메뉴 건너뛰기




Volumn 29, Issue 2, 2013, Pages 236-248

Development of sustained-release microspheres for the delivery of SAR 1118, an LFA-1 antagonist intended for the treatment of vascular complications of the eye

Author keywords

[No Author keywords available]

Indexed keywords

LIFITEGRAST; LYMPHOCYTE FUNCTION ASSOCIATED ANTIGEN 1; MICROSPHERE; POLYGLACTIN; POLYMER;

EID: 84875038704     PISSN: 10807683     EISSN: 15577732     Source Type: Journal    
DOI: 10.1089/jop.2012.0210     Document Type: Article
Times cited : (15)

References (27)
  • 1
    • 39149121847 scopus 로고    scopus 로고
    • Current and future ophthalmic drug delivery systems. A shift to the posterior segment
    • Del Amo, E.M., & Urtti, A. Current and future ophthalmic drug delivery systems. A shift to the posterior segment. Drug Discov. Today. 13:135-143, 2008.
    • (2008) Drug Discov. Today. , vol.13 , pp. 135-143
    • Del Amo, E.M.1    Urtti, A.2
  • 2
    • 0035980341 scopus 로고    scopus 로고
    • Biodegradable microspheres for vitreoretinal drug delivery
    • Herrero-Vanrell, R., & Refojo, M.F. Biodegradable microspheres for vitreoretinal drug delivery. Adv. Drug Deliv. Rev. 52:5-16, 2001.
    • (2001) Adv. Drug Deliv. Rev. , vol.52 , pp. 5-16
    • Herrero-Vanrell, R.1    Refojo, M.F.2
  • 3
    • 15744404419 scopus 로고    scopus 로고
    • Subconjunctivally administered celecoxib-PLGA microparticles sustain retinal drug levels and alleviate diabetes-induced oxidative stress in a rat model
    • Ayalasomayajula, S.P., & Kompella, U.B. Subconjunctivally administered celecoxib-PLGA microparticles sustain retinal drug levels and alleviate diabetes-induced oxidative stress in a rat model. Eur. J. Pharmacol. 511:191-198, 2005.
    • (2005) Eur. J. Pharmacol. , vol.511 , pp. 191-198
    • Ayalasomayajula, S.P.1    Kompella, U.B.2
  • 4
    • 79954520410 scopus 로고    scopus 로고
    • Recent advances in ophthalmic drug delivery
    • Kompella, U.B., Kadam, R.S., & Lee, V.H. Recent advances in ophthalmic drug delivery. Ther. Deliv. 1:435-456, 2011.
    • (2011) Ther. Deliv. , vol.1 , pp. 435-456
    • Kompella, U.B.1    Kadam, R.S.2    Lee, V.H.3
  • 5
    • 0343247711 scopus 로고    scopus 로고
    • Biodegradation and biocompatibility of PLA and PLGA microspheres
    • Shive, M.S., & Anderson, J.M. Biodegradation and biocompatibility of PLA and PLGA microspheres. Adv. Drug Deliv. Rev. 28:5-24, 1997.
    • (1997) Adv. Drug Deliv. Rev. , vol.28 , pp. 5-24
    • Shive, M.S.1    Anderson, J.M.2
  • 6
    • 41949120596 scopus 로고    scopus 로고
    • Safety evaluation of ocular drug delivery formulations: Techniques and practical considerations
    • Short, B.G. Safety evaluation of ocular drug delivery formulations: techniques and practical considerations. Toxicol. Pathol. 36:49-62, 2008.
    • (2008) Toxicol. Pathol. , vol.36 , pp. 49-62
    • Short, B.G.1
  • 7
    • 0034984424 scopus 로고    scopus 로고
    • Biodegradable polymers for ocular drug delivery
    • Kimura, H., & Ogura, Y. Biodegradable polymers for ocular drug delivery. Ophthalmologica. 215:143-155, 2001.
    • (2001) Ophthalmologica. , vol.215 , pp. 143-155
    • Kimura, H.1    Ogura, Y.2
  • 8
    • 84861184389 scopus 로고    scopus 로고
    • A phase 2 randomized, double-masked, placebocontrolled study of a novel integrin antagonist (SAR 1118) for the treatment of dry eye
    • e1051
    • Semba, C.P., Torkildsen, G.L., Lonsdale, J.D., McLaurin, E.B., Geffin, J.A., Mundorf, T.K., Kennedy, K.S., & Ousler, G.W. A phase 2 randomized, double-masked, placebocontrolled study of a novel integrin antagonist (SAR 1118) for the treatment of dry eye. Am. J. Ophthalmol. 153:1050-1060 e1051, 2012.
    • (2012) Am. J. Ophthalmol. , vol.153 , pp. 1050-1060
    • Semba, C.P.1    Torkildsen, G.L.2    Lonsdale, J.D.3    McLaurin, E.B.4    Geffin, J.A.5    Mundorf, T.K.6    Kennedy, K.S.7    Ousler, G.W.8
  • 11
    • 20044377802 scopus 로고    scopus 로고
    • Optimizing drug delivery systems using systematic "design of experiments." Part I: Fundamental aspects
    • Singh, B., Kumar, R., & Ahuja, N. Optimizing drug delivery systems using systematic "design of experiments." Part I: fundamental aspects. Crit. Rev. Ther. Drug Carrier Syst. 22:27-105, 2005.
    • (2005) Crit. Rev. Ther. Drug Carrier Syst. , vol.22 , pp. 27-105
    • Singh, B.1    Kumar, R.2    Ahuja, N.3
  • 12
    • 23844484653 scopus 로고    scopus 로고
    • Optimizing drug delivery systems using systematic "design of experiments." Part II: Retrospect and prospects
    • Singh, B., Dahiya, M., Saharan, V., & Ahuja, N. Optimizing drug delivery systems using systematic "design of experiments." Part II: retrospect and prospects. Crit. Rev. Ther. Drug Carrier Syst. 22:215-294, 2005.
    • (2005) Crit. Rev. Ther. Drug Carrier Syst. , vol.22 , pp. 215-294
    • Singh, B.1    Dahiya, M.2    Saharan, V.3    Ahuja, N.4
  • 15
    • 33846852628 scopus 로고    scopus 로고
    • Quality by design: Understanding the formulation variables of a cyclosporine A self-nanoemulsified drug delivery systems by Box-Behnken design and desirability function
    • Zidan, A.S., Sammour, O.A., Hammad, M.A., Megrab, N.A., Habib, M.J., & Khan, M.A. Quality by design: understanding the formulation variables of a cyclosporine A self-nanoemulsified drug delivery systems by Box-Behnken design and desirability function. Int. J. Pharm. 332:55-63, 2007.
    • (2007) Int. J. Pharm. , vol.332 , pp. 55-63
    • Zidan, A.S.1    Sammour, O.A.2    Hammad, M.A.3    Megrab, N.A.4    Habib, M.J.5    Khan, M.A.6
  • 16
    • 84946657020 scopus 로고
    • Some new three-level designs for the study of quantitative variables
    • Box, G.E.P., & Behnken, D.W. Some new three-level designs for the study of quantitative variables. Technometrics. 2:455-475, 1960.
    • (1960) Technometrics. , vol.2 , pp. 455-475
    • Box, G.E.P.1    Behnken, D.W.2
  • 17
    • 84862989504 scopus 로고    scopus 로고
    • Intravitreal poly(L-lactide) microparticles sustain retinal and choroidal delivery of TG-0054, a hydrophilic drug intended for neovascular diseases
    • Shelke, N.B., Kadam, R., Tyagi, P., Rao, V.R., & Kompella, U.B. Intravitreal poly(L-lactide) microparticles sustain retinal and choroidal delivery of TG-0054, a hydrophilic drug intended for neovascular diseases. Drug Deliv. Transl. Res. 1:76-90, 2011.
    • (2011) Drug Deliv. Transl. Res. , vol.1 , pp. 76-90
    • Shelke, N.B.1    Kadam, R.2    Tyagi, P.3    Rao, V.R.4    Kompella, U.B.5
  • 18
    • 55949123862 scopus 로고    scopus 로고
    • Assessment of the influence factors on in vitro testing of nasal sprays using Box-Behnken experimental design
    • Guo, C., Stine, K.J., Kauffman, J.F., & Doub, W.H. Assessment of the influence factors on in vitro testing of nasal sprays using Box-Behnken experimental design. Eur. J. Pharm. Sci. 35:417-426, 2008.
    • (2008) Eur. J. Pharm. Sci. , vol.35 , pp. 417-426
    • Guo, C.1    Stine, K.J.2    Kauffman, J.F.3    Doub, W.H.4
  • 19
    • 78349309563 scopus 로고    scopus 로고
    • Optimization of formulation and process variable of nanosuspension: An industrial perspective
    • Singare, D.S., Marella, S., Gowthamrajan, K., Kulkarni, G.T., Vooturi, R., & Rao, P.S. Optimization of formulation and process variable of nanosuspension: an industrial perspective. Int. J. Pharm. 402:213-220, 2010.
    • (2010) Int. J. Pharm. , vol.402 , pp. 213-220
    • Singare, D.S.1    Marella, S.2    Gowthamrajan, K.3    Kulkarni, G.T.4    Vooturi, R.5    Rao, P.S.6
  • 21
    • 55649104973 scopus 로고    scopus 로고
    • Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles
    • Wischke, C., & Schwendeman, S.P. Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles. Int. J. Pharm. 364:298-327, 2008.
    • (2008) Int. J. Pharm. , vol.364 , pp. 298-327
    • Wischke, C.1    Schwendeman, S.P.2
  • 22
    • 0035255916 scopus 로고    scopus 로고
    • Morphology drug distribution, and in vitro release profiles of biodegradable polymeric microspheres containing protein fabricated by double-emulsion solvent extraction/evaporation method
    • Yang, Y.Y., Chung, T.S., & Ng, N.P. Morphology, drug distribution, and in vitro release profiles of biodegradable polymeric microspheres containing protein fabricated by double-emulsion solvent extraction/evaporation method. Biomaterials. 22:231-241, 2001.
    • (2001) Biomaterials. , vol.22 , pp. 231-241
    • Yang, Y.Y.1    Chung, T.S.2    Ng, N.P.3
  • 23
    • 33749457740 scopus 로고    scopus 로고
    • The effect of different grades of PLGA on characteristics of microspheres encapsulated with cyclosporine A
    • Malaekeh-Nikouei, B., Sajadi Tabassi, S.A., & Jaafari, M.R. The effect of different grades of PLGA on characteristics of microspheres encapsulated with cyclosporine A. Curr. Drug Deliv. 3:343-349, 2006.
    • (2006) Curr. Drug Deliv. , vol.3 , pp. 343-349
    • Malaekeh-Nikouei, B.1    Sajadi Tabassi, S.A.2    Jaafari, M.R.3
  • 24
    • 0024264030 scopus 로고
    • Polylactic acid microspheres containing quinidine base and quinidine sulphate prepared by the solvent evaporation method. III. Morphology of the microspheres during dissolution studies
    • Bodmeier, R., & McGinity, J.W. Polylactic acid microspheres containing quinidine base and quinidine sulphate prepared by the solvent evaporation method. III. Morphology of the microspheres during dissolution studies. J. Microencapsul. 5:325-330, 1988.
    • (1988) J. Microencapsul. , vol.5 , pp. 325-330
    • Bodmeier, R.1    McGinity, J.W.2
  • 25
    • 79951901317 scopus 로고    scopus 로고
    • Factors effecting the morphology of eudragit S-100 based microsponges bearing dicyclomine for colonic delivery
    • Jain, V., Jain, D., & Singh, R. Factors effecting the morphology of eudragit S-100 based microsponges bearing dicyclomine for colonic delivery. J. Pharm. Sci. 100:1545-1552, 2010.
    • (2010) J. Pharm. Sci. , vol.100 , pp. 1545-1552
    • Jain, V.1    Jain, D.2    Singh, R.3
  • 26
    • 34147150618 scopus 로고    scopus 로고
    • Estradiol loaded PLGA nanoparticles for oral administration: Effect of polymer molecular weight and copolymer composition on release behavior in vitro and in vivo
    • Mittal, G., Sahana, D.K., Bhardwaj, V., & Ravi Kumar, M.N. Estradiol loaded PLGA nanoparticles for oral administration: effect of polymer molecular weight and copolymer composition on release behavior in vitro and in vivo. J. Control Release. 119:77-85, 2007.
    • (2007) J. Control Release. , vol.119 , pp. 77-85
    • Mittal, G.1    Sahana, D.K.2    Bhardwaj, V.3    Ravi Kumar, M.N.4
  • 27
    • 33846061644 scopus 로고    scopus 로고
    • Particle size analysis in pharmaceutics: Principles, methods and applications
    • Shekunov, B.Y., Chattopadhyay, P., Tong, H.H., and Chow, A.H. Particle size analysis in pharmaceutics: principles, methods and applications. Pharm. Res. 24:203-227, 2007.
    • (2007) Pharm. Res. , vol.24 , pp. 203-227
    • Shekunov, B.Y.1    Chattopadhyay, P.2    Tong, H.H.3    Chow, A.H.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.