CELLS; HUMANS; ISOLEUCINE; LIGANDS; OLIGOPEPTIDES; PROTEIN BINDING; RECEPTOR, ANGIOTENSIN, TYPE 2; SWINE;

EID: 84891878190 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.12.040 Document Type: Article

Times cited : (6)

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