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Volumn 8, Issue 4, 2013, Pages 603-613

Effect of C7 Modifications on Benzothiadiazine-1,1-dioxide Derivatives on Their Inhibitory Activity and Selectivity toward Aldose Reductase

(7) Zhang, Shuzhen a Chen, Xin a Parveen, Shagufta a Hussain, Saghir a Yang, Yanchun a Jing, Chaojun a Zhu, Changjin a

a BEIJING INSTITUTE OF TECHNOLOGY (China)

Author keywords

Aldehyde reductase; Aldose reductase; Benzothiadiazines; Inhibitors; Structure activity relationships

Indexed keywords

ALDEHYDE REDUCTASE; BENZOTHIADIAZINE 1,1 DIOXIDE DERIVATIVE; BENZOTHIADIAZINE DERIVATIVE; CARBAMIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; DRUG INHIBITION; DRUG POTENCY; DRUG SELECTIVITY; HYDROPHOBICITY; IC 50; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ALDEHYDE REDUCTASE; ANIMALS; BENZOTHIADIAZINES; BINDING SITES; CATALYTIC DOMAIN; ENZYME INHIBITORS; MOLECULAR DOCKING SIMULATION; PROTEIN BINDING; RATS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84875624311 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201200386 Document Type: Article

Times cited : (19)

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