Potential utility of histamine H3 receptor antagonist pharmacophore in antipsychotics

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 2, 2009, Pages 538-542

  von Coburg, Y ^a   Kottke, T ^a   Weizel, L ^a   Ligneau, X ^b   Stark, H ^a  

^a GOETHE UNIVERSITY   (Germany)

^b Bioprojet Biotech   (France)

Author keywords

[No Author keywords available]

Indexed keywords

AMITRIPTYLINE; CHLORPROMAZINE; CHLORPROTHIXENE; CLOZAPINE; FLUPHENAZINE; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR ANTAGONIST; MAPROTILINE; NEUROLEPTIC AGENT;

ARTICLE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; PHARMACOPHORE; RECEPTOR AFFINITY; STRUCTURE ANALYSIS;

ANIMALS; ANTIPSYCHOTIC AGENTS; CELL LINE; CHO CELLS; CRICETINAE; CRICETULUS; HISTAMINE ANTAGONISTS; HUMANS; RADIOLIGAND ASSAY; RECEPTORS, HISTAMINE H3;

EID: 57849138847     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.09.012     Document Type: Article

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