Fluorescent GPCR ligands as new tools in pharmacology

Current Medicinal Chemistry

Volumn 15, Issue 21, 2008, Pages 2132-2143

  Kuder, Kamil ^a   Kieć Kononowicz, Katarzyna ^a  

^a JAGIELLONIAN UNIVERSITY MEDICAL COLLEGE   (Poland)

Author keywords

Flourescent ligands; Fluorescence; Fluorophores; GPCRs

Indexed keywords

1 FLUORO 2,4 DINITROBENZENE; 1 NAPHTHALENESULFONIC ACID [4 [(4 AMINO 2 QUINAZOLINYLAMINO)METHYL]CYCLOHEXYLMETHYL]AMIDE; 2 PHENYLIMIDAZO[1,2 A]PYRIDINE DERIVATIVE; 4 (3 TERT BUTYLAMINO 2 HYDROXYPROPOXY) 2 BENZIMIDAZOLONE; ADENOSINE 5' (N ETHYLCARBOXAMIDE) DERIVATIVE; ADRENERGIC RECEPTOR LIGAND; ALEXA 532; AMINOPOTENTIDINE DERIVATIVE; CANNABINOID 2 RECEPTOR LIGAND; CYANINE DYE; DOPAMINE RECEPTOR LIGAND; DYE; FLUORESCENT DYE; FLUORESCENT G PROTEIN COUPLED RECEPTOR LIGAND; HISTAMINE H1 RECEPTOR LIGAND; HISTAMINE H2 RECEPTOR LIGAND; HISTAMINE H3 RECEPTOR LIGAND; IODOPOTENTIDINE I 125; MUSCARINIC RECEPTOR LIGAND; NALPHA (DIPHENYLACETYL) N (4 HYDROXYBENZYL) DEXTRO ARGININAMIDE DERIVATE; NAPHTHALIMIDE DERIVATIVE; NEUROPEPTIDE Y1 RECEPTOR LIGAND; NEUROPEPTIDE Y5 RECEPTOR LIGAND; NITROBENZOXADIAZOLE; NORADRENALIN; PIRENZEPINE; RADIOLIGAND; SEROTONIN 1A RECEPTOR LIGAND; SEROTONIN 4 RECEPTOR LIGAND; UNCLASSIFIED DRUG; UNINDEXED DRUG; G PROTEIN COUPLED RECEPTOR; LIGAND;

BINDING AFFINITY; CONFOCAL MICROSCOPY; DRUG RESEARCH; EPIFLUORESCENCE MICROSCOPY; FLUORESCENCE ANALYSIS; FLUORESCENCE CORRELATION SPECTROSCOPY; FLUORESCENCE RESONANCE ENERGY TRANSFER; HUMAN; LIGAND BINDING; NONHUMAN; PROTEIN ANALYSIS; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR OCCUPANCY; REVIEW; ANIMAL; BINDING SITE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECT; METABOLISM;

ANIMALS; BINDING SITES; FLUORESCENT DYES; HUMANS; LIGANDS; MOLECULAR STRUCTURE; RECEPTORS, G-PROTEIN-COUPLED;

EID: 54849163500     PISSN: 09298673     EISSN: None     Source Type: Journal    
DOI: 10.2174/092986708785747599     Document Type: Review

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