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Volumn 7, Issue 9, 2012, Pages 1601-1611

An Efficient Synthesis of a Hydroxyethylamine (HEA) Isostere and Its α-Aminophosphonate and Phosphoramidate Derivatives as Potential Anti-HIV Agents

(4) Bhattacharya, Asish K a Rana, Kalpeshkumar C a Pannecouque, Christophe b DeClercq, Eric b

a NATIONAL CHEMICAL LABORATORY (India)

b REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

Author keywords

aminophosphonates; Antiviral agents; Hydroxyethylamine isosteres; Phosphoramidates; Synthesis

Indexed keywords

ALPHA AMINOPHOSPHONATE; AMPRENAVIR; ANTIVIRUS AGENT; HYDROXYETHYLAMINE ISOSTERE; INDINAVIR; NELFINAVIR; PHOSPHORAMIDIC ACID DERIVATIVE; RITONAVIR; SAQUINAVIR; UNCLASSIFIED DRUG;

ACQUIRED IMMUNE DEFICIENCY SYNDROME; ANTIVIRAL ACTIVITY; ARTICLE; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; MUTANT; NONHUMAN; ONE POT SYNTHESIS; PRIORITY JOURNAL; VIRUS STRAIN; WILD TYPE;

AMIDES; CELL LINE; ETHYLAMINES; HIV; HIV INFECTIONS; HIV PROTEASE INHIBITORS; HUMANS; MODELS, MOLECULAR; PHOSPHORIC ACIDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84865583060 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201200271 Document Type: Article

Times cited : (46)

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