메뉴 건너뛰기




Volumn 100, Issue 7, 2011, Pages 2642-2657

Molecular dynamics of the cryomilled base and hydrochloride ziprasidones by means of dielectric spectroscopy

Author keywords

Crystallization; Dielectric spectroscopy; Dissolution rate; Milling; Molecular Dynamics; Ziprasidone

Indexed keywords

CHLORIDE; TRAMADOL; ZIPRASIDONE;

EID: 79955613205     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.22479     Document Type: Article
Times cited : (27)

References (57)
  • 2
    • 0343515548 scopus 로고
    • Bioavailability and in vitro liberation of glibenclamide from a new dosage form
    • Rupp W, Badian M, Heptner W, Malerczyk V. 1984. Bioavailability and in vitro liberation of glibenclamide from a new dosage form. Biopharm Pharmacokinet Eur Congr 2(1):413-420.
    • (1984) Biopharm Pharmacokinet Eur Congr , vol.2 , Issue.1 , pp. 413-420
    • Rupp, W.1    Badian, M.2    Heptner, W.3    Malerczyk, V.4
  • 3
    • 0031859673 scopus 로고    scopus 로고
    • Micronisation: A method of improving the bioavailability of poorly solubledrugs
    • Chaumeil JC. 1998. Micronisation: A method of improving the bioavailability of poorly solubledrugs. Methods Find Exp Clin Pharmacol 20:211-215.
    • (1998) Methods Find Exp Clin Pharmacol , vol.20 , pp. 211-215
    • Chaumeil, J.C.1
  • 4
    • 0031469675 scopus 로고    scopus 로고
    • Bioavailability of hydrochlorothiazide from pellets, made by extrusion spheronisation, containing polyethylene glycol 400 as a dissolution enhancer
    • Vervaet C, Remon JP. 1997. Bioavailability of hydrochlorothiazide from pellets, made by extrusion spheronisation, containing polyethylene glycol 400 as a dissolution enhancer. Pharm Res 14:1644-1646.
    • (1997) Pharm Res , vol.14 , pp. 1644-1646
    • Vervaet, C.1    Remon, J.P.2
  • 5
    • 0037027875 scopus 로고    scopus 로고
    • Preparation and dissolution characteristics of griseofulvin solid dispersions with saccharides
    • Saito M, Ugajin T, Nozawa Y, Sadzuka Y, Miyagishima A, Sonobe T. 2002. Preparation and dissolution characteristics of griseofulvin solid dispersions with saccharides. Int J Pharm 249:71-79.
    • (2002) Int J Pharm , vol.249 , pp. 71-79
    • Saito, M.1    Ugajin, T.2    Nozawa, Y.3    Sadzuka, Y.4    Miyagishima, A.5    Sonobe, T.6
  • 6
    • 0036096613 scopus 로고    scopus 로고
    • Formulation approaches for orally administered poorly soluble drugs
    • Pinnamaneni S, Das NG, Das SK. 2002. Formulation approaches for orally administered poorly soluble drugs. Pharmazie 57:291-300.
    • (2002) Pharmazie , vol.57 , pp. 291-300
    • Pinnamaneni, S.1    Das, N.G.2    Das, S.K.3
  • 8
    • 0019809124 scopus 로고
    • Differences in physico-pharmaceutical properties between crystalline and noncrystalline 9,3'-diacetylmidecamycin
    • Sato T, Okada A, Sdekiguchi K, Tsuda Y. 1981. Differences in physico-pharmaceutical properties between crystalline and noncrystalline 9, 3'-diacetylmidecamycin. Chem Pharm Bull 29:2675-2682.
    • (1981) Chem Pharm Bull , vol.29 , pp. 2675-2682
    • Sato, T.1    Okada, A.2    Sdekiguchi, K.3    Tsuda, Y.4
  • 9
    • 0023028276 scopus 로고
    • Some physicochemical properties of glassy indomethacin
    • Fukuoka E, Makita M, Yamamura S. 1986. Some physicochemical properties of glassy indomethacin. Chem Pharm Bull 34:4314-4321.
    • (1986) Chem Pharm Bull , vol.34 , pp. 4314-4321
    • Fukuoka, E.1    Makita, M.2    Yamamura, S.3
  • 10
    • 0002611989 scopus 로고
    • Molekulargalenik als grundlage moderner arzneiformung
    • Huttenrauch R. 1978. Molekulargalenik als grundlage moderner arzneiformung. Acta Pharm Technol Suppl 6:55.
    • (1978) Acta Pharm Technol Suppl , vol.6 , pp. 55
    • Huttenrauch, R.1
  • 11
    • 0017178826 scopus 로고
    • Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose
    • Yamamoto K, Nakano M, Arita T, Takayama Y, Nakai Y. 1976. Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose. J Pharm Sci 65:1484-1488.
    • (1976) J Pharm Sci , vol.65 , pp. 1484-1488
    • Yamamoto, K.1    Nakano, M.2    Arita, T.3    Takayama, Y.4    Nakai, Y.5
  • 13
    • 1142303337 scopus 로고    scopus 로고
    • What is the true solubility advantage for amorphous pharmaceuticals
    • Hancock BC, Parks M. 2000. What is the true solubility advantage for amorphous pharmaceuticals. Pharm Res 17:393-414.
    • (2000) Pharm Res , vol.17 , pp. 393-414
    • Hancock, B.C.1    Parks, M.2
  • 14
    • 0017857869 scopus 로고
    • Quantitative crystallinity determinations for β-lactam antibiotics by solution calorimetry: Correlations with stability
    • Pikal MJ, Lukes AL, Lang JE, Gaines K. 1978. Quantitative crystallinity determinations for β-lactam antibiotics by solution calorimetry: Correlations with stability. J Pharm Sci 67:767-773.
    • (1978) J Pharm Sci , vol.67 , pp. 767-773
    • Pikal, M.J.1    Lukes, A.L.2    Lang, J.E.3    Gaines, K.4
  • 16
    • 0035991640 scopus 로고    scopus 로고
    • Physical stability of amorphous pharmaceuticals: Importance of configurational thermodynamic quantities and molecular mobility
    • Zhou D, Zhang GGZ, Law D, Grant DJW, Schmitt EA. 2002. Physical stability of amorphous pharmaceuticals: Importance of configurational thermodynamic quantities and molecular mobility. J Pharm Sci 91:1863-1872.
    • (2002) J Pharm Sci , vol.91 , pp. 1863-1872
    • Zhou, D.1    Zhang, G.G.Z.2    Law, D.3    Grant, D.J.W.4    Schmitt, E.A.5
  • 17
    • 43249092894 scopus 로고    scopus 로고
    • Role of thermodynamic, molecular, and kinetic factors in crystallization from the amorphous state
    • Bhugra C, Pikal MJ. 2007. Role of thermodynamic, molecular, and kinetic factors in crystallization from the amorphous state. J Pharm Sci 97:1329-1349.
    • (2007) J Pharm Sci , vol.97 , pp. 1329-1349
    • Bhugra, C.1    Pikal, M.J.2
  • 18
    • 0000974873 scopus 로고    scopus 로고
    • Beta molecular rearrangement process, but not an alpha process, as governing the homogeneous crystal nucleation rate in supercooled liquid
    • Hikima T, Hanaya M, Oguni M. 1996. Beta molecular rearrangement process, but not an alpha process, as governing the homogeneous crystal nucleation rate in supercooled liquid. Bull Chem Soc Jpn 69:1863-1868.
    • (1996) Bull Chem Soc Jpn , vol.69 , pp. 1863-1868
    • Hikima, T.1    Hanaya, M.2    Oguni, M.3
  • 19
    • 0033608977 scopus 로고    scopus 로고
    • Microscopic observation of a peculiar crystallization in the glass transition region and [beta]-process as potentially controlling the growth rate in triphenylethylene
    • Hikima T, Hanaya M, Oguni M. 1999. Microscopic observation of a peculiar crystallization in the glass transition region and [beta]-process as potentially controlling the growth rate in triphenylethylene. J Mol Struct 479:245-250.
    • (1999) J Mol Struct , vol.479 , pp. 245-250
    • Hikima, T.1    Hanaya, M.2    Oguni, M.3
  • 20
    • 0030196932 scopus 로고    scopus 로고
    • Discovery of crystal nucleation proceeding much below the glass transition temperature in a supercooled liquid
    • Okamoto N, Oguni M. 1996. Discovery of crystal nucleation proceeding much below the glass transition temperature in a supercooled liquid. Solid State Commun 99:53-56.
    • (1996) Solid State Commun , vol.99 , pp. 53-56
    • Okamoto, N.1    Oguni, M.2
  • 21
    • 3242714321 scopus 로고    scopus 로고
    • Effect of preparation method on physical properties of amorphous trehalose
    • Surana R, Pyne A, Suryanarayanan R. 2004. Effect of preparation method on physical properties of amorphous trehalose. Pharm Res 21:1167-1176.
    • (2004) Pharm Res , vol.21 , pp. 1167-1176
    • Surana, R.1    Pyne, A.2    Suryanarayanan, R.3
  • 22
    • 45549083586 scopus 로고    scopus 로고
    • Hiking down the energy landscape: Progress toward the Kauzmann temperature via vapor deposition
    • Kearns KL, Swallen SF, Ediger MD, Wu T, Sun Y, Yu L. 2008. Hiking down the energy landscape: Progress toward the Kauzmann temperature via vapor deposition. J Phys Chem B 112:4934-4942.
    • (2008) J Phys Chem B , vol.112 , pp. 4934-4942
    • Kearns, K.L.1    Swallen, S.F.2    Ediger, M.D.3    Wu, T.4    Sun, Y.5    Yu, L.6
  • 23
    • 38449103877 scopus 로고    scopus 로고
    • Influence of substrate temperature on the stability of glasses prepared by vapor deposition
    • Kearns KL, Swallen SF, Ediger MD, Wu T, Yu L. 2007. Influence of substrate temperature on the stability of glasses prepared by vapor deposition. J Chem Phys 127:154702-154710.
    • (2007) J Chem Phys , vol.127 , pp. 154702-154710
    • Kearns, K.L.1    Swallen, S.F.2    Ediger, M.D.3    Wu, T.4    Yu, L.5
  • 24
    • 0036171845 scopus 로고    scopus 로고
    • Cryogenic grinding of indomethacin polymorphs and solvates: Assesement of amorhous phase formation and amorphous physical stability
    • Crowley KJ, Zografi G. 2002. Cryogenic grinding of indomethacin polymorphs and solvates: Assesement of amorhous phase formation and amorphous physical stability. J Pharm Sci 91:492-507.
    • (2002) J Pharm Sci , vol.91 , pp. 492-507
    • Crowley, K.J.1    Zografi, G.2
  • 25
    • 0022517252 scopus 로고
    • Effect of seed crystals on solid-state transformation of polymorphs of chloramphenicol palmitate during grinding
    • Otsuka M, Kaneniwa N. 1986. Effect of seed crystals on solid-state transformation of polymorphs of chloramphenicol palmitate during grinding. J Pharm Sci 75:506-511.
    • (1986) J Pharm Sci , vol.75 , pp. 506-511
    • Otsuka, M.1    Kaneniwa, N.2
  • 26
    • 0030606872 scopus 로고    scopus 로고
    • Polymorphic transitions of cimetidine during manufacture of solid dosage forms
    • Bauer-Brandl A. 1996. Polymorphic transitions of cimetidine during manufacture of solid dosage forms. Int J Pharm Sci 140:195-206.
    • (1996) Int J Pharm Sci , vol.140 , pp. 195-206
    • Bauer-Brandl, A.1
  • 27
    • 0022601812 scopus 로고
    • Effect of environmental temperature on polymorphic solid-state transformation of indomethacin during grinding
    • Otsuka M, Matsumoto T, Kaneniwa N. 1986. Effect of environmental temperature on polymorphic solid-state transformation of indomethacin during grinding. Chem Pharm Bull (Tokyo) 34:1784-1793.
    • (1986) Chem Pharm Bull (Tokyo) , vol.34 , pp. 1784-1793
    • Otsuka, M.1    Matsumoto, T.2    Kaneniwa, N.3
  • 28
    • 22744433672 scopus 로고    scopus 로고
    • Polymorphic transformation of the G-form of D-sorbitol upon milling: Structural and nanostructural analyses
    • Willart JF, Lefebvre J, Danede F, Comini S, Looten P, Descamps M. 2005. Polymorphic transformation of the G-form of D-sorbitol upon milling: Structural and nanostructural analyses. Solid State Commun 135:519-524.
    • (2005) Solid State Commun , vol.135 , pp. 519-524
    • Willart, J.F.1    Lefebvre, J.2    Danede, F.3    Comini, S.4    Looten, P.5    Descamps, M.6
  • 29
    • 33749457920 scopus 로고    scopus 로고
    • Analysis of amorphous and nanocrystalline solids from their X-ray diffraction patterns
    • Bates S, Zografi G, Engers D, Morris K, Crowley K, Newman A. 2006. Analysis of amorphous and nanocrystalline solids from their X-ray diffraction patterns. Pharm Res 23:2333-2349.
    • (2006) Pharm Res , vol.23 , pp. 2333-2349
    • Bates, S.1    Zografi, G.2    Engers, D.3    Morris, K.4    Crowley, K.5    Newman, A.6
  • 30
    • 64649086799 scopus 로고    scopus 로고
    • Solid state amorphization of pharmaceuticals
    • Willart JF, Descamps M. 2008. Solid state amorphization of pharmaceuticals. Mol Pharm 5:905-920.
    • (2008) Mol Pharm , vol.5 , pp. 905-920
    • Willart, J.F.1    Descamps, M.2
  • 34
    • 70349272428 scopus 로고    scopus 로고
    • Study of molecular dynamics of pharmaceutically important protic ionic liquid verapamil hydrochloride. I. Test of thermodynamic scaling
    • Wojnarowska Z, Paluch M, Grzybowski A, Adrjanowicz K, Grzybowska K, Kaminski K, Wlodarczyk P, Pionteck J. 2009. Study of molecular dynamics of pharmaceutically important protic ionic liquid verapamil hydrochloride. I. Test of thermodynamic scaling. J Chem Phys 131:104505-104518.
    • (2009) J Chem Phys , vol.131 , pp. 104505-104518
    • Wojnarowska, Z.1    Paluch, M.2    Grzybowski, A.3    Adrjanowicz, K.4    Grzybowska, K.5    Kaminski, K.6    Wlodarczyk, P.7    Pionteck, J.8
  • 35
    • 0034019632 scopus 로고    scopus 로고
    • Interpretation of relaxation time constants for amorphous pharmaceutical systems
    • Shamblin SL, Hancock BC, Dupuis Y, Pikal MJ. 1999. Interpretation of relaxation time constants for amorphous pharmaceutical systems. J Pharm Sci 89:417-427.
    • (1999) J Pharm Sci , vol.89 , pp. 417-427
    • Shamblin, S.L.1    Hancock, B.C.2    Dupuis, Y.3    Pikal, M.J.4
  • 36
    • 27944497469 scopus 로고    scopus 로고
    • Dielectric studies of molecular motions in amorphous solid and ultraviscous acetaminophen
    • Johari GP, Kim S, Shanker RM. 2005. Dielectric studies of molecular motions in amorphous solid and ultraviscous acetaminophen. J Pharm Sci 94:2207-2223.
    • (2005) J Pharm Sci , vol.94 , pp. 2207-2223
    • Johari, G.P.1    Kim, S.2    Shanker, R.M.3
  • 37
    • 0036722688 scopus 로고    scopus 로고
    • Discovery of homogeneous-nucleation-based crystallization in simple glass-forming liquid of toluene below its glass-transition temperature
    • Hatase M, Hanaya M, Hikima T, Oguni M. 2003. Discovery of homogeneous-nucleation-based crystallization in simple glass-forming liquid of toluene below its glass-transition temperature. J Non-Cryst Solids 307-310:257-263.
    • (2003) J Non-Cryst Solids , vol.307-310 , pp. 257-263
    • Hatase, M.1    Hanaya, M.2    Hikima, T.3    Oguni, M.4
  • 38
    • 2442671463 scopus 로고    scopus 로고
    • Relation between some secondary relaxations and the α relaxations in glass-forming materials according to the coupling model
    • Ngai KL. 1998. Relation between some secondary relaxations and the α relaxations in glass-forming materials according to the coupling model. J Chem Phys 109:6982-6994.
    • (1998) J Chem Phys , vol.109 , pp. 6982-6994
    • Ngai, K.L.1
  • 39
    • 0037467252 scopus 로고    scopus 로고
    • An extended coupling model description of the evolution of dynamics with time in supercooled liquids and ionic conductors
    • Ngai KL. 2003. An extended coupling model description of the evolution of dynamics with time in supercooled liquids and ionic conductors. J Phys Condens Mat 15:S1107-S1125.
    • (2003) J Phys Condens Mat , vol.15
    • Ngai, K.L.1
  • 40
    • 0842301322 scopus 로고    scopus 로고
    • Classification of secondary relaxation in glass-formers based on dynamic properties
    • Ngai KL, Paluch M. 2004. Classification of secondary relaxation in glass-formers based on dynamic properties. J Chem Phys 120:857-873.
    • (2004) J Chem Phys , vol.120 , pp. 857-873
    • Ngai, K.L.1    Paluch, M.2
  • 43
    • 31144447946 scopus 로고    scopus 로고
    • Dynamics of the amorphous and crystalline α-, γ-phases of indomethacin
    • Carpentier L, Decressain R, Desprez S, Descamps M. 2006. Dynamics of the amorphous and crystalline α-, γ-phases of indomethacin. J Phys Chem B 110:457-464.
    • (2006) J Phys Chem B , vol.110 , pp. 457-464
    • Carpentier, L.1    Decressain, R.2    Desprez, S.3    Descamps, M.4
  • 46
    • 56449092347 scopus 로고    scopus 로고
    • Dielectric relaxation study of the dynamics of monosaccharides: D-Ribose and 2-deoxy-D-ribose
    • Kaminski K, Kaminska E, Wlodarczyk P, Paluch M, Ziolo J, Ngai KL. 2008. Dielectric relaxation study of the dynamics of monosaccharides: D-Ribose and 2-deoxy-D-ribose. J Phys Condens Matter 20:335104-335112.
    • (2008) J Phys Condens Matter , vol.20 , pp. 335104-335112
    • Kaminski, K.1    Kaminska, E.2    Wlodarczyk, P.3    Paluch, M.4    Ziolo, J.5    Ngai, K.L.6
  • 47
    • 0142072152 scopus 로고    scopus 로고
    • Two-order-parameter description of liquids. I. A general model of glass transition covering its strong to fragile limit
    • Tanaka HJ. 1999. Two-order-parameter description of liquids. I. A general model of glass transition covering its strong to fragile limit. J Chem Phys 111:3163-3175.
    • (1999) J Chem Phys , vol.111 , pp. 3163-3175
    • Tanaka, H.J.1
  • 48
    • 27444434179 scopus 로고    scopus 로고
    • Two-order-parameter model of the liquid-glass transition. I. Relation between glass transition and crystallization
    • Tanaka H. Two-order-parameter model of the liquid-glass transition. I. Relation between glass transition and crystallization. J Non-Cryst. Solids 351:3371-3384.
    • J Non-Cryst. Solids , vol.351 , pp. 3371-3384
    • Tanaka, H.1
  • 49
    • 33645755595 scopus 로고    scopus 로고
    • Frustration on the way to crystallization in glass
    • Shintani H, Tanaka H. 2006. Frustration on the way to crystallization in glass. Nature Phys. 2:200-206.
    • (2006) Nature Phys. , vol.2 , pp. 200-206
    • Shintani, H.1    Tanaka, H.2
  • 50
    • 0001785405 scopus 로고
    • A complex plane analysis of a-dispersion in some polymer systems
    • Havriliak S, Negami S. 1966. A complex plane analysis of a-dispersion in some polymer systems. J Polym Sci C 14:99.
    • (1966) J Polym Sci C , vol.14 , pp. 99
    • Havriliak, S.1    Negami, S.2
  • 51
    • 0036829807 scopus 로고    scopus 로고
    • Dielectric spectroscopy of glass-forming materials: A relaxation and excess wing
    • Lunkenheimer P, Loidl A. 2002. Dielectric spectroscopy of glass-forming materials: A relaxation and excess wing. Chem Phys 284:205-219.
    • (2002) Chem Phys , vol.284 , pp. 205-219
    • Lunkenheimer, P.1    Loidl, A.2
  • 52
    • 4243295846 scopus 로고    scopus 로고
    • From strong to fragile glass formers: Secondary relaxation in polyalcohols
    • Döß A, Paluch M, Sillescu H, Hinze G. 2002. From strong to fragile glass formers: Secondary relaxation in polyalcohols. Phys Rev Lett 88:095701-095705.
    • (2002) Phys Rev Lett , vol.88 , pp. 095701-095705
    • Döß, A.1    Paluch, M.2    Sillescu, H.3    Hinze, G.4
  • 53
    • 0037428571 scopus 로고    scopus 로고
    • Self-diffusion of tris-naphthylbenzene near the glass transition
    • Swallen SF, Bonvallet PA, McMahon RJ, Ediger MD. 2003. Self-diffusion of tris-naphthylbenzene near the glass transition. Phys Rev Lett 90:015901-015905.
    • (2003) Phys Rev Lett , vol.90 , pp. 015901-015905
    • Swallen, S.F.1    Bonvallet, P.A.2    McMahon, R.J.3    Ediger, M.D.4
  • 54
    • 0000729009 scopus 로고    scopus 로고
    • Flow, diffusion and crystallization of supercooled liquids: Revisited
    • Ngai KL, Magill JH, Plazek DJ. 2000. Flow, diffusion and crystallization of supercooled liquids: Revisited. J Chem Phys 112:1887-1892.
    • (2000) J Chem Phys , vol.112 , pp. 1887-1892
    • Ngai, K.L.1    Magill, J.H.2    Plazek, D.J.3
  • 55
    • 33748565282 scopus 로고
    • Dispersion and absorption in dielecttrics.I Alternating current characteristics
    • Cole KS, Cole RH. 1941. Dispersion and absorption in dielecttrics.I Alternating current characteristics. J Chem Phys 9:341.
    • (1941) J Chem Phys , vol.9 , pp. 341
    • Cole, K.S.1    Cole, R.H.2
  • 56
    • 42749103225 scopus 로고    scopus 로고
    • Glass transition and relaxation processes in supercooled water
    • Cerveny S, Schwartz GA, Bergman R, Swenson J. 2004. Glass transition and relaxation processes in supercooled water. Phys Rev Lett 93:245702-245706.
    • (2004) Phys Rev Lett , vol.93 , pp. 245702-245706
    • Cerveny, S.1    Schwartz, G.A.2    Bergman, R.3    Swenson, J.4
  • 57


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.