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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 19, 2012, Pages 6233-6236

Synthesis, radiolabeling and initial in vivo evaluation of [ 11C]KSM-01 for imaging PPAR-α receptors

(10) Solingapuram Sai, Kiran Kumar a Kil, Kun Eek a Tu, Zhude a Chu, Wenhua a Finck, Brian N a Rothfuss, Justin M a Shoghi, Kooresh I a Welch, Michael J a Gropler, Robert J a Mach, Robert H a

a WASHINGTON UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

Oxidation; Cardiomyopathy; Peroxisome proliferator activated receptor alpha (PPAR ); PET imaging; Ureido thioisobutyric acid (TiBA)

Indexed keywords

2 [4 [2 [3 CYCLOHEXYL 1 (4 CYCLOHEXYLBUTYL)UREIDO]ETHYL]PHENYLTHIO] 2 METHYLPROPIONIC ACID; P METHOXY PHENYL UREIDO THIOBUTYRIC ACID DERIVATIVE C 11; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA AGONIST; RADIOISOTOPE; RADIOPHARMACEUTICAL AGENT; SODIUM HYDROXIDE; UNCLASSIFIED DRUG;

ALKYLATION; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; COMPUTER ASSISTED EMISSION TOMOGRAPHY; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG DISTRIBUTION; DRUG SCREENING; DRUG SYNTHESIS; GENE OVEREXPRESSION; HUMAN; HUMAN CELL; IN VIVO STUDY; ISOTOPE LABELING; MALE; MOUSE; NONHUMAN; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION; WILD TYPE;

ANIMALS; BUTYRATES; HUMANS; ISOTOPE LABELING; MICE; MICE, TRANSGENIC; PHENYLUREA COMPOUNDS; POSITRON-EMISSION TOMOGRAPHY; PPAR ALPHA; RADIOPHARMACEUTICALS; TISSUE DISTRIBUTION; TOMOGRAPHY, X-RAY COMPUTED;

MUS MUSCULUS;

EID: 84866369043 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.08.010 Document Type: Article

Times cited : (11)

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