메뉴 건너뛰기




Volumn 10, Issue 6, 2013, Pages 2270-2282

Relaxation dynamics and crystallization study of sildenafil in the liquid and glassy states

Author keywords

amorphous drug; dielectric relaxation; isothermal crystallization; molecular mobility; non isothermal crystallization; physical stability; sildenafil; viagra

Indexed keywords

SILDENAFIL;

EID: 84878631153     PISSN: 15438384     EISSN: 15438392     Source Type: Journal    
DOI: 10.1021/mp300479r     Document Type: Article
Times cited : (61)

References (56)
  • 3
    • 79956151039 scopus 로고    scopus 로고
    • Comprehensive studies on physical and chemical stability in liquid and glassy states of telmisartan (TEL): Solubility advantages given by cryomilled and quenched material
    • Adrjanowicz, K.; Grzybowska, K.; Kaminski, K.; Hawelek, L.; Paluch, M.; Zakowiecki, D. Comprehensive studies on physical and chemical stability in liquid and glassy states of telmisartan (TEL): solubility advantages given by cryomilled and quenched material Philos. Mag. 2011, 91, 1926-1948
    • (2011) Philos. Mag. , vol.91 , pp. 1926-1948
    • Adrjanowicz, K.1    Grzybowska, K.2    Kaminski, K.3    Hawelek, L.4    Paluch, M.5    Zakowiecki, D.6
  • 8
    • 0346639265 scopus 로고    scopus 로고
    • Dielectric study of the molecular mobility and the isothermal crystallization kinetics of an amorphous pharmaceutical drug substance
    • Alie, J.; Menegotto, J.; Cardon, P.; Duplaa, H.; Caron, A.; Lacabanne, C.; Bauer, M. Dielectric study of the molecular mobility and the isothermal crystallization kinetics of an amorphous pharmaceutical drug substance J. Pharm. Sci. 2004, 93, 218-233
    • (2004) J. Pharm. Sci. , vol.93 , pp. 218-233
    • Alie, J.1    Menegotto, J.2    Cardon, P.3    Duplaa, H.4    Caron, A.5    Lacabanne, C.6    Bauer, M.7
  • 9
    • 0342869049 scopus 로고
    • Kinetics of Phase Change. i General Theory
    • Avrami, M. Kinetics of Phase Change. I General Theory J. Chem. Phys. 1939, 7, 1103
    • (1939) J. Chem. Phys. , vol.7 , pp. 1103
    • Avrami, M.1
  • 10
    • 0001336124 scopus 로고
    • Kinetics of Phase Change. II Transformation-Time Relations for Random Distribution of Nuclei
    • Avrami, M. Kinetics of Phase Change. II Transformation-Time Relations for Random Distribution of Nuclei J. Chem. Phys. 1940, 8, 212
    • (1940) J. Chem. Phys. , vol.8 , pp. 212
    • Avrami, M.1
  • 11
    • 27644598487 scopus 로고    scopus 로고
    • New Method to Analyze Data on Overall Crystallization Kinetics
    • Avramov, I.; Avramova, K.; Russel, C. New Method to Analyze Data on Overall Crystallization Kinetics J. Cryst. Growth 2005, 285, 394-399
    • (2005) J. Cryst. Growth , vol.285 , pp. 394-399
    • Avramov, I.1    Avramova, K.2    Russel, C.3
  • 12
    • 0015034365 scopus 로고
    • Kinetics of non-isothermal crystallization
    • Ozawa, T. Kinetics of non-isothermal crystallization Polymer 1971, 12, 150
    • (1971) Polymer , vol.12 , pp. 150
    • Ozawa, T.1
  • 13
    • 0000682032 scopus 로고
    • Variation of peak temperature with heating rate in differential thermal analysis
    • Kissinger, H. E. Variation of peak temperature with heating rate in differential thermal analysis J. Res. Natl. Bur. Stand. 1956, 57, 217-221
    • (1956) J. Res. Natl. Bur. Stand. , vol.57 , pp. 217-221
    • Kissinger, H.E.1
  • 14
    • 33646003938 scopus 로고
    • Calculation of the Avrami parameters for heterogeneous solid state reactions using a modified the Kissinger method
    • Augis, J. A.; Bennett, J. E. Calculation of the Avrami parameters for heterogeneous solid state reactions using a modified the Kissinger method J. Therm. Anal. 1978, 13, 283-292
    • (1978) J. Therm. Anal. , vol.13 , pp. 283-292
    • Augis, J.A.1    Bennett, J.E.2
  • 15
    • 68949132727 scopus 로고    scopus 로고
    • Local mobility in amorphous pharmaceuticals - Characterization and implications on stability
    • Bhattacharya, S.; Suryanarayanan, R. Local mobility in amorphous pharmaceuticals-characterization and implications on stability J. Pharm. Sci. 2009, 98, 2935-2953
    • (2009) J. Pharm. Sci. , vol.98 , pp. 2935-2953
    • Bhattacharya, S.1    Suryanarayanan, R.2
  • 16
    • 43249092894 scopus 로고    scopus 로고
    • Role of thermodynamic, molecular, and kinetic factors in crystallization from the amorphous state
    • Bhugra, C.; Pikal, M. J. Role of thermodynamic, molecular, and kinetic factors in crystallization from the amorphous state J. Pharm. Sci. 2008, 97, 1329-1349
    • (2008) J. Pharm. Sci. , vol.97 , pp. 1329-1349
    • Bhugra, C.1    Pikal, M.J.2
  • 17
    • 34249006283 scopus 로고    scopus 로고
    • Dielectric relaxation and crystallization of ultraviscous melt and glassy states of aspirin, ibuprofen, progesterone, and quinidine
    • Johari, G. P.; Kim, S.; Shanker, R. M. Dielectric relaxation and crystallization of ultraviscous melt and glassy states of aspirin, ibuprofen, progesterone, and quinidine J. Pharm. Sci. 2007, 96, 1159-1175
    • (2007) J. Pharm. Sci. , vol.96 , pp. 1159-1175
    • Johari, G.P.1    Kim, S.2    Shanker, R.M.3
  • 19
    • 26944469990 scopus 로고    scopus 로고
    • Physical stability and relaxation of amorphous indomethacin
    • Vyazovkin, S.; Dranca, I. Physical stability and relaxation of amorphous indomethacin J. Phys. Chem. B 2005, 109, 18637-18644
    • (2005) J. Phys. Chem. B , vol.109 , pp. 18637-18644
    • Vyazovkin, S.1    Dranca, I.2
  • 20
    • 33645755595 scopus 로고    scopus 로고
    • Frustration on the way to crystallization in glass
    • Shintani, H.; Tanaka, H. Frustration on the way to crystallization in glass Nat. Phys. 2006, 2, 200-206
    • (2006) Nat. Phys. , vol.2 , pp. 200-206
    • Shintani, H.1    Tanaka, H.2
  • 23
    • 80052213580 scopus 로고    scopus 로고
    • Dynamic heterogeneity in amorphous materials
    • Berthier, L. Dynamic heterogeneity in amorphous materials Physics 2011, 4, 42-1-42-7
    • (2011) Physics , vol.4 , pp. 421-427
    • Berthier, L.1
  • 24
    • 77957740119 scopus 로고    scopus 로고
    • Correlation of nonexponentiality with dynamic heterogeneity from four-point dynamic susceptibility χ4(t) and its approximation χt(t)
    • Roland, C. M.; Fragiadakis, D.; Coslovich, D.; Capaccioli, S.; Ngai, K. L. Correlation of nonexponentiality with dynamic heterogeneity from four-point dynamic susceptibility χ4(t) and its approximation χT(t) J. Chem. Phys. 2010, 133, 124507
    • (2010) J. Chem. Phys. , vol.133 , pp. 124507
    • Roland, C.M.1    Fragiadakis, D.2    Coslovich, D.3    Capaccioli, S.4    Ngai, K.L.5
  • 25
    • 81555196464 scopus 로고    scopus 로고
    • Comparing dynamic correlation lengths from an approximation to the four-point dynamic susceptibility and from the picosecond vibrational dynamics
    • Fragiadakis, D.; Casalini, R.; Roland, C. M. Comparing dynamic correlation lengths from an approximation to the four-point dynamic susceptibility and from the picosecond vibrational dynamics Phys. Rev. E 2011, 84, 042501
    • (2011) Phys. Rev. e , vol.84 , pp. 042501
    • Fragiadakis, D.1    Casalini, R.2    Roland, C.M.3
  • 26
    • 84863311332 scopus 로고    scopus 로고
    • Effects of lowering temperature and raising pressure on the spatially heterogeneous dynamics of glass-forming van der Waals liquids
    • Grzybowski, A.; Kolodziejczyk, K.; Koperwas, K.; Grzybowska, K.; Paluch, M. Effects of lowering temperature and raising pressure on the spatially heterogeneous dynamics of glass-forming van der Waals liquids Phys. Rev. B 2012, 85, 220201(R)
    • (2012) Phys. Rev. B , vol.85
    • Grzybowski, A.1    Kolodziejczyk, K.2    Koperwas, K.3    Grzybowska, K.4    Paluch, M.5
  • 27
    • 55149123526 scopus 로고    scopus 로고
    • Non-isothermal crystallization and melting of ethylene-vinyl acetate copolymers with different vinyl acetate contents
    • Shi, X. M.; Zhang, J.; Jin, J.; Chen, S. J. Non-isothermal crystallization and melting of ethylene-vinyl acetate copolymers with different vinyl acetate contents eXPRESS Polym. Lett. 2008, 2, 623-629
    • (2008) EXPRESS Polym. Lett. , vol.2 , pp. 623-629
    • Shi, X.M.1    Zhang, J.2    Jin, J.3    Chen, S.J.4
  • 28
    • 0032974343 scopus 로고    scopus 로고
    • Rheological studies of barley (1→3)(1→4)-β-glucan in concentrated solution: Mechanistic and kinetic investigation of the gel formation
    • Böhm, N.; Kulicke, W.-M. Rheological studies of barley (1→3)(1→4)-β-glucan in concentrated solution: mechanistic and kinetic investigation of the gel formation Carbohydr. Res. 1999, 315, 302-311
    • (1999) Carbohydr. Res. , vol.315 , pp. 302-311
    • Böhm, N.1    Kulicke, W.-M.2
  • 29
    • 33748733089 scopus 로고    scopus 로고
    • Molecular dynamics and crystallization behaviour of isopentyl cyanobiphenyl as studied by dielectric relaxation spectroscopy
    • Massalska-Arodz, M.; Williams, G.; Smith, I. K.; Conolly, C.; Aldridge, G. A.; Dabrowski, R. Molecular dynamics and crystallization behaviour of isopentyl cyanobiphenyl as studied by dielectric relaxation spectroscopy J. Chem. Soc., Faraday Trans. 1998, 94, 387-394
    • (1998) J. Chem. Soc., Faraday Trans. , vol.94 , pp. 387-394
    • Massalska-Arodz, M.1    Williams, G.2    Smith, I.K.3    Conolly, C.4    Aldridge, G.A.5    Dabrowski, R.6
  • 30
    • 0037213873 scopus 로고    scopus 로고
    • 80 chalcogenide glass
    • 80 chalcogenide glass Physica B 2003, 325, 372-379
    • (2003) Physica B , vol.325 , pp. 372-379
    • Abu-Sehly, A.A.1
  • 31
    • 9244255262 scopus 로고    scopus 로고
    • Nonisothermal cold-crystallization kinetics of poly(trimethylene terephthalate)
    • Supaphol, P.; Apiwanthanakorn, N. Nonisothermal cold-crystallization kinetics of poly(trimethylene terephthalate) J. Polym. Sci., B: Polym. Phys. 2004, 42 (22) 4151-4163
    • (2004) J. Polym. Sci., B: Polym. Phys. , vol.42 , Issue.22 , pp. 4151-4163
    • Supaphol, P.1    Apiwanthanakorn, N.2
  • 32
    • 79954491963 scopus 로고    scopus 로고
    • Nonisothermal and Isothermal Cold Crystallization Behaviors of Biodegradable Poly(p-dioxanone)
    • Zeng, J. B.; Srinivansan, M.; Li, S. L.; Narayan, R.; Wang, Y. Z. Nonisothermal and Isothermal Cold Crystallization Behaviors of Biodegradable Poly(p-dioxanone) Ind. Eng. Chem. Res. 2011, 50, 4471-4477
    • (2011) Ind. Eng. Chem. Res. , vol.50 , pp. 4471-4477
    • Zeng, J.B.1    Srinivansan, M.2    Li, S.L.3    Narayan, R.4    Wang, Y.Z.5
  • 35
    • 0000119222 scopus 로고
    • Das Temperaturabhangigkeitgesetz der Viskosität von Flüssigkeiten
    • Vogel, H. Das Temperaturabhangigkeitgesetz der Viskosität von Flüssigkeiten J. Phys. Z. 1921, 22, 645-646
    • (1921) J. Phys. Z. , vol.22 , pp. 645-646
    • Vogel, H.1
  • 36
    • 84977689852 scopus 로고
    • Analysis of Recent Measurements of the Viscosity of Glasses
    • Fulcher, G. S. Analysis of Recent Measurements of the Viscosity of Glasses J. Am. Ceram. Soc. 1925, 8, 339-355
    • (1925) J. Am. Ceram. Soc. , vol.8 , pp. 339-355
    • Fulcher, G.S.1
  • 37
    • 84982343610 scopus 로고
    • Die Abhängigkeit der Viscosität von der Temperatur bie unterkühlten Flüssigkeiten
    • Tammann, G.; Hesse, W. Die Abhängigkeit der Viscosität von der Temperatur bie unterkühlten Flüssigkeiten Z. Anorg. Allg. Chem. 1926, 156, 245-257
    • (1926) Z. Anorg. Allg. Chem. , vol.156 , pp. 245-257
    • Tammann, G.1    Hesse, W.2
  • 38
    • 0037045179 scopus 로고    scopus 로고
    • Direct determinetaion of kinetic fragility indicates of glassforming liquids by differentional scanning calorimetry: Kinetic versus thermodynamic fragilities
    • Wang, L.-M.; Velikov, V.; Angell, C. A. Direct determinetaion of kinetic fragility indicates of glassforming liquids by differentional scanning calorimetry: Kinetic versus thermodynamic fragilities J. Chem. Phys. 2002, 117, 10184-10355
    • (2002) J. Chem. Phys. , vol.117 , pp. 10184-10355
    • Wang, L.-M.1    Velikov, V.2    Angell, C.A.3
  • 39
    • 20244375319 scopus 로고    scopus 로고
    • Response to "comment on 'Direct determination of the fragility indexes of glassforming liquids by differential scanning calorimetry. Kinetic vs thermodynamic fragilities'"
    • Wang, L.-M.; Angell, C. A. Response to "Comment on 'Direct determination of the fragility indexes of glassforming liquids by differential scanning calorimetry. Kinetic vs thermodynamic fragilities'" J. Chem. Phys. 2003, 118, 10353-10355
    • (2003) J. Chem. Phys. , vol.118 , pp. 10353-10355
    • Wang, L.-M.1    Angell, C.A.2
  • 40
    • 15444373850 scopus 로고    scopus 로고
    • Relationship among glass-forming ability, fragility, and short-range bond ordering of liquids
    • Tanaka, H. Relationship among glass-forming ability, fragility, and short-range bond ordering of liquids J. Non-Cryst. Solids 2005, 351, 678-690
    • (2005) J. Non-Cryst. Solids , vol.351 , pp. 678-690
    • Tanaka, H.1
  • 41
    • 73649093048 scopus 로고    scopus 로고
    • Influence of Fragility on Polymer Cold Crystallization
    • Sanz, A.; Nogales, A.; Ezquerra, T. A. Influence of Fragility on Polymer Cold Crystallization Macromolecules 2010, 43, 29-32
    • (2010) Macromolecules , vol.43 , pp. 29-32
    • Sanz, A.1    Nogales, A.2    Ezquerra, T.A.3
  • 42
    • 34250310890 scopus 로고    scopus 로고
    • Effect of a reduced mobility layer on the interplay between molecular relaxations and diffusion limited crystallization rate in ultrathin polymer films
    • Napolitano, S.; Wübbenhorst, M. Effect of a reduced mobility layer on the interplay between molecular relaxations and diffusion limited crystallization rate in ultrathin polymer films J. Phys. Chem. B 2007, 111, 5775-5780
    • (2007) J. Phys. Chem. B , vol.111 , pp. 5775-5780
    • Napolitano, S.1    Wübbenhorst, M.2
  • 43
    • 77956361367 scopus 로고    scopus 로고
    • Prediction of Onset of Crystallization in Amorphous Pharmaceutical Systems: Phenobarbital, Nifedipine/PVP, and Phenobarbital/PVP
    • Caron, V.; Bhugra, C.; Pikal, M. J. Prediction Of Onset Of Crystallization In Amorphous Pharmaceutical Systems: Phenobarbital, Nifedipine/PVP, and Phenobarbital/PVP J. Pharm. Sci. 2010, 99, 3887-3900
    • (2010) J. Pharm. Sci. , vol.99 , pp. 3887-3900
    • Caron, V.1    Bhugra, C.2    Pikal, M.J.3
  • 44
    • 53549126335 scopus 로고    scopus 로고
    • Correlation between Molecular Mobility and Crystal Growth of Amorphous Phenobarbital and Phenobarbital with Polyvinylpyrrolidone and L-Proline
    • Korhonen, O.; Bhugra, C.; Pikal, M. J. Correlation between Molecular Mobility and Crystal Growth of Amorphous Phenobarbital and Phenobarbital with Polyvinylpyrrolidone and L-Proline J. Pharm. Sci. 2008, 97, 3830-3841
    • (2008) J. Pharm. Sci. , vol.97 , pp. 3830-3841
    • Korhonen, O.1    Bhugra, C.2    Pikal, M.J.3
  • 45
    • 38349180826 scopus 로고    scopus 로고
    • Prediction of Onset of Crystallization from Experimental Relaxation Times. II. Comparison between Predicted and Experimental Onset Times
    • Bhugra, C.; Shmeis, R.; Krill, S. L.; Pikal, M. J. Prediction of Onset of Crystallization from Experimental Relaxation Times. II. Comparison between Predicted and Experimental Onset Times J. Pharm. Sci. 2008, 97, 455-472
    • (2008) J. Pharm. Sci. , vol.97 , pp. 455-472
    • Bhugra, C.1    Shmeis, R.2    Krill, S.L.3    Pikal, M.J.4
  • 46
    • 72649095414 scopus 로고    scopus 로고
    • Crystal Nucleation in a Supercooled Liquid with Glassy Dynamics
    • Saika-Voivod, I.; Bowles, R. K.; Poole, P. H. Crystal Nucleation in a Supercooled Liquid with Glassy Dynamics Phys. Rev. Lett. 2009, 225701
    • (2009) Phys. Rev. Lett. , pp. 225701
    • Saika-Voivod, I.1    Bowles, R.K.2    Poole, P.H.3
  • 47
    • 36248932204 scopus 로고    scopus 로고
    • Correlation between Dynamic Heterogeneity and Medium-Range Order in Two-Dimensional Glass-Forming Liquids
    • Kawasaki, T.; Araki, T.; Tanaka, H. Correlation between Dynamic Heterogeneity and Medium-Range Order in Two-Dimensional Glass-Forming Liquids Phys. Rev. Lett. 2007, 99, 215701
    • (2007) Phys. Rev. Lett. , vol.99 , pp. 215701
    • Kawasaki, T.1    Araki, T.2    Tanaka, H.3
  • 48
    • 34548447644 scopus 로고    scopus 로고
    • Topological persistence and dynamical heterogeneities near jamming
    • Abate, A. R.; Durian, D. J. Topological persistence and dynamical heterogeneities near jamming Phys. Rev. E 2007, 76, 021306
    • (2007) Phys. Rev. e , vol.76 , pp. 021306
    • Abate, A.R.1    Durian, D.J.2
  • 49
    • 51849102130 scopus 로고    scopus 로고
    • Dynamically correlated regions and congurational entropy in supercooled liquids
    • S. Capaccioli, S.; Ruocco, G.; Zamponi, F. Dynamically correlated regions and congurational entropy in supercooled liquids J. Phys. Chem. B 2008, 112, 10652-10658
    • (2008) J. Phys. Chem. B , vol.112 , pp. 10652-10658
    • Capaccioli S, S.1    Ruocco, G.2    Zamponi, F.3
  • 51
    • 0347936294 scopus 로고
    • On the temperature dependence of cooperative relaxation properties in glass forming liquids
    • Adam, G.; Gibbs, J. H. On the temperature dependence of cooperative relaxation properties in glass forming liquids J. Chem. Phys. 1965, 43, 139-146
    • (1965) J. Chem. Phys. , vol.43 , pp. 139-146
    • Adam, G.1    Gibbs, J.H.2
  • 52
    • 0001182230 scopus 로고    scopus 로고
    • Characterization of the time scales of molecular motion in pharmaceutically important glasses
    • Shamblin, S. L.; Tang, X.; Chang, L.; Hancock, B. C.; Pikal, M. J. Characterization of the time scales of molecular motion in pharmaceutically important glasses J. Phys. Chem. B 1999, 103, 4113-4121
    • (1999) J. Phys. Chem. B , vol.103 , pp. 4113-4121
    • Shamblin, S.L.1    Tang, X.2    Chang, L.3    Hancock, B.C.4    Pikal, M.J.5
  • 53
    • 0030188824 scopus 로고    scopus 로고
    • Strong and fragile liquids - A brief critique
    • Hodge, I. M. Strong and fragile liquids-a brief critique J. Non-Cryst. Solids 1996, 202, 164-172
    • (1996) J. Non-Cryst. Solids , vol.202 , pp. 164-172
    • Hodge, I.M.1
  • 54
    • 0035861398 scopus 로고    scopus 로고
    • Molecular mobility of amorphous pharmaceuticals determined using differential scanning calorimetry
    • Hancock, B. C.; Shamblin, S. L. Molecular mobility of amorphous pharmaceuticals determined using differential scanning calorimetry Thermochim. Acta 2001, 380, 95-107
    • (2001) Thermochim. Acta , vol.380 , pp. 95-107
    • Hancock, B.C.1    Shamblin, S.L.2
  • 55
    • 0842301322 scopus 로고    scopus 로고
    • Classification of secondary relaxation in glass-formers based on dynamic properties
    • Ngai, K. L.; Paluch, M. Classification of secondary relaxation in glass-formers based on dynamic properties J. Chem. Phys. 2004, 120, 857-873
    • (2004) J. Chem. Phys. , vol.120 , pp. 857-873
    • Ngai, K.L.1    Paluch, M.2
  • 56
    • 0037467252 scopus 로고    scopus 로고
    • An extended coupling model description of the evolution of dynamics with time in supercooled liquids and ionic conductors
    • Ngai, K. L. An extended coupling model description of the evolution of dynamics with time in supercooled liquids and ionic conductors J. Phys.: Condens. Matter 2003, 15, S1107
    • (2003) J. Phys.: Condens. Matter , vol.15 , pp. 1107
    • Ngai, K.L.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.