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Volumn 4, Issue 2, 2013, Pages 269-273

Bodilisant - A novel fluorescent, highly affine histamine H3 receptor ligand

Author keywords

BODIPY; displacement; fluorescence confocal laser scanning microscopy; GPCR; H3 receptor; HEK 293 cells; histamine; nonimidazole derivative; pharmacological tool; tissue labeling

Indexed keywords

BODILISANT; CIPROXIFAN; HISTAMINE H3 RECEPTOR; HISTAMINERGIC RECEPTOR AFFECTING AGENT; UNCLASSIFIED DRUG;

EID: 84873947024     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml300383n     Document Type: Article
Times cited : (24)

References (39)
  • 1
    • 84857974978 scopus 로고    scopus 로고
    • Histamine receptor subtypes: S century of rational drug design
    • Walter, M.; Stark, H. Histamine receptor subtypes: S century of rational drug design Front. Biosci. (Schol. Ed.) 2012, 4, 461-488
    • (2012) Front. Biosci. (Schol. Ed.) , vol.4 , pp. 461-488
    • Walter, M.1    Stark, H.2
  • 5
    • 0035847647 scopus 로고    scopus 로고
    • Immunological identification of the mammalian H3 histamine receptor in the mouse brain
    • Chazot, P. L.; Hann, V.; Wilson, C.; Lees, G.; Thompson, C. L. Immunological identification of the mammalian H3 histamine receptor in the mouse brain NeuroReport 2001, 12, 259-262
    • (2001) NeuroReport , vol.12 , pp. 259-262
    • Chazot, P.L.1    Hann, V.2    Wilson, C.3    Lees, G.4    Thompson, C.L.5
  • 7
    • 22244483775 scopus 로고    scopus 로고
    • Technical Aspects of Immunohistochemistry
    • Ramos-Vara, J. A. Technical Aspects of Immunohistochemistry Vet. Pathol. 2005, 42, 405-426
    • (2005) Vet. Pathol. , vol.42 , pp. 405-426
    • Ramos-Vara, J.A.1
  • 9
    • 54849163500 scopus 로고    scopus 로고
    • Fluorescent GPCR ligands as new tools in pharmacology
    • Kuder, K. J.; Kiec-Kononowicz, K. Fluorescent GPCR ligands as new tools in pharmacology Curr. Med. Chem. 2008, 21, 2132-2143
    • (2008) Curr. Med. Chem. , vol.21 , pp. 2132-2143
    • Kuder, K.J.1    Kiec-Kononowicz, K.2
  • 14
    • 36849053388 scopus 로고    scopus 로고
    • BODIPY Dyes and Their Derivatives: Syntheses and Spectroscopic Properties
    • Loudet, A.; Burgess, K. BODIPY Dyes and Their Derivatives: Syntheses and Spectroscopic Properties Chem. Rev. 2007, 107, 4891-4932
    • (2007) Chem. Rev. , vol.107 , pp. 4891-4932
    • Loudet, A.1    Burgess, K.2
  • 15
    • 33748708626 scopus 로고    scopus 로고
    • Synthesis of new, BODIPY-based sensors and labels
    • Kálai, T.; Hideg, K. Synthesis of new, BODIPY-based sensors and labels Tetrahedron 2006, 62, 10352-10360
    • (2006) Tetrahedron , vol.62 , pp. 10352-10360
    • Kálai, T.1    Hideg, K.2
  • 16
    • 67049086245 scopus 로고    scopus 로고
    • Novel Fluorescent Probe for Analysis of Hydroperoxides Based on Boron Dipyrromethane Fluorophore
    • Inoue, N.; Suzuki, Y.; Yokoyama, K.; Karube, I. Novel Fluorescent Probe for Analysis of Hydroperoxides Based on Boron Dipyrromethane Fluorophore Biosci., Biotechnol., Biochem. 2009, 73, 1215-1217
    • (2009) Biosci., Biotechnol., Biochem. , vol.73 , pp. 1215-1217
    • Inoue, N.1    Suzuki, Y.2    Yokoyama, K.3    Karube, I.4
  • 19
    • 1642312091 scopus 로고    scopus 로고
    • Application of fluorescence correlation spectroscopy to the measurement of agonist binding to a G-protein coupled receptor at the single cell level
    • Briddon, S. J.; Middleton, R. J.; Yates, A. S.; George, M. W.; Kellamb, B.; Hill, S. J. Application of fluorescence correlation spectroscopy to the measurement of agonist binding to a G-protein coupled receptor at the single cell level Faraday Discuss. 2004, 126, 197-207
    • (2004) Faraday Discuss. , vol.126 , pp. 197-207
    • Briddon, S.J.1    Middleton, R.J.2    Yates, A.S.3    George, M.W.4    Kellamb, B.5    Hill, S.J.6
  • 21
    • 84857763898 scopus 로고    scopus 로고
    • New potent, short-linker BODIPY-630/650 labelled fluorescent adenosine receptor agonists
    • Dale, C. L.; Hill, S. J.; Kellam, B. New potent, short-linker BODIPY-630/650 labelled fluorescent adenosine receptor agonists Med. Chem. Comm. 2012, 3, 333-338
    • (2012) Med. Chem. Comm. , vol.3 , pp. 333-338
    • Dale, C.L.1    Hill, S.J.2    Kellam, B.3
  • 23
    • 3843100563 scopus 로고    scopus 로고
    • Fluorescent Pirenzepine Derivatives as Potential Bitopic Ligands of the Human M1Muscarinic Receptor
    • Tahtaoui, C.; Parrot, I.; Klotz, P.; Guillier, F.; Galzi, J.-L.; Hibert, M.; Ilien, B. Fluorescent Pirenzepine Derivatives as Potential Bitopic Ligands of the Human M1Muscarinic Receptor J. Med. Chem. 2004, 47, 4300-4315
    • (2004) J. Med. Chem. , vol.47 , pp. 4300-4315
    • Tahtaoui, C.1    Parrot, I.2    Klotz, P.3    Guillier, F.4    Galzi, J.-L.5    Hibert, M.6    Ilien, B.7
  • 24
    • 0024550388 scopus 로고
    • Characterization of Novel Fluorescent Ligands with High Affinity for D1 and D2 Dopaminergic Receptors
    • Monsma, F. J.; Barton, A. C.; Kang, H. C.; Brassard, D. L.; Haugland, R. P.; Sibley, D. R. Characterization of Novel Fluorescent Ligands with High Affinity for D1 and D2 Dopaminergic Receptors J. Neurochem. 1989, 52, 1641-1644
    • (1989) J. Neurochem. , vol.52 , pp. 1641-1644
    • Monsma, F.J.1    Barton, A.C.2    Kang, H.C.3    Brassard, D.L.4    Haugland, R.P.5    Sibley, D.R.6
  • 25
    • 84857467320 scopus 로고    scopus 로고
    • A novel fluorescent histamine H1 receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands
    • Rose, R. H.; Briddon, S. J.; Hill, S. J. A novel fluorescent histamine H1 receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands Br. J. Pharmacol. 2012, 165, 1789-1800
    • (2012) Br. J. Pharmacol. , vol.165 , pp. 1789-1800
    • Rose, R.H.1    Briddon, S.J.2    Hill, S.J.3
  • 26
    • 33745140228 scopus 로고    scopus 로고
    • Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine
    • Xie, S.-X.; Petrache, G.; Schneider, E.; Ye, Q.-Z.; Bernhardt, G.; Seifert, R.; Buschauer, A. Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine Bioorg. Med. Chem. Lett. 2006, 16, 3886-3890
    • (2006) Bioorg. Med. Chem. Lett. , vol.16 , pp. 3886-3890
    • Xie, S.-X.1    Petrache, G.2    Schneider, E.3    Ye, Q.-Z.4    Bernhardt, G.5    Seifert, R.6    Buschauer, A.7
  • 29
    • 84946384343 scopus 로고
    • About the theory of the formation of ethers
    • Williamson, A. About the theory of the formation of ethers Ann. Chem. 1851, 77, 37-49
    • (1851) Ann. Chem. , vol.77 , pp. 37-49
    • Williamson, A.1
  • 30
    • 0001728437 scopus 로고    scopus 로고
    • Are Fluorescence Quantum Yields so Tricky to Measure? A Demonstration Using Familiar Stationary Products
    • Fery-Forgues, S.; Lavabre, D. Are Fluorescence Quantum Yields So Tricky to Measure? A Demonstration Using Familiar Stationary Products J. Chem. Educ. 1999, 76, 1260-1264
    • (1999) J. Chem. Educ. , vol.76 , pp. 1260-1264
    • Fery-Forgues, S.1    Lavabre, D.2
  • 31
    • 0001433022 scopus 로고    scopus 로고
    • Fluorescence Quantum Yields and Their Relation to Lifetime of Rhodamine 6G and Fluorescein in Nine Solvents: Improved Absolute Standards for Quantum Yields
    • Madge, D.; Wong, R.; Seybold, P. G. Fluorescence Quantum Yields and Their Relation to Lifetime of Rhodamine 6G and Fluorescein in Nine Solvents: Improved Absolute Standards for Quantum Yields Photochem. Photobiol. 2002, 75, 327-334
    • (2002) Photochem. Photobiol. , vol.75 , pp. 327-334
    • Madge, D.1    Wong, R.2    Seybold, P.G.3
  • 33
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantification of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford, M. M. A rapid and sensitive method for the quantification of microgram quantities of protein utilizing the principle of protein-dye binding Anal. Biochem. 1976, 72, 248-254
    • (1976) Anal. Biochem. , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 35
    • 57849138847 scopus 로고    scopus 로고
    • Potential utility of histamine H3 receptor antagonist pharmacophore in antipsychotics
    • Von Coburg, Y.; Kottke, T.; Weizel, L.; Ligneau, X.; Stark., H. Potential utility of histamine H3 receptor antagonist pharmacophore in antipsychotics Bioorg. Med. Chem. Lett. 2009, 19, 538-542
    • (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 538-542
    • Von Coburg, Y.1    Kottke, T.2    Weizel, L.3    Ligneau, X.4    Stark, H.5
  • 39
    • 33846790927 scopus 로고    scopus 로고
    • The CD11a Binding Site of Efalizumab in Psoriatic Skin Tissue as Analyzed by Multi-Epitope Ligand Cartography Robot Technology
    • Bonnekoh, B.; Böckelmann, R.; Pommer, A. J.; Malykh, Y.; Phillipsen, L. The CD11a Binding Site of Efalizumab in Psoriatic Skin Tissue as Analyzed by Multi-Epitope Ligand Cartography Robot Technology Skin Pharmacol. Physiol. 2007, 20, 96-111
    • (2007) Skin Pharmacol. Physiol. , vol.20 , pp. 96-111
    • Bonnekoh, B.1    Böckelmann, R.2    Pommer, A.J.3    Malykh, Y.4    Phillipsen, L.5


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