Contribution of TRPV1 and multidrug resistance proteins in the permeation of capsaicin across different intestinal regions

International Journal of Pharmaceutics

Volumn 445, Issue 1-2, 2013, Pages 134-140

  Duan, Lian ^a   Yan, Yuan ^a   Sun, Yabin ^a   Zhao, Boxin ^a   Hu, Wenjun ^b   Li, Guofeng ^a  

^a SOUTHERN MEDICAL UNIVERSITY   (China)

^b Institute for Drug and Instrument Control of Guangzhou Military Area   (China)

Author keywords

Capsaicin; Intestinal permeability; Multidrug resistance proteins; Regional difference; TRPV1

Indexed keywords

BREAST CANCER RESISTANCE PROTEIN; CAPSAICIN; MULTIDRUG RESISTANCE PROTEIN 2; NOVOBIOCIN; PROBENECID; RUTHENIUM RED; VANILLOID RECEPTOR 1; VERAPAMIL;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; COLON; CONTROLLED STUDY; DRUG PENETRATION; DRUG TRANSPORT; ILEUM; INTESTINE MUCOSA PERMEABILITY; JEJUNUM; MALE; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; ATP-BINDING CASSETTE TRANSPORTERS; CAPSAICIN; INTESTINAL ABSORPTION; LOWER GASTROINTESTINAL TRACT; MALE; NOVOBIOCIN; P-GLYCOPROTEIN; PERMEABILITY; PROBENECID; RATS; RATS, SPRAGUE-DAWLEY; RUTHENIUM RED; TRPV CATION CHANNELS; VERAPAMIL;

EID: 84874944838     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2013.02.007     Document Type: Article

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