메뉴 건너뛰기




Volumn 17, Issue 2, 2013, Pages 237-243

Synthesis, characterization and antimicrobial evaluation of novel halopyrazole derivatives

Author keywords

5 Chloro 3 methyl 1 phenylpyrazole 4 carboxaldehyde; Antibacterial activity; Antifungal activity; Pyrazoles

Indexed keywords


EID: 84875482421     PISSN: 13196103     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jscs.2011.03.016     Document Type: Article
Times cited : (84)

References (29)
  • 1
    • 32044442249 scopus 로고    scopus 로고
    • Synthesis and antibacterial activity of some new 1-heteroaryl-5-amino-3H-methyl-4-phenylpyrazoles
    • Agarwal R., Kumar V., Tyagi P., Singh S.P. Synthesis and antibacterial activity of some new 1-heteroaryl-5-amino-3H-methyl-4-phenylpyrazoles. Bioorg. Med. Chem. 2006, 14:1785-1791.
    • (2006) Bioorg. Med. Chem. , vol.14 , pp. 1785-1791
    • Agarwal, R.1    Kumar, V.2    Tyagi, P.3    Singh, S.P.4
  • 2
    • 16244365216 scopus 로고    scopus 로고
    • Antibacterial and antifungal activities of new pyrazolo[3,4-d] pyridazin derivatives
    • Akbas E., Berber I. Antibacterial and antifungal activities of new pyrazolo[3,4-d] pyridazin derivatives. Eur. J. Med. Chem. 2005, 40:401-405.
    • (2005) Eur. J. Med. Chem. , vol.40 , pp. 401-405
    • Akbas, E.1    Berber, I.2
  • 4
    • 40049108415 scopus 로고    scopus 로고
    • Design and synthesis of some substituted 1H-pyrazolyl-thiazolo[4,5-d]pyrimidines as anti-inflammatory, antimicrobial agents
    • Bekhit A.A., Ashour H.M.A., Ghany Y.S.A., Bekhit A.E.A., Baraka A. Design and synthesis of some substituted 1H-pyrazolyl-thiazolo[4,5-d]pyrimidines as anti-inflammatory, antimicrobial agents. Eur. J. Med. Chem. 2008, 43:456-463.
    • (2008) Eur. J. Med. Chem. , vol.43 , pp. 456-463
    • Bekhit, A.A.1    Ashour, H.M.A.2    Ghany, Y.S.A.3    Bekhit, A.E.A.4    Baraka, A.5
  • 5
    • 0038166643 scopus 로고    scopus 로고
    • Comparison of Staphylococcus species. Cellular and extracellular proteins
    • Berber I., Cokmus C., Atalan E. Comparison of Staphylococcus species. Cellular and extracellular proteins. Mikrobiologia 2003, 72:54-55.
    • (2003) Mikrobiologia , vol.72 , pp. 54-55
    • Berber, I.1    Cokmus, C.2    Atalan, E.3
  • 6
    • 0022319015 scopus 로고
    • Incidence of severe side effects during therapy with sulfonylurea and biguanides
    • Berger S. Incidence of severe side effects during therapy with sulfonylurea and biguanides. Horm. Metab. Res. 1985, 17:111-115.
    • (1985) Horm. Metab. Res. , vol.17 , pp. 111-115
    • Berger, S.1
  • 9
    • 33747214078 scopus 로고    scopus 로고
    • Reaction of N-monosubstituted hydrazones with nitroolefins: a novel regioselective pyrazole synthesis
    • Deng X., Mani N.S. Reaction of N-monosubstituted hydrazones with nitroolefins: a novel regioselective pyrazole synthesis. Org. Lett. 2006, 8:3505-3508.
    • (2006) Org. Lett. , vol.8 , pp. 3505-3508
    • Deng, X.1    Mani, N.S.2
  • 10
    • 45549094745 scopus 로고    scopus 로고
    • Base-mediated reaction of hydrazones and nitroolefins with a reversed regioselectivity: a novel synthesis of 1,3,4-trisubstituted pyrazoles
    • Deng X., Mani N.S. Base-mediated reaction of hydrazones and nitroolefins with a reversed regioselectivity: a novel synthesis of 1,3,4-trisubstituted pyrazoles. Org. Lett. 2008, 10:1307-1310.
    • (2008) Org. Lett. , vol.10 , pp. 1307-1310
    • Deng, X.1    Mani, N.S.2
  • 12
    • 77956190055 scopus 로고    scopus 로고
    • Padmashree Synthesis and pharmacological study of 1-acetyl/propyl-3-aryl-5-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-2-pyrazoline
    • Girisha K.S., Kalluraya B., Narayana V., Padmashree Synthesis and pharmacological study of 1-acetyl/propyl-3-aryl-5-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-2-pyrazoline. Eur. J. Med. Chem. 2010, 45:4640-4644.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 4640-4644
    • Girisha, K.S.1    Kalluraya, B.2    Narayana, V.3
  • 14
    • 0035955896 scopus 로고    scopus 로고
    • Preparation of 5-formyl and 5-acetylbarbituric acids, including the corresponding Schiff bases and phenylhydrazones
    • Jursic B.S., Neumann D.M. Preparation of 5-formyl and 5-acetylbarbituric acids, including the corresponding Schiff bases and phenylhydrazones. Tetrahedron Lett. 2001, 42:8435-8439.
    • (2001) Tetrahedron Lett. , vol.42 , pp. 8435-8439
    • Jursic, B.S.1    Neumann, D.M.2
  • 15
    • 0035812782 scopus 로고    scopus 로고
    • Regioselective synthesis of polysubstituted pyrazoles and isoxazoles
    • Katritzky A.R., Wang M., Zhang S., Voronkov M.V. Regioselective synthesis of polysubstituted pyrazoles and isoxazoles. J. Org. Chem. 2001, 66:6787-6791.
    • (2001) J. Org. Chem. , vol.66 , pp. 6787-6791
    • Katritzky, A.R.1    Wang, M.2    Zhang, S.3    Voronkov, M.V.4
  • 17
    • 50949087331 scopus 로고    scopus 로고
    • Synthesis and in vitro antibacterial activity of new steroidal thiosemicarbazone derivatives
    • Khan S.A., Kumar P., Joshi R., Iqbal P.F., Saleem K. Synthesis and in vitro antibacterial activity of new steroidal thiosemicarbazone derivatives. Eur. J. Med. Chem. 2008, 43:2029-2034.
    • (2008) Eur. J. Med. Chem. , vol.43 , pp. 2029-2034
    • Khan, S.A.1    Kumar, P.2    Joshi, R.3    Iqbal, P.F.4    Saleem, K.5
  • 18
    • 68249115313 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity of 4-[5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl]-dihydropyridines and 4-[5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl]-3,4-dihydropyrimidine-2-ones
    • Kumar R., Malik S., Chandra R. Synthesis and antimicrobial activity of 4-[5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl]-dihydropyridines and 4-[5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl]-3,4-dihydropyrimidine-2-ones. Ind. J. Chem. 2009, 48B:718-724.
    • (2009) Ind. J. Chem. , vol.48 B , pp. 718-724
    • Kumar, R.1    Malik, S.2    Chandra, R.3
  • 22
    • 0037931484 scopus 로고
    • Studies on Vilsmeier-Hack reaction: a versatile new synthesis of 5-chloro-3-methylpyrazole-4-carboxaldehyde, 5-chloro-3-methyl-1-phenylpyrazole-4-carboxaldehyde and related fused heterocyclic compounds and heterocyclic Schiff bases
    • Pawar R.A., Patil A.A. Studies on Vilsmeier-Hack reaction: a versatile new synthesis of 5-chloro-3-methylpyrazole-4-carboxaldehyde, 5-chloro-3-methyl-1-phenylpyrazole-4-carboxaldehyde and related fused heterocyclic compounds and heterocyclic Schiff bases. Ind. J. Chem. 1994, 33B:156-158.
    • (1994) Ind. J. Chem. , vol.33 B , pp. 156-158
    • Pawar, R.A.1    Patil, A.A.2
  • 24
    • 38949175741 scopus 로고    scopus 로고
    • Synthesis and antifungal activity of some new 3-hydroxy-2-(1-phenyl-3-aryl-4-pyrazolyl) chromones
    • 43, 435-440. Celecoxib). J. Med. Chem.
    • Prakash, O., Kumar, R., Parkash, V., 2008. Synthesis and antifungal activity of some new 3-hydroxy-2-(1-phenyl-3-aryl-4-pyrazolyl) chromones. Eur. J. Med. Chem. 43, 435-440. Celecoxib). J. Med. Chem. 40, 1347-1365.
    • (2008) Eur. J. Med. Chem. , vol.40 , pp. 1347-1365
    • Prakash, O.1    Kumar, R.2    Parkash, V.3
  • 25
    • 22244478593 scopus 로고    scopus 로고
    • Enterotoxigenic Escherichia coli in developing countries: epidemiology, microbiology, clinical features, treatment, and prevention
    • Qadri F., Svennerholm A.M., Faruque A.S.G., Sack R.B. Enterotoxigenic Escherichia coli in developing countries: epidemiology, microbiology, clinical features, treatment, and prevention. Clin. Microbiol. Rev. 2005, 18:465-483.
    • (2005) Clin. Microbiol. Rev. , vol.18 , pp. 465-483
    • Qadri, F.1    Svennerholm, A.M.2    Faruque, A.S.G.3    Sack, R.B.4
  • 26
    • 75849131926 scopus 로고    scopus 로고
    • New pyrazoles incorporating pyrazolylpyrazole moiety:synthesis, anti-HCV and antitumor activity
    • Riyadh S.M., Farghaly T.A., Abdallah M.A., Abdalla M.M., Abd El-Aziz M.R. New pyrazoles incorporating pyrazolylpyrazole moiety:synthesis, anti-HCV and antitumor activity. Eur. J. Med. Chem. 2010, 45:1042-1050.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 1042-1050
    • Riyadh, S.M.1    Farghaly, T.A.2    Abdallah, M.A.3    Abdalla, M.M.4    Abd El-Aziz, M.R.5
  • 27
    • 20444431197 scopus 로고    scopus 로고
    • Synthesis of (1,4)-naphthoquinono-(3,2-c)-1H-pyrazoles and their (1,4)- naphthohydroquinone derivatives as antifungal, antibacterial and anticancer agents
    • Tandon V.K., Yadav D.B., Chaturvedi A.K., Shukla P.K. Synthesis of (1,4)-naphthoquinono-(3,2-c)-1H-pyrazoles and their (1,4)- naphthohydroquinone derivatives as antifungal, antibacterial and anticancer agents. Bioorg. Med. Chem. Lett. 2005, 15:3288-3291.
    • (2005) Bioorg. Med. Chem. Lett. , vol.15 , pp. 3288-3291
    • Tandon, V.K.1    Yadav, D.B.2    Chaturvedi, A.K.3    Shukla, P.K.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.