Next-generation integrase inhibitors: Where to after raltegravir?

Drugs

Volumn 73, Issue 3, 2013, Pages 213-228

  Karmon, Sharon L ^a,b   Markowitz, Martin ^a,b  

^a AARON DIAMOND AIDS RESEARCH CENTER   (United States)

^b ROCKEFELLER UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ABACAVIR; ATAZANAVIR; ATAZANAVIR PLUS RITONAVIR; BI 224436; COBICISTAT; COBICISTAT PLUS ELVITEGRAVIR PLUS EMTRICITABINE PLUS TENOFOVIR DISOPROXIL; DIDANOSINE; DOLUTEGRAVIR; EFAVIRENZ; EFAVIRENZ PLUS EMTRICITABINE PLUS TENOFOVIR DISOPROXIL; ELVITEGRAVIR; EMTRICITABINE; EMTRICITABINE PLUS TENOFOVIR DISOPROXIL; ENFUVIRTIDE; ETRAVIRINE; INTEGRASE; INTEGRASE INHIBITOR; LAMIVUDINE; LOPINAVIR; LOPINAVIR PLUS RITONAVIR; PLACEBO; PROTEINASE INHIBITOR; RALTEGRAVIR; RITONAVIR; RNA DIRECTED DNA POLYMERASE INHIBITOR; S GSK 1265744; STAVUDINE; TENOFOVIR; TIPRANAVIR; UNCLASSIFIED DRUG; UNINDEXED DRUG; ZIDOVUDINE;

ACUTE STRESS DISORDER; ALANINE AMINOTRANSFERASE BLOOD LEVEL; ALLERGIC REACTION; ANTIVIRAL ACTIVITY; ANTIVIRAL RESISTANCE; ANTIVIRAL THERAPY; AREA UNDER THE CURVE; CONSTIPATION; CROSS RESISTANCE; DIARRHEA; DIZZINESS; DOSAGE SCHEDULE COMPARISON; DRUG BINDING SITE; DRUG DOSE COMPARISON; DRUG DOSE ESCALATION; DRUG ELIMINATION; DRUG HALF LIFE; DRUG MECHANISM; DRUG METABOLISM; DRUG PROTEIN BINDING; DRUG SUBSTITUTION; DRUG TOLERABILITY; DRUG WITHDRAWAL; FATIGUE; FEVER; GLOMERULUS FILTRATION RATE; HEADACHE; HUMAN; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS 1 INFECTION; IC 50; INJECTION SITE NODULE; INJECTION SITE PAIN; INJECTION SITE REACTION; INSOMNIA; LIVER FUNCTION TEST; MENTAL DISEASE; MONOTHERAPY; MULTICENTER STUDY (TOPIC); MYOPATHY; NAUSEA; NEUROLOGIC DISEASE; NONHUMAN; ORAL PARESTHESIA; PHASE 1 CLINICAL TRIAL (TOPIC); PHASE 2 CLINICAL TRIAL (TOPIC); PHASE 3 CLINICAL TRIAL (TOPIC); RANDOMIZED CONTROLLED TRIAL (TOPIC); RASH; REPEATED DRUG DOSE; REVIEW; RHABDOMYOLYSIS; RHINOPHARYNGITIS; SIDE EFFECT; TREATMENT RESPONSE; UPPER ABDOMINAL PAIN; VIRUS CELL INTERACTION; VIRUS LOAD; VOMITING;

CLINICAL TRIALS AS TOPIC; DRUG DISCOVERY; HETEROCYCLIC COMPOUNDS, 3-RING; HIV INFECTIONS; HIV INTEGRASE INHIBITORS; HUMANS; PYRROLIDINONES; QUINOLONES;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 84877123280     PISSN: 00126667     EISSN: 11791950     Source Type: Journal    
DOI: 10.1007/s40265-013-0015-5     Document Type: Review

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