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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 20, 2013, Pages 5578-5585

A Casein kinase 1/Checkpoint kinase 1 pyrazolo-pyridine protein kinase inhibitor as novel activator of the p53 pathway

(9) Huart, Anne Sophie a Saxty, Barbara b Merritt, Andy b Nekulova, Marta c Lewis, Stephen b Huang, Yide d Vojtesek, Borivoj c Kettleborough, Catherine b Hupp, Ted R a

a UNIVERSITY OF EDINBURGH (United Kingdom)

b MEDICAL RESEARCH COUNCIL (United Kingdom)

c MASARYK MEMORIAL CANCER INSTITUTE (Czech Republic)

d FUJIAN NORMAL UNIVERSITY (China)

Author keywords

Casein kinase 1; Checkpoint kinase 1; Kinase inhibitor; p53 Pathway activation

Indexed keywords

CASEIN KINASE I; CHECKPOINT KINASE 1; D 4476; MRT 00033659; MRT 00033680; MRT 00055778; PROTEIN KINASE INHIBITOR; PROTEIN P53; PYRAZOLE DERIVATIVE; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BIOLOGICAL ACTIVITY; CELL DEATH; CELL VIABILITY; COMPARATIVE STUDY; CONTROLLED STUDY; DRUG SOLUBILITY; FLUORESCENCE ACTIVATED CELL SORTING; HUMAN; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SIGNAL TRANSDUCTION;

CASEIN KINASE 1; CHECKPOINT KINASE 1; KINASE INHIBITOR; P53 PATHWAY ACTIVATION;

CASEIN KINASE I; CELL CYCLE CHECKPOINTS; CELL LINE; CELL SURVIVAL; HCT116 CELLS; HUMANS; KINETICS; PROTEIN KINASE INHIBITORS; PROTEIN KINASES; PYRAZOLES; PYRIDINES; RNA INTERFERENCE; RNA, SMALL INTERFERING; TUMOR SUPPRESSOR PROTEIN P53;

EID: 84884286856 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.08.046 Document Type: Article

Times cited : (13)

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