Characterization of a ligand binding site in the human transient receptor potential ankyrin 1 pore

Biophysical Journal

Volumn 104, Issue 4, 2013, Pages 798-806

  Klement, Göran ^a   Eisele, Lina ^a   Malinowsky, David ^a   Nolting, Andreas ^a   Svensson, Mats ^a   Terp, Gitte ^a   Weigelt, Dirk ^a   Dabrowski, Michael ^a  

^a ASTRAZENECA R AND D   (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

A 967079; CALCIUM CHANNEL; LIGAND; NERVE PROTEIN; OXIME; POTASSIUM CHANNEL KV1.2; TRANSIENT RECEPTOR POTENTIAL CHANNEL; TRPA1 PROTEIN, HUMAN;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANIMAL; ARTICLE; BINDING SITE; CHEMISTRY; DRUG ANTAGONISM; GENETICS; HUMAN; METABOLISM; MOLECULAR DOCKING; MOLECULAR GENETICS; POINT MUTATION; PROTEIN TERTIARY STRUCTURE; RAT; SEQUENCE HOMOLOGY; XENOPUS;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANIMALS; BINDING SITES; CALCIUM CHANNELS; HUMANS; KV1.2 POTASSIUM CHANNEL; LIGANDS; MOLECULAR DOCKING SIMULATION; MOLECULAR SEQUENCE DATA; NERVE TISSUE PROTEINS; OXIMES; POINT MUTATION; PROTEIN STRUCTURE, TERTIARY; RATS; SEQUENCE HOMOLOGY; TRANSIENT RECEPTOR POTENTIAL CHANNELS; XENOPUS;

EID: 84874184374     PISSN: 00063495     EISSN: 15420086     Source Type: Journal    
DOI: 10.1016/j.bpj.2013.01.008     Document Type: Article

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