Thiosuccinyl peptides as Sirt5-specific inhibitors

Journal of the American Chemical Society

Volumn 134, Issue 4, 2012, Pages 1922-1925

  He, Bin ^a   Du, Jintang ^a,b   Lin, Hening ^a  

^a Department of Obstetrics Gynecology   (United States)

^b SCRIPPS RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYL GROUPS; ACYL GROUP; BIOLOGICAL PROCESS; DRUG DEVELOPMENT; HUMAN DISEASE; LYSINE RESIDUES; NICOTINAMIDE ADENINE; SIRTUIN; SMALL MOLECULES; SPECIFIC INHIBITORS;

AMIDES; AMINO ACIDS;

PEPTIDES;

AMINO ACID; HISTONE DEACETYLASE INHIBITOR; HISTONE H3 LYSINE 9 THIOSUCCINYL PEPTIDE; LYSINE; SIRTUIN 5; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; HUMAN; PROTEIN HYDROLYSIS;

ENZYME INHIBITORS; HUMANS; MOLECULAR STRUCTURE; PEPTIDES; SIRTUINS; STRUCTURE-ACTIVITY RELATIONSHIP; SUCCINATES; SULFHYDRYL COMPOUNDS;

EID: 84863010942     PISSN: 00027863     EISSN: 15205126     Source Type: Journal    
DOI: 10.1021/ja2090417     Document Type: Article

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