메뉴 건너뛰기




Volumn 7, Issue 1, 2013, Pages 1-7

Topical non steroidal anti inflammatory drug (NSAIDs) microemulsions: Rationale, review and future prospective

Author keywords

Droplet size; Microemulsion; Solubility; Surfactant

Indexed keywords

COSURFACTANT; NONSTEROID ANTIINFLAMMATORY AGENT; SURFACTANT;

EID: 84877135543     PISSN: 09738398     EISSN: 1998409X     Source Type: Journal    
DOI: 10.4103/0973-8398.110929     Document Type: Review
Times cited : (14)

References (49)
  • 1
    • 84877132491 scopus 로고
    • Topical drug delivery formulations
    • New York
    • David AO, Anton HA. Topical Drug Delivery Formulations. New York: Marcel Dekker; 1990. p. 1.
    • (1990) Marcel Dekker , pp. 1
    • David, A.O.1    Anton, H.A.2
  • 2
    • 0000965958 scopus 로고
    • Transparent water in oil dispersions: The oleopathic hydromicelle
    • Hoar TP, Schulman JH. Transparent water in oil dispersions: The oleopathic hydromicelle. Nat 1943;152:102-3.
    • (1943) Nat , vol.152 , pp. 102-103
    • Hoar, T.P.1    Schulman, J.H.2
  • 4
    • 0033778512 scopus 로고    scopus 로고
    • Oral versus topical NSAIDs in rheumatic diseases: A comparison
    • Heyneman CA, Lawless-Liday C, Wall GC. Oral versus topical NSAIDs in rheumatic diseases: A comparison. Drugs 2000;60:555-74.
    • (2000) Drugs , vol.60 , pp. 555-574
    • Heyneman, C.A.1    Lawless-Liday, C.2    Wall, G.C.3
  • 5
    • 13444306287 scopus 로고    scopus 로고
    • AOT water-in-oil microemulsions as a penetration enhancer in transdermal drug delivery of 5-fluorouracil
    • Gupta RR, Jain SK, Varshney M. AOT water-in-oil microemulsions as a penetration enhancer in transdermal drug delivery of 5-fluorouracil. Colloids Surf B Biointerfaces 2005;41:25-32.
    • (2005) Colloids Surf B Biointerfaces , vol.41 , pp. 25-32
    • Gupta, R.R.1    Jain, S.K.2    Varshney, M.3
  • 7
    • 33644620735 scopus 로고    scopus 로고
    • Transdermal permeation of tetracaine hydrochloride by lecithin microemulsion: In vivo
    • Changez M, Chander J, Dinda AK. Transdermal permeation of tetracaine hydrochloride by lecithin microemulsion: In vivo. Colloids Surf B Biointerfaces 2006;48:58-66.
    • (2006) Colloids Surf B Biointerfaces , vol.48 , pp. 58-66
    • Changez, M.1    Chander, J.2    Dinda, A.K.3
  • 8
    • 4143126493 scopus 로고    scopus 로고
    • A study of microemulsion systems for transdermal delivery of triptolide
    • Chen H, Chang X, Weng T, Zhao X, Gao Z, Yang Y, et al., A study of microemulsion systems for transdermal delivery of triptolide. J Control Release 2004;98:427-36.
    • (2004) J Control Release , vol.98 , pp. 427-436
    • Chen, H.1    Chang, X.2    Weng, T.3    Zhao, X.4    Gao, Z.5    Yang, Y.6
  • 9
    • 33646354629 scopus 로고    scopus 로고
    • Microemulsion-based hydrogel formulation of ibuprofen for topical delivery
    • Chen H, Chang X, Du D, Li J, Xu H, Yang X. Microemulsion-based hydrogel formulation of ibuprofen for topical delivery. Int J Pharm 2006;315:52-8.
    • (2006) Int J Pharm , vol.315 , pp. 52-58
    • Chen, H.1    Chang, X.2    Du, D.3    Li, J.4    Xu, H.5    Yang, X.6
  • 11
    • 0031891234 scopus 로고    scopus 로고
    • Triglyceride-based microemulsion for intravenous administration of sparingly soluble substances
    • von Corswant C, Thorén P, Engström S. Triglyceride-based microemulsion for intravenous administration of sparingly soluble substances. J Pharm Sci 1998;87:200-8.
    • (1998) J Pharm Sci , vol.87 , pp. 200-208
    • Von Corswant, C.1    Thorén, P.2    Engström, S.3
  • 12
    • 0029050215 scopus 로고
    • Investigations into the formation and characterization of phospholipids microemulsions. Iv. pseudo-ternary phase diagrams of systems containing water-lecithin-alcohol and oil; The influence of oil
    • Aboofazeli R, Patel N, Thomas M, Lawrence MJ. Investigations into the formation and characterization of phospholipids microemulsions. iv. pseudo-ternary phase diagrams of systems containing water-lecithin-alcohol and oil; the influence of oil. Int J Pharm 1995;125:107-16.
    • (1995) Int J Pharm , vol.125 , pp. 107-116
    • Aboofazeli, R.1    Patel, N.2    Thomas, M.3    Lawrence, M.J.4
  • 13
    • 0030476053 scopus 로고    scopus 로고
    • Current status and future prospects of transdermal drug delivery
    • Guy RH. Current status and future prospects of transdermal drug delivery. Pharm Res 1996;13:1765-9.
    • (1996) Pharm Res , vol.13 , pp. 1765-1769
    • Guy, R.H.1
  • 14
    • 33846156172 scopus 로고    scopus 로고
    • Four myths about transdermal drug delivery
    • Gordon RD, Peterson TA. Four myths about transdermal drug delivery. Drug Deliv Technol 2003;3:1-7.
    • (2003) Drug Deliv Technol , vol.3 , pp. 1-7
    • Gordon, R.D.1    Peterson, T.A.2
  • 15
    • 4644371740 scopus 로고    scopus 로고
    • Trends in the use of ultrasound-mediated transdermal drug delivery
    • Boucaud A. Trends in the use of ultrasound-mediated transdermal drug delivery. Drug Discov Today 2004;9:827-8.
    • (2004) Drug Discov Today , vol.9 , pp. 827-828
    • Boucaud, A.1
  • 16
    • 1242308254 scopus 로고    scopus 로고
    • Current status and future potential of transdermal drug delivery
    • Prausnitz MR, Mitragotri S, Langer R. Current status and future potential of transdermal drug delivery. Nat Rev Drug Discov 2004;3:115-24.
    • (2004) Nat Rev Drug Discov , vol.3 , pp. 115-124
    • Prausnitz, M.R.1    Mitragotri, S.2    Langer, R.3
  • 18
    • 0030955275 scopus 로고    scopus 로고
    • Characterization and stability of various liposome-encapsulated enoxacin formulations
    • Fang JY, Lin HH, Hsu LR, Tsai YH. Characterization and stability of various liposome-encapsulated enoxacin formulations. Chem Pharm Bull (Tokyo) 1997;45:1504-9.
    • (1997) Chem Pharm Bull (Tokyo) , vol.45 , pp. 1504-1509
    • Fang, J.Y.1    Lin, H.H.2    Hsu, L.R.3    Tsai, Y.H.4
  • 19
  • 20
    • 84877106432 scopus 로고
    • Coarse dispersions
    • In: 4th ed. New Delhi: B.I. Waverly Pvt, Ltd
    • Martin A. Coarse dispersions. In: Physical Pharmacy. 4th ed. New Delhi: B.I. Waverly Pvt, Ltd; 1994. p. 495-6.
    • (1994) Physical Pharmacy , pp. 495-496
    • Martin, A.1
  • 21
    • 0000443093 scopus 로고
    • Structure of water in microemulsions: Electrical, birefringence, and nuclear magnetic resonance studies
    • Shah DO, Hamlin RM Jr. Structure of water in microemulsions: Electrical, birefringence, and nuclear magnetic resonance studies. Science 1971;171:483-5.
    • (1971) Science , vol.171 , pp. 483-485
    • Shah, D.O.1    Hamlin Jr., R.M.2
  • 23
    • 0033430984 scopus 로고    scopus 로고
    • Microemulsions: An overview and pharmaceutical applications
    • Tenjarla S. Microemulsions: An overview and pharmaceutical applications. Crit Rev Ther Drug Carrier Syst 1999;16:461-521.
    • (1999) Crit Rev Ther Drug Carrier Syst , vol.16 , pp. 461-521
    • Tenjarla, S.1
  • 24
    • 0026757902 scopus 로고
    • Phase studies of oil-in water phospoholipid microemulsions
    • Attwood D, Mallon C, Taylor CJ. Phase studies of oil-in water phospoholipid microemulsions. Int J Pharm 1992;84:45-8.
    • (1992) Int J Pharm , vol.84 , pp. 45-48
    • Attwood, D.1    Mallon, C.2    Taylor, C.J.3
  • 25
    • 33646547331 scopus 로고    scopus 로고
    • Microemulsions: A potential drug delivery system
    • Ghosh PK, Murthy RS. Microemulsions: A potential drug delivery system. Curr Drug Deliv 2006;3:167-80.
    • (2006) Curr Drug Deliv , vol.3 , pp. 167-180
    • Ghosh, P.K.1    Murthy, R.S.2
  • 26
    • 0034614208 scopus 로고    scopus 로고
    • Microemulsion-based media as novel drug delivery systems
    • Lawrence MJ, Rees GD. Microemulsion-based media as novel drug delivery systems. Adv Drug Deliv Rev 2000;45:89-121.
    • (2000) Adv Drug Deliv Rev , vol.45 , pp. 89-121
    • Lawrence, M.J.1    Rees, G.D.2
  • 27
    • 49049123075 scopus 로고
    • Effect of alcohol cosurfactant length on microemulsion structure
    • Stilbs P, Lindman B, Rapacki k. Effect of alcohol cosurfactant length on microemulsion structure. J Colloid Interface Sci 1983;95:583-5.
    • (1983) J Colloid Interface Sci , vol.95 , pp. 583-585
    • Stilbs, P.1    Lindman, B.2    Rapacki, K.3
  • 28
    • 0030159231 scopus 로고    scopus 로고
    • Biological microemulsions V: Mutual mixing of oils, amphiphiles and water in ternary and quaternary combinations
    • Mitra N, Mukherjee L, Bhattacharya PK, Moulik SP. Biological microemulsions V: Mutual mixing of oils, amphiphiles and water in ternary and quaternary combinations. Indian J Biochem Biophys 1996;33:206-12.
    • (1996) Indian J Biochem Biophys , vol.33 , pp. 206-212
    • Mitra, N.1    Mukherjee, L.2    Bhattacharya, P.K.3    Moulik, S.P.4
  • 29
    • 79952021431 scopus 로고    scopus 로고
    • Design and evaluation of microemulsions based drug delivery system
    • Jadhav KR, Shetye SL, Kadam VJ. Design and evaluation of microemulsions based drug delivery system. Int J Adv Pharm Sci 2010;1:156-66.
    • (2010) Int J Adv Pharm Sci , vol.1 , pp. 156-166
    • Jadhav, K.R.1    Shetye, S.L.2    Kadam, V.J.3
  • 30
    • 0034602595 scopus 로고    scopus 로고
    • NMR characterisation and transdermal drug delivery potential of microemulsion systems
    • Kreilgaard M, Pedersen EJ, Jaroszewski JW. NMR characterisation and transdermal drug delivery potential of microemulsion systems. J Control Release 2000;69:421-33.
    • (2000) J Control Release , vol.69 , pp. 421-433
    • Kreilgaard, M.1    Pedersen, E.J.2    Jaroszewski, J.W.3
  • 31
    • 17344386412 scopus 로고
    • A comparison between non-ionic micelles and microemulsions as a means of incorporating the poorly water soluble drug diazepam
    • Malcolmson C, Lawrence MJ. A comparison between non-ionic micelles and microemulsions as a means of incorporating the poorly water soluble drug diazepam. J Pharm Pharmacol 1990;42:6.
    • (1990) J Pharm Pharmacol , vol.42 , pp. 6
    • Malcolmson, C.1    Lawrence, M.J.2
  • 32
    • 0031888408 scopus 로고    scopus 로고
    • Effect of oil on the level of solubilization of testosterone propionate into nonionic oil-in-water microemulsions
    • Malcolmson C, Satra C, Kantaria S, Sidhu A, Lawrence MJ. Effect of oil on the level of solubilization of testosterone propionate into nonionic oil-in-water microemulsions. J Pharm Sci 1998;87:109-16.
    • (1998) J Pharm Sci , vol.87 , pp. 109-116
    • Malcolmson, C.1    Satra, C.2    Kantaria, S.3    Sidhu, A.4    Lawrence, M.J.5
  • 33
    • 0027414119 scopus 로고
    • A comparison of the incorporation of model steroids into non-ionic micellar and microemulsion systems
    • Malcolmson C, Lawrence MJ. A comparison of the incorporation of model steroids into non-ionic micellar and microemulsion systems. J Pharm Pharmacol 1993;45:141-3.
    • (1993) J Pharm Pharmacol , vol.45 , pp. 141-143
    • Malcolmson, C.1    Lawrence, M.J.2
  • 34
    • 0343909521 scopus 로고
    • Conditions to produce so-called microemulsions: Factors to increase the mutual solubility of oil and water by solubilizer
    • Shinoda K, Kunieda H. Conditions to produce so-called microemulsions: Factors to increase the mutual solubility of oil and water by solubilizer. J Colloid Interface Sci 1973;42:381.
    • (1973) J Colloid Interface Sci , vol.42 , pp. 381
    • Shinoda, K.1    Kunieda, H.2
  • 37
    • 84877129942 scopus 로고
    • Microemulsions and method for preparing microemulsion
    • Rosano HL. Microemulsions and method for preparing microemulsion. J Colloid Interface Sci 1973;44:242.
    • (1973) J Colloid Interface Sci , vol.44 , pp. 242
    • Rosano, H.L.1
  • 38
    • 84864742069 scopus 로고    scopus 로고
    • Formulation, development and evaluation of topical microemulsion gels for nimsulide
    • Pawar AY. Formulation, development and evaluation of topical microemulsion gels for nimsulide. J Pharm Res 2011;4:1004-6.
    • (2011) J Pharm Res , vol.4 , pp. 1004-1006
    • Pawar, A.Y.1
  • 40
    • 77953175267 scopus 로고    scopus 로고
    • Fabrication and evaluation of hydrogel thickened microemulsion of ibuprofen for topical delivery
    • Gohel MC, Nagori SA. Fabrication and evaluation of hydrogel thickened microemulsion of ibuprofen for topical delivery. Indian J Pharm Educ Res 2010;44:189-96.
    • (2010) Indian J Pharm Educ Res , vol.44 , pp. 189-196
    • Gohel, M.C.1    Nagori, S.A.2
  • 41
  • 42
    • 77953411664 scopus 로고    scopus 로고
    • The novel formulation design of o/w microemulsion of ketoprofen for improving transdermal absorption
    • Dhamankar AK, Manwar JV, Kumbhar DD. The novel formulation design of o/w microemulsion of ketoprofen for improving transdermal absorption. Int J Pharm Tech Res 2009;1:1449-57.
    • (2009) Int J Pharm Tech Res , vol.1 , pp. 1449-1457
    • Dhamankar, A.K.1    Manwar, J.V.2    Kumbhar, D.D.3
  • 43
    • 84862748198 scopus 로고    scopus 로고
    • Topical delivery of diclofenac using microemulsion systems
    • Dima S, Popescu M. Topical delivery of diclofenac using microemulsion systems. Rom Biotechnol Lett 2008;13:49-55.
    • (2008) Rom Biotechnol Lett , vol.13 , pp. 49-55
    • Dima, S.1    Popescu, M.2
  • 44
    • 70849104994 scopus 로고    scopus 로고
    • Microemulsion as vehicle for transdermal permeation of drugs
    • Zabka M, Skoviera F. Microemulsion as vehicle for transdermal permeation of drugs. Acta Facult Pharm Univ Comenianae 2003;50:147-55.
    • (2003) Acta Facult Pharm Univ Comenianae , vol.50 , pp. 147-155
    • Zabka, M.1    Skoviera, F.2
  • 45
    • 0041418440 scopus 로고    scopus 로고
    • Fluorescence quenching of Acridine Orange in microemulsions induced by the non-steroidal anti-inflammatory drug Piroxicam
    • Andrade SM, Costa SM. Fluorescence quenching of Acridine Orange in microemulsions induced by the non-steroidal anti-inflammatory drug Piroxicam. Photochem Photobiol Sci 2003;2:605-10.
    • (2003) Photochem Photobiol Sci , vol.2 , pp. 605-610
    • Andrade, S.M.1    Costa, S.M.2
  • 46
    • 0037026275 scopus 로고    scopus 로고
    • Lecithin microemulsions for the topical administration of ketoprofen: Percutaneous adsorption through human skin and in vivo human skin tolerability
    • Paolino D, Ventura CA, Nisticò S, Puglisi G, Fresta M. Lecithin microemulsions for the topical administration of ketoprofen: Percutaneous adsorption through human skin and in vivo human skin tolerability. Int J Pharm 2002;244:21-31.
    • (2002) Int J Pharm , vol.244 , pp. 21-31
    • Paolino, D.1    Ventura, C.A.2    Nisticò, S.3    Puglisi, G.4    Fresta, M.5
  • 47
    • 0035834177 scopus 로고    scopus 로고
    • Transdermal delivery of ketoprofen using microemulsions
    • Rhee YS, Choi JG, Park ES, Chi SC. Transdermal delivery of ketoprofen using microemulsions. Int J Pharm 2001;228:161-70.
    • (2001) Int J Pharm , vol.228 , pp. 161-170
    • Rhee, Y.S.1    Choi, J.G.2    Park, E.S.3    Chi, S.C.4
  • 48
    • 0035800244 scopus 로고    scopus 로고
    • Inclusion complex of piroxicam with beta-cyclodextrin and incorporation in cationic microemulsion. In vitro drug release and in vivo topical anti-inflammatory effect
    • Dalmora ME, Dalmora SL, Oliveira AG. Inclusion complex of piroxicam with beta-cyclodextrin and incorporation in cationic microemulsion. In vitro drug release and in vivo topical anti-inflammatory effect. Int J Pharm 2001;222:45-55.
    • (2001) Int J Pharm , vol.222 , pp. 45-55
    • Dalmora, M.E.1    Dalmora, S.L.2    Oliveira, A.G.3
  • 49
    • 0032806764 scopus 로고    scopus 로고
    • Influence of phase transformation on indomethacin release from microemulsions
    • 49
    • Trotta M. Influence of phase transformation on indomethacin release from microemulsions. J Control Release 1999;60:399-405.49.
    • (1999) J Control Release , vol.60 , pp. 399-399
    • Trotta, M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.