SCOPUS 정보 검색 플랫폼

Volumn 131, Issue 7, 2000, Pages 1247-1250

Distinct pharmacology of rat and human histamine H3 receptors: Role of two amino acids in the third transmembrane domain

(9) Ligneau, X a,b Morisset, S a Tardivel Lacombe, J a Gbahou, F a Ganellin, C R c Stark, H d Schunack, W d Schwartz, J C a Arrang, J M a

a CENTRE PAUL BROCA (France)

b Bioprojet (France)

c UNIVERSITY COLLEGE LONDON (United Kingdom)

d FREIE UNIVERSITÄT BERLIN (Germany)

Author keywords

Ciproxifan; Clobenpropit; FUB 349; G protein coupled receptors; Histamine; Site directed mutagenesis; Thioperamide

Indexed keywords

ALPHA METHYLHISTAMINE; AMINO ACID; AMMONIA; ASPARTIC ACID; CIPROXIFAN; CLOBENPROPIT; COMPLEMENTARY DNA; FUB 349; G PROTEIN COUPLED RECEPTOR; HISTAMINE; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR ANTAGONIST; IODOPROXYFAN; THIOPERAMIDE; UNCLASSIFIED DRUG;

AMINO ACID SUBSTITUTION; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG DISCRIMINATION; DRUG POTENCY; DRUG RECEPTOR BINDING; HUMAN; MOLECULAR CLONING; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; RAT; RECEPTOR AFFINITY; SEQUENCE HOMOLOGY; STRUCTURE ACTIVITY RELATION;

EID: 0033638021 PISSN: 00071188 EISSN: None Source Type: Journal
DOI: 10.1038/sj.bjp.0703712 Document Type: Article

Times cited : (154)

References (16)

1
- 0023819431
- 3-receptors control histamine release in human brain
- (1988) J. Neurochem. , vol.51 , pp. 105-108
- Arrang, J.M.¹ Devaux, B.² Chodkiewicz, J.P.³ Schwartz, J.-C.⁴

2
- 0023653116
- 3-receptors
- (1987) Nature (Lond). , vol.327 , pp. 117-123
- Arrang, J.M.¹ Garbarg, M.² Lancelot, J.C.³ Lecomte, J.M.⁴ Pollard, H.⁵ Robba, M.⁶ Schunack, W.⁷ Schwartz, J.-C.⁸

3
- 0020587209
- 3) of histamine receptor
- (1983) Nature (Lond). , vol.302 , pp. 832-837
- Arrang, J.M.¹ Garbarg, M.² Schwartz, J.-C.³

4
- 0015861774
- 50) of an enzymatic reaction
- (1973) Biochem. Pharmacol. , vol.22 , pp. 3099-3108
- Cheng, Y.C.¹ Prussoff, W.H.²

5
- 0026615172
- 3 receptor negatively coupled to phosphoinositide turnover in the human gastric cell line HGT1
- (1992) J. Biol. Chem. , vol.267 , pp. 25315-25320
- Cherifi, Y.¹ Pigeon, C.² Le Romancer, M.³ Bado, A.⁴ Reyl-Desmars, F.⁵ Lewin, M.J.M.⁶

6
- 0030772640
- International union of pharmacology. XIII. Classification of histamine receptors
- (1997) Pharmacol. Rev. , vol.49 , pp. 253-278
- Hill, S.J.¹ Ganellin, C.R.² Timmerman, H.³ Schwartz, J.-C.⁴ Shankley, N.P.⁵ Young, J.M.⁶ Schunack, W.⁷ Levi, R.⁸ Haas, H.L.⁹

7
- 0028171146
- 3 receptors
- (1994) J. Pharmacol. Exp. Ther. , vol.271 , pp. 452-459
- Ligneau, X.¹ Garbarg, M.² Vizuete, M.L.³ Diaz, J.⁴ Purand, K.⁵ Stark, H.⁶ Schunack, W.⁷ Schwartz, J.-C.⁸

8
- 0032463756
- 3-receptor antagonist
- (1998) J. Pharmacol. Exp. Ther. , vol.287 , pp. 658-666
- Ligneau, X.¹ Lin, J.-S.² Vanni-Mercier, G.³ Jouvet, M.⁴ Muir, J.L.⁵ Ganellin, C.R.⁶ Stark, H.⁷ Elz, S.⁸ Schunack, W.⁹ Schwartz, J.-C.¹⁰

9
- 0034047202
- 3 receptor reveals distinct species pharmacological profiles
- (2000) J. Pharmacol. Exp. Ther. , vol.293 , pp. 771-778
- Lovenberg, T.W.¹ Pyati, J.² Chang, H.³ Wilson, S.J.⁴ Erlander, M.G.⁵

10
- 0033051582
- 3 receptor
- (1999) Mol. Pharmacol. , vol.56 , pp. 1101-1107
- Lovenberg, T.W.¹ Roland, B.L.² Wilson, S.J.³ Jiang, X.⁴ Pyati, J.⁵ Huvar, A.⁶ Jackson, M.R.⁷ Erlander, M.G.⁸

11
- 0015049463
- Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists
- (1971) J. Pharmacol. Exp. Ther. , vol.177 , pp. 1-12
- Parker, R.B.¹ Waud, D.R.²

12
- 2642708346
- 3-receptor antagonist of high oral in vivo potency with 4(ω-(arylalkyloxy)alkyl)-1H-imidazole structure
- (1998) Arch. Pharm. Pharm. Med. Chem. , vol.331 , pp. 211-218
- Stark, H.¹ Huls, A.² Ligneau, X.³ Purand, K.⁴ Pertz, H.⁵ Arrang, J.M.⁶ Schwartz, J.-C.⁷ Schunack, W.⁸

13
- 0032483065
- 3-receptor antagonists: Change of a paradigm
- (1998) Bioorg. Med. Chem. Lett. , vol.8 , pp. 2011-2016
- Stark, H.¹ Ligneau, X.² Arrang, J.M.³ Schwartz, J.-C.⁴ Schunack, W.⁵

14
- 0034689572
- 3 receptor: Evidence for two isoforms
- (2000) NeuroReport , vol.11 , pp. 775-759
- Tardivel-Lacombe, J.¹ Rouleau, A.² Heron, A.³ Morisset, S.⁴ Pillot, C.⁵ Cochois, V.⁶ Schwartz, J.-C.⁷ Arrang, J.M.⁸

15
- 0026788102
- 3-receptor
- (1992) Eur. J. Med Chem. , vol.27 , pp. 511-517
- Van Der Goot, H.¹ Schepers, M.J.P.² Sterk, G.J.³ Timmerman, H.⁴

16
- 0345593406
- 3H]N(α)-methylhistamine binding differ from that of rodents
- (1999) Eur. J. Pharmacol. , vol.377 , pp. 233-239
- West R.E., Jr.¹ Wu, R.L.² Billah, M.M.³ Egan, R.W.⁴ Anthes, J.C.⁵

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.