-
1
-
-
57649202225
-
Synthesis and antimicrobial activity of some new quinazolin-4(3H)-one derivatives
-
Alafeefy A.M. Synthesis and antimicrobial activity of some new quinazolin-4(3H)-one derivatives. Pharm. Biol. 2008, 46(10):751-756.
-
(2008)
Pharm. Biol.
, vol.46
, Issue.10
, pp. 751-756
-
-
Alafeefy, A.M.1
-
2
-
-
0034678644
-
4-Thiazolidinones: novel inhibitors of the bacterial enzyme MurB
-
Andres C.J., Bronson J.J., D'Andrea S.V., Deshpande M.S., Falk P.J., Grant-Young K.A., Harte W.E., Ho H., Misco P.F., Robertson J.G., Stock D., Sun Y., Walsh A.W. 4-Thiazolidinones: novel inhibitors of the bacterial enzyme MurB. Bioorg. Med. Chem. Lett. 2000, 10:715-717.
-
(2000)
Bioorg. Med. Chem. Lett.
, vol.10
, pp. 715-717
-
-
Andres, C.J.1
Bronson, J.J.2
D'Andrea, S.V.3
Deshpande, M.S.4
Falk, P.J.5
Grant-Young, K.A.6
Harte, W.E.7
Ho, H.8
Misco, P.F.9
Robertson, J.G.10
Stock, D.11
Sun, Y.12
Walsh, A.W.13
-
3
-
-
0035821593
-
2-(2-Oxo-1,4-dihydro-2H-quinazoli-3-yl)- and 2-(2,2-dioxo-1,4-dihydro-2H-6 benzo[1,2,6]thiadiazin-3-yl)-N-hydroxy-acetamides as potent and selective peptide deformylase inhibitors
-
Apfel C., Banner D.W., Bur D., Dietz M., Hubschwerlen C., Locher H., Marlin F., Masciadri R., Pirson W., Stalder H. 2-(2-Oxo-1,4-dihydro-2H-quinazoli-3-yl)- and 2-(2,2-dioxo-1,4-dihydro-2H-6 benzo[1,2,6]thiadiazin-3-yl)-N-hydroxy-acetamides as potent and selective peptide deformylase inhibitors. J. Med. Chem. 2001, 44:1847-1852.
-
(2001)
J. Med. Chem.
, vol.44
, pp. 1847-1852
-
-
Apfel, C.1
Banner, D.W.2
Bur, D.3
Dietz, M.4
Hubschwerlen, C.5
Locher, H.6
Marlin, F.7
Masciadri, R.8
Pirson, W.9
Stalder, H.10
-
4
-
-
0038166643
-
Comparison of Staphylococcus spp. cellular and extracellular proteins
-
Berber I., Cokmus C., Atalan E. Comparison of Staphylococcus spp. cellular and extracellular proteins. Mikrobiologia 2003, 72:54-59.
-
(2003)
Mikrobiologia
, vol.72
, pp. 54-59
-
-
Berber, I.1
Cokmus, C.2
Atalan, E.3
-
5
-
-
0035043010
-
The chemical and biological aspects of fluoroquinolones: reality and dreams
-
Bhanot S.K., Singh M., Chaterjee N.R. The chemical and biological aspects of fluoroquinolones: reality and dreams. Curr. Pharm. Des. 2001, 7:311-335.
-
(2001)
Curr. Pharm. Des.
, vol.7
, pp. 311-335
-
-
Bhanot, S.K.1
Singh, M.2
Chaterjee, N.R.3
-
6
-
-
0344689962
-
Researches on quinazolines (Twenty-second paper). On 2-methyl-3-amino-4-quinazolone and certain of its derivatives
-
Bogert M.T., Coriner R.A. Researches on quinazolines (Twenty-second paper). On 2-methyl-3-amino-4-quinazolone and certain of its derivatives. J. Am. Chem. Soc. 1909, 31:943-947.
-
(1909)
J. Am. Chem. Soc.
, vol.31
, pp. 943-947
-
-
Bogert, M.T.1
Coriner, R.A.2
-
7
-
-
1842503232
-
Daptomycin: another novel agent for treating infections due to drug-resistant grampositive pathogens
-
Carpenter C.F., Champers H.F. Daptomycin: another novel agent for treating infections due to drug-resistant grampositive pathogens. Clin. Infect. Dis. 2004, 38:994-1000.
-
(2004)
Clin. Infect. Dis.
, vol.38
, pp. 994-1000
-
-
Carpenter, C.F.1
Champers, H.F.2
-
8
-
-
33846932835
-
Therapeutic and prophylactic potential of small interfering RNAs against severe acute respiratory syndrome: progress to date
-
Chang Z., Babiuk L.A., Hu J. Therapeutic and prophylactic potential of small interfering RNAs against severe acute respiratory syndrome: progress to date. Bio. Drugs 2007, 21:9-15.
-
(2007)
Bio. Drugs
, vol.21
, pp. 9-15
-
-
Chang, Z.1
Babiuk, L.A.2
Hu, J.3
-
9
-
-
0035829416
-
New pyridoquinoline derivatives as potential inhibitors of the fluoroquinolone efflux pump in resistant Enterobacter aerogenes strains
-
Chevalier J., Atifi S., Eyraud A., Mahamoud A., Barbe J., Pajes J. New pyridoquinoline derivatives as potential inhibitors of the fluoroquinolone efflux pump in resistant Enterobacter aerogenes strains. J. Med. Chem. 2001, 44:4023-4026.
-
(2001)
J. Med. Chem.
, vol.44
, pp. 4023-4026
-
-
Chevalier, J.1
Atifi, S.2
Eyraud, A.3
Mahamoud, A.4
Barbe, J.5
Pajes, J.6
-
10
-
-
0035942523
-
Quinazolin-4-one a-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor antagonists: structure-activity relationship of the C-2 side chain tether
-
Chenard B.L., Welch W.M., Blake J.F., Butler T.W., Reinhold A., Ewing F.E., Menniti F.S., Pagnozzi M.J. Quinazolin-4-one a-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor antagonists: structure-activity relationship of the C-2 side chain tether. J. Med. Chem. 2001, 44:1710-1717.
-
(2001)
J. Med. Chem.
, vol.44
, pp. 1710-1717
-
-
Chenard, B.L.1
Welch, W.M.2
Blake, J.F.3
Butler, T.W.4
Reinhold, A.5
Ewing, F.E.6
Menniti, F.S.7
Pagnozzi, M.J.8
-
11
-
-
3042588256
-
DNA binding to guide the development of tetrahydroindeno[1,2-b]pyrido[4,3,2-de]quinoline derivatives as cytotoxic agents
-
Ctoen-Chackal S., Facompre M., Houssin R., Pommery N., Gossens J.F., Colson P., Bailly C., Henichart J.P. DNA binding to guide the development of tetrahydroindeno[1,2-b]pyrido[4,3,2-de]quinoline derivatives as cytotoxic agents. J. Med. Chem. 2004, 47(14):3665-3673.
-
(2004)
J. Med. Chem.
, vol.47
, Issue.14
, pp. 3665-3673
-
-
Ctoen-Chackal, S.1
Facompre, M.2
Houssin, R.3
Pommery, N.4
Gossens, J.F.5
Colson, P.6
Bailly, C.7
Henichart, J.P.8
-
12
-
-
0026023327
-
Synthesis and anticonvulsant activity o imidooxy derivatives
-
Edafiogho I.O., Scott K.R., Moore J.A., Farrar Y.A., Nicholson J.M. Synthesis and anticonvulsant activity o imidooxy derivatives. J. Med. Chem. 1991, 34:387-392.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 387-392
-
-
Edafiogho, I.O.1
Scott, K.R.2
Moore, J.A.3
Farrar, Y.A.4
Nicholson, J.M.5
-
13
-
-
33646584802
-
Structural features of new quinolones and relationship to antibacterial activity against gram-positive bacteria
-
Emami S., Shafiee A., Alireza F. Structural features of new quinolones and relationship to antibacterial activity against gram-positive bacteria. Mini Rev. Med. Chem. 2006, 6:375-386.
-
(2006)
Mini Rev. Med. Chem.
, vol.6
, pp. 375-386
-
-
Emami, S.1
Shafiee, A.2
Alireza, F.3
-
14
-
-
0027145572
-
Synthesis and calculated log P correlation of imidooxy anticonvulsants
-
Farror Y.A., Rutkowaka M.C., Grochowski J., Serda P., Pilati T., Cory M., Nicholson J.M., Scott K.R. Synthesis and calculated log P correlation of imidooxy anticonvulsants. J. Med. Chem. 1993, 36:3517-3525.
-
(1993)
J. Med. Chem.
, vol.36
, pp. 3517-3525
-
-
Farror, Y.A.1
Rutkowaka, M.C.2
Grochowski, J.3
Serda, P.4
Pilati, T.5
Cory, M.6
Nicholson, J.M.7
Scott, K.R.8
-
16
-
-
34247326968
-
Synthesis and antifungal activity of novel S-substituted 6-fluoro-4-alkyl(aryl)thioquinazoline derivatives
-
Guang-Fang X., Bao-An S., Pinaki S.B., Song Y., Pei-Quan Z., Lin-Hong J., Wei X., De-Yu H., Ping L. Synthesis and antifungal activity of novel S-substituted 6-fluoro-4-alkyl(aryl)thioquinazoline derivatives. Bioorg. Med. Chem. 2007, 15:3768-3774.
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 3768-3774
-
-
Guang-Fang, X.1
Bao-An, S.2
Pinaki, S.B.3
Song, Y.4
Pei-Quan, Z.5
Lin-Hong, J.6
Wei, X.7
De-Yu, H.8
Ping, L.9
-
17
-
-
46249096760
-
Synthesis and antimicrobial evaluation of some novel imidazolylmercaptoacetylthiosemicarbazide and 4-thiazolidinone analogs
-
Gursoy A., Otuk G., Terzioglu N. Synthesis and antimicrobial evaluation of some novel imidazolylmercaptoacetylthiosemicarbazide and 4-thiazolidinone analogs. Turkish J. Pharm. Sci. 2005, 2:1-10.
-
(2005)
Turkish J. Pharm. Sci.
, vol.2
, pp. 1-10
-
-
Gursoy, A.1
Otuk, G.2
Terzioglu, N.3
-
18
-
-
0003495102
-
Goodman and Gilman's
-
Springer
-
Hardman J.G., Limbird E.L., Molinoff P.B., Ruddon R.W., Gilman A.G. Goodman and Gilman's. The Pharmacological Basis of Therapeutics 2002, Springer, p. 1065. ninth ed.
-
(2002)
The Pharmacological Basis of Therapeutics
, pp. 1065
-
-
Hardman, J.G.1
Limbird, E.L.2
Molinoff, P.B.3
Ruddon, R.W.4
Gilman, A.G.5
-
21
-
-
77950299185
-
Design, synthesis and antibiofilm activity of 2-arylimino-3-aryl-thiazolidine-4-ones
-
Pan B., Huang R.Z., Ying H.J. Design, synthesis and antibiofilm activity of 2-arylimino-3-aryl-thiazolidine-4-ones. Bioorg. Med. Chem. Lett. 2010, 20:2461-2464.
-
(2010)
Bioorg. Med. Chem. Lett.
, vol.20
, pp. 2461-2464
-
-
Pan, B.1
Huang, R.Z.2
Ying, H.J.3
-
22
-
-
0033029184
-
Synthesis of new 3-(3-phenyl-isoxazo-5-yl) or 3-[(3-phenylisoxazol-5-yl)-amino]-substituted 4(3H)quinazoli- none derivatives with antineoplastic activity
-
Raffa D., Daidone G., Schillaci D., Maggio B., Plescia F. Synthesis of new 3-(3-phenyl-isoxazo-5-yl) or 3-[(3-phenylisoxazol-5-yl)-amino]-substituted 4(3H)quinazoli- none derivatives with antineoplastic activity. Pharmazie 1999, 54:251-254.
-
(1999)
Pharmazie
, vol.54
, pp. 251-254
-
-
Raffa, D.1
Daidone, G.2
Schillaci, D.3
Maggio, B.4
Plescia, F.5
-
23
-
-
2942690036
-
Microwave-assisted synthesis of benzimidazole and thiazolidinone derivatives as HIV-1 RT inhibitors
-
Rao A., Zappala M. Microwave-assisted synthesis of benzimidazole and thiazolidinone derivatives as HIV-1 RT inhibitors. Arkivoc 1999, v:147-155.
-
(1999)
Arkivoc
, vol.5
, pp. 147-155
-
-
Rao, A.1
Zappala, M.2
-
24
-
-
70349253477
-
-
Churchill, B.I., Livingstone, New Delhi
-
Rattan A. Antimicrobials in laboratory medicine 2000, Churchill, B.I., Livingstone, New Delhi, pp. 85-105.
-
(2000)
Antimicrobials in laboratory medicine
, pp. 85-105
-
-
Rattan, A.1
-
25
-
-
31544467289
-
Synthesis of some new 2,3-diaryl-1,3-thiazolidin-4-ones as antibacterial agents
-
Sayyed M., Mokle S. Synthesis of some new 2,3-diaryl-1,3-thiazolidin-4-ones as antibacterial agents. Arkivoc 2006, ii:187-192.
-
(2006)
Arkivoc
, vol.2
, pp. 187-192
-
-
Sayyed, M.1
Mokle, S.2
-
26
-
-
42049117506
-
Synthesis, characterization and antimicrobial studies of 3-[(2-hydroxy-quinolin-3-ylmethylene)-amino]-2-phenyl-3H-quinazolin-4-one and its Metal(II) complexes
-
Siddappa K., Reddy K., Reddy C.V. Synthesis, characterization and antimicrobial studies of 3-[(2-hydroxy-quinolin-3-ylmethylene)-amino]-2-phenyl-3H-quinazolin-4-one and its Metal(II) complexes. E-J. chem. 2008, 5:155-162.
-
(2008)
E-J. chem.
, vol.5
, pp. 155-162
-
-
Siddappa, K.1
Reddy, K.2
Reddy, C.V.3
-
27
-
-
24544435741
-
4-Thiazolidones. IV. The preparation of some 3-alkylaminoalkyl-2-aryl derivatives
-
Surrey A.R. 4-Thiazolidones. IV. The preparation of some 3-alkylaminoalkyl-2-aryl derivatives. J. Am. Chem. Soc. 1949, 71:3354-3356.
-
(1949)
J. Am. Chem. Soc.
, vol.71
, pp. 3354-3356
-
-
Surrey, A.R.1
-
28
-
-
33846897468
-
Structure activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitors
-
Taun P.T., Edmund L.E., Joseph P.S., Brian M.W., Michael A.S., Hollis S., John M.D., Martin A.S., Themis J., Stephen J.G., Dai Q.N., Paul B., Judy Y., Anurag S., Chan H., Saeed R., Xiujuan W., Rajeshwar S. Structure activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitors. Bioorg. Med. Chem. Lett. 2007, 17:1312-1320.
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 1312-1320
-
-
Taun, P.T.1
Edmund, L.E.2
Joseph, P.S.3
Brian, M.W.4
Michael, A.S.5
Hollis, S.6
John, M.D.7
Martin, A.S.8
Themis, J.9
Stephen, J.G.10
Dai, Q.N.11
Paul, B.12
Judy, Y.13
Anurag, S.14
Chan, H.15
Saeed, R.16
Xiujuan, W.17
Rajeshwar, S.18
-
29
-
-
0000058354
-
The Synthesis of 2,3-disubstituted-4-thiazolidones
-
Troutman H.D., Long L.M. The Synthesis of 2,3-disubstituted-4-thiazolidones. J. Am. Chem. Soc. 1948, 70:3436-3439.
-
(1948)
J. Am. Chem. Soc.
, vol.70
, pp. 3436-3439
-
-
Troutman, H.D.1
Long, L.M.2
-
30
-
-
0037251953
-
Structure-activity relationships of 6-fluoroquinazolines: dual-acting compounds with inhibitory activities toward both TNF alpha production and T cell proliferation
-
Tobe M., Isobe Y., Tomizawa H., Nagasaki T., Obara F., Hayashi H. Structure-activity relationships of 6-fluoroquinazolines: dual-acting compounds with inhibitory activities toward both TNF alpha production and T cell proliferation. Bioorg. Med. Chem. 2003, 11:609-616.
-
(2003)
Bioorg. Med. Chem.
, vol.11
, pp. 609-616
-
-
Tobe, M.1
Isobe, Y.2
Tomizawa, H.3
Nagasaki, T.4
Obara, F.5
Hayashi, H.6
-
31
-
-
19544369670
-
Linzolid versus vancomycin in treatment of complicated skin and soft tissue infections
-
Weigelt J., Itani K., Stevens D., Lau W., Dryden M., Knirsch C. Linzolid versus vancomycin in treatment of complicated skin and soft tissue infections. Antimicrob. Agents Chemother. 2005, 49:2260-2266.
-
(2005)
Antimicrob. Agents Chemother.
, vol.49
, pp. 2260-2266
-
-
Weigelt, J.1
Itani, K.2
Stevens, D.3
Lau, W.4
Dryden, M.5
Knirsch, C.6
-
32
-
-
0345019797
-
New visions in the pharmacology of anticonvulsion
-
Wolfgang L. New visions in the pharmacology of anticonvulsion. Eur. J. Pharmcol. 1998, 342:1-13.
-
(1998)
Eur. J. Pharmcol.
, vol.342
, pp. 1-13
-
-
Wolfgang, L.1
-
33
-
-
33947705587
-
Recent developments in the virology and antiviral research of severe acute respiratory syndrome coronavirus
-
Yeung K.S., Meanwell N.A. Recent developments in the virology and antiviral research of severe acute respiratory syndrome coronavirus. Infect. Dis. 2007, 7:29-41.
-
(2007)
Infect. Dis.
, vol.7
, pp. 29-41
-
-
Yeung, K.S.1
Meanwell, N.A.2
-
34
-
-
77249133540
-
Synthesis and biological evaluation of novel pyrazolyl-2,4-thiazolidinediones as anti-inflammatory and neuroprotective agents
-
Youssef A.M., White M.S., Klegeris A. Synthesis and biological evaluation of novel pyrazolyl-2,4-thiazolidinediones as anti-inflammatory and neuroprotective agents. Biorg. Med. Chem. 2010, 20:2019-2028.
-
(2010)
Biorg. Med. Chem.
, vol.20
, pp. 2019-2028
-
-
Youssef, A.M.1
White, M.S.2
Klegeris, A.3
|