Cinnamic Acid/Chloroquinoline Conjugates as Potent Agents against Chloroquine-Resistant Plasmodium falciparum

ChemMedChem

Volumn 7, Issue 9, 2012, Pages 1537-1540

  Pérez, Bianca ^a   Teixeira, Cátia ^a,b   Gut, Jiri ^c   Rosenthal, Philip J ^c   Gomes, José R B ^b   Gomes, Paula ^a  

^a UNIVERSITY OF PORTO   (Portugal)

^b UNIVERSITY OF AVEIRO   (Portugal)

^c UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Aminoquinolines; Cinnamic acids; Malaria; Permeability pathways; Plasmodium falciparum

Indexed keywords

ANTIMALARIAL AGENT; ARTEMISININ; CHLOROQUINE; CINNAMIC ACID CHLOROQUINE CONJUGATE; PRIMAQUINE; UNCLASSIFIED DRUG;

ANTIMALARIAL ACTIVITY; ANTIMALARIAL DRUG RESISTANCE; ARTICLE; CRYSTALLIZATION; ERYTHROCYTE; IC 50; IN VITRO STUDY; LIPOPHILICITY; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL;

ANTIMALARIALS; CHLOROQUINE; CINNAMATES; DRUG RESISTANCE; ERYTHROCYTES; HUMANS; MALARIA, FALCIPARUM; PLASMODIUM FALCIPARUM;

EID: 84865578263     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.201200257     Document Type: Article

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