Leucettamols, bifunctionalized marine sphingoids, act as modulators of TRPA1 and TRPM8 channels

Marine Drugs

Volumn 10, Issue 11, 2012, Pages 2435-2447

  Chianese, Giuseppina ^a   Fattorusso, Ernesto ^a   Putra, Masteria Yunovilsa ^a,b   Calcinai, Barbara ^b   Bavestrello, Giorgio ^c   Schiano Moriello, Aniello ^d   De Petrocellis, Luciano ^d   Di Marzo, Vincenzo ^e   Taglialatela Scafati, Orazio ^a  

^a UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^b UNIVERSITÀ POLITECNICA DELLE MARCHE   (Italy)

^c UNIVERSITY OF GENOA   (Italy)

^d CNR   (Italy)

^e CNR Consiglio Nazionale delle Ricerche   (Italy)

Author keywords

Leucettamols; Pain modulation; TRP receptors

Indexed keywords

CANNABINOID 1 RECEPTOR; CANNABINOID 2 RECEPTOR; LEUCETTAMOL A; LEUCETTAMOL B; LEUCETTAMOL DERIVATIVE; NATURAL PRODUCT; TRANSIENT RECEPTOR POTENTIAL CHANNEL A1; TRANSIENT RECEPTOR POTENTIAL CHANNEL M8; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CELL STRAIN HEK293; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFICACY; DRUG ISOLATION; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG TARGETING; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; INHIBITION KINETICS; LEUCETTA; NEUROMODULATION; NONHUMAN; RAT; SPONGE (PORIFERA); STABLE TRANSFECTION; STRUCTURE ACTIVITY RELATION;

EID: 84870045413     PISSN: None     EISSN: 16603397     Source Type: Journal    
DOI: 10.3390/md10112435     Document Type: Article

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