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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 8, 2013, Pages 2380-2383

Synthesis and biological activity of 4-substituted benzoxazolone derivatives as a new class of sEH inhibitors with high anti-inflammatory activity in vivo

(6) Tang, Li a Ma, Wen Hua a Ma, Yun Long a Ban, Shu Rong a Feng, Xiu E a Li, Qing Shan a

a SHANXI MEDICAL UNIVERSITY (China)

Author keywords

4 Substituted benzoxazolone; Anti inflammatory activity; sEH inhibitory activity; Synthesis

Indexed keywords

2 BENZOXAZOLONE DERIVATIVE; 4 SUBSTITUTED BENZOXAZOLONE DERIVATIVE; AMINO ACID; ANTIINFLAMMATORY AGENT; CHLORZOXAZONE; UNCLASSIFIED DRUG; XYLENE;

ANTIINFLAMMATORY ACTIVITY; ARTICLE; BIOLOGICAL ACTIVITY; DRUG ACTIVITY; DRUG SYNTHESIS; EAR EDEMA; IC 50; IN VITRO STUDY; IN VIVO STUDY; LIPOPHILICITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTI-INFLAMMATORY AGENTS; BENZOXAZOLES; ENZYME INHIBITORS; EPOXIDE HYDROLASES; HUMANS; MICE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84875477750 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.02.048 Document Type: Article

Times cited : (21)

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