Tuned-affinity bivalent ligands for the characterization of opioid receptor heteromers

ACS Medicinal Chemistry Letters

Volumn 3, Issue 8, 2012, Pages 640-644

  Harvey, Jessica H ^a,b   Long, Darcie H ^a   England, Pamela M ^b   Whistler, Jennifer L ^a,b  

^a UNIVERSITY OF CALIFORNIA SAN FRANCISCO   (United States)

^b UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

bivalent ligand; chronic pain; heteromers; opioid receptors

Indexed keywords

DELTA OPIATE RECEPTOR; LIGAND; MU OPIATE RECEPTOR; NALTREXONE; OXYMORPHONE;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG DESIGN; DRUG SYNTHESIS; PAIN; PHARMACOPHORE; PRIORITY JOURNAL;

EID: 84864982116     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml300083p     Document Type: Article

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