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Applications of fluorescence- and bioluminescence-resonance energy transfer to drug discovery at G protein-coupled receptors
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E. Alvarez-Curto, J.D. Pediani, and G. Milligan Applications of fluorescence- and bioluminescence-resonance energy transfer to drug discovery at G protein-coupled receptors Analytical and Bioanalytical Chemistry 398 2010 167 180
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Developing chemical genetic approaches to explore G protein-coupled receptor function: Validation of the use a Receptor Activated Solely by Synthetic Ligand (RASSL)
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3 muscarinic acetylcholine receptors analyzed by fluorescence resonance energy transfer (FRET) imaging and homogenous time-resolved FRET
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Cell surface delivery and structural re-organisation by pharmacological chaperones of an oligomerisation-defective alpha(1b)-adrenoceptor mutants demonstrates membrane targeting of GPCR oligomers
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Cell-surface protein-protein interaction analysis with time-resolved FRET and SNAP-tag technologies: Application to GPCR oligomerisation
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G protein coupled receptor dimerisation: Molecular basis and relevance to function
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A day in the life of a G-protein coupled receptor: The contribution to function of G-protein coupled receptor dimerisation
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The role of dimerisation in the cellular trafficking of G-protein-coupled receptors
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CXCR2 chemokine receptor antagonism enhances DOP opioid receptor function via allosteric regulation of the CXCR2-DOP receptor heterodimer
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A monomeric G-protein coupled receptor isolated in a high-density lipoprotein particle efficiently activates its G protein
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