-
1
-
-
0004043489
-
-
Wiley Interscience, John Wiley and Sons, New York
-
G. Lombardino, "Nonsteroidal Antiinflammatory Drugs", Wiley Interscience, John Wiley and Sons, New York, 1985, pp. 97-107.
-
(1985)
Nonsteroidal Antiinflammatory Drugs
, pp. 97-107
-
-
Lombardino, G.1
-
2
-
-
0342647359
-
6-Benzylidenethiazolo[3,2-b]-1,2,4-triazole-5(6H)-ones substituted with ibuprofen: Synthesis, characterization and evaluation of anti-inflammatory activity
-
B. Tozkoparan, N. Gökhan, G. Aktay, E. Yeşilada and M. Ertan, "6-Benzylidenethiazolo[3,2-b]-1,2,4-triazole-5(6H)-ones substituted with ibuprofen: synthesis, characterization and evaluation of anti-inflammatory activity", Eur. J. Med. Chem., 35, 743-750 (2000).
-
(2000)
Eur. J. Med. Chem.
, vol.35
, pp. 743-750
-
-
Tozkoparan, B.1
Gökhan, N.2
Aktay, G.3
Yeşilada, E.4
Ertan, M.5
-
3
-
-
34447267965
-
1-Acylthiosemicarbazides, 1,2,4-triazole-5(4H)-thiones,1,3,4-thiadiazoles and hydrazones containing 5-methyl-2-benzoxazolinones: Synthesis, analgesic-anti-inflammatory and antimicrobial activities
-
U. Salgin-Göksen, N. Gökhan-Kelekç Ö. Göktas, Y. Köysal, E. Kiliç, Ş. IşiK, G. Aktay and M. Özalp, "1-Acylthiosemicarbazides, 1,2,4-triazole-5(4H)-thiones,1,3,4- thiadiazoles and hydrazones containing 5-methyl-2-benzoxazolinones: Synthesis, analgesic-anti-inflammatory and antimicrobial activities", Bioorg. & Med. Chem., 15, 5738-5751 (2007).
-
(2007)
Bioorg. & Med. Chem.
, vol.15
, pp. 5738-5751
-
-
Salgin-Göksen, U.1
Gökhan-Kelekç, N.2
Göktas, Ö.3
Köysal, Y.4
Kiliç, E.5
IşiK, Ş.6
Aktay, G.7
Özalp, M.8
-
5
-
-
1242339542
-
Synthesis and biological evaluations of novel benzimidazoles as potential antibacterial agents
-
Y. He, J. Yang, B. Wu, L. Risen and E. E. Swayze, "Synthesis and biological evaluations of novel benzimidazoles as potential antibacterial agents", Bioorg. & Med. Chem. lett., 14, 1217-1220 (2004).
-
(2004)
Bioorg. & Med. Chem. Lett.
, vol.14
, pp. 1217-1220
-
-
He, Y.1
Yang, J.2
Wu, B.3
Risen, L.4
Swayze, E.E.5
-
6
-
-
61349171339
-
Convenient one pot synthesis of novel 2-substituted benzimidazoles, tetrahydrobenzimidazoles and imidazoles and evaluation of their in-vitro antibacterial and antifungal activities
-
S. Sharma, S. Gangal and A. Rauf, "Convenient one pot synthesis of novel 2-substituted benzimidazoles, tetrahydrobenzimidazoles and imidazoles and evaluation of their in-vitro antibacterial and antifungal activities", Eur. J. Med. Chem., 44, 1751-1757 (2009).
-
(2009)
Eur. J. Med. Chem.
, vol.44
, pp. 1751-1757
-
-
Sharma, S.1
Gangal, S.2
Rauf, A.3
-
7
-
-
62749112851
-
Synthesis, pharmacological screening, quantum chemical and in-vitro permeability studies of N-Mannich bases of benzimidazoles through bovine cornea
-
E. P. Jesudason, S. K. Sridhar, E. P. Malar, P. Shanmuggapandiyan, M. Inayathullah, V. Arul, D. Selvaraj and R. Jayakumar, "Synthesis, pharmacological screening, quantum chemical and in-vitro permeability studies of N-Mannich bases of benzimidazoles through bovine cornea", ibid., 44, 2307-2312 (2009).
-
(2009)
Eur. J. Med. Chem.
, vol.44
, pp. 2307-2312
-
-
Jesudason, E.P.1
Sridhar, S.K.2
Malar, E.P.3
Shanmuggapandiyan, P.4
Inayathullah, M.5
Arul, V.6
Selvaraj, D.7
Jayakumar, R.8
-
8
-
-
75749088570
-
Structure-Based Design of Benzimidazole Sugar Conjugates: Synthesis, SAR and in-vivo Anti-inflammatory and Analgesic Activities
-
A. O. El-Nezhawy, S. T. Gaballah, M. A. Radwan, A. R. Baiuomy and O. M. Abdel-Salam, "Structure-Based Design of Benzimidazole Sugar Conjugates: Synthesis, SAR and in-vivo Anti-inflammatory and Analgesic Activities", Medicinal Chemistry, 5, 558-569 (2009).
-
(2009)
Medicinal Chemistry
, vol.5
, pp. 558-569
-
-
El-Nezhawy, A.O.1
Gaballah, S.T.2
Radwan, M.A.3
Baiuomy, A.R.4
Abdel-Salam, O.M.5
-
9
-
-
1842664458
-
Synthesis of 5-(2-,3- and 4-methoxyphenyl)-4H-1,2,4-triazole-3-thiol derivatives exhibiting anti-inflammatory activity
-
L. Labanauskas, E. Udrenaite, P. Gaidelis and A. Brukştus, "Synthesis of 5-(2-,3- and 4-methoxyphenyl)-4H-1,2,4-triazole-3-thiol derivatives exhibiting anti-inflammatory activity", Il Farmaco, 59, 255-259 (2004).
-
(2004)
Il Farmaco
, vol.59
, pp. 255-259
-
-
Labanauskas, L.1
Udrenaite, E.2
Gaidelis, P.3
Brukştus, A.4
-
10
-
-
60149087906
-
Synthesis, analgesic, anti-inflammatory and antimicrobial studies of 2,4-dichoro-5-fluorophenyl containing thiazolotriazoles
-
M. S. Karthikeyan, "Synthesis, analgesic, anti-inflammatory and antimicrobial studies of 2,4-dichoro-5-fluorophenyl containing thiazolotriazoles", Eur. J. Med. Chem., 44, 827-833 (2009).
-
(2009)
Eur. J. Med. Chem.
, vol.44
, pp. 827-833
-
-
Karthikeyan, M.S.1
-
11
-
-
34249330953
-
Discovery of novel indazole-linked triazoles as antifungal agents
-
J. S. Park, K. A. Yu, T. H. Kang, S. Kim and Y. G. Suh, "Discovery of novel indazole-linked triazoles as antifungal agents", Bioorg. & Med. Chem. lett., 17, 3486-3400 (2007).
-
(2007)
Bioorg. & Med. Chem. Lett.
, vol.17
, pp. 3486-13400
-
-
Park, J.S.1
Yu, K.A.2
Kang, T.H.3
Kim, S.4
Suh, Y.G.5
-
12
-
-
67349229119
-
Synthesis of some new 1,3,4-thiadiazol-2-ylmethyl-1,2,4-triazole derivatives and investigation of their antimicrobial activities
-
A. Demirbas, D. Sahin, N. Demirbas and S. A. Karaoglu, "Synthesis of some new 1,3,4-thiadiazol-2-ylmethyl-1,2,4-triazole derivatives and investigation of their antimicrobial activities", Eur. J. Med. Chem., 44, 2896-2903 (2009).
-
(2009)
Eur. J. Med. Chem.
, vol.44
, pp. 2896-2903
-
-
Demirbas, A.1
Sahin, D.2
Demirbas, N.3
Karaoglu, S.A.4
-
13
-
-
85069129975
-
Synthesis of some new benzimidazole derivatives with potential antimicrobial activity
-
N. Sharaf El-Din, "Synthesis of some new benzimidazole derivatives with potential antimicrobial activity", Zagazig J. Pharm. Sci., 4 (2), 198-203 (1995).
-
(1995)
Zagazig J. Pharm. Sci.
, vol.4
, Issue.2
, pp. 198-203
-
-
Sharaf El-Din, N.1
-
14
-
-
33144465711
-
Synthesis and antimicrobial activity of some new 1-alkyl-2-alkylthio-1,2, 4-triazolobenzimidazole derivatives
-
B.G. Mohammad, M. A. Hussein, A.M. Abdel-Alim and M. Hashem, "Synthesis and antimicrobial activity of some new 1-alkyl-2-alkylthio-1,2, 4-triazolobenzimidazole derivatives", Arch. Pharm. Res., 29, 26-33 (2006).
-
(2006)
Arch. Pharm. Res.
, vol.29
, pp. 26-33
-
-
Mohammad, B.G.1
Hussein, M.A.2
Abdel-Alim, A.M.3
Hashem, M.4
-
15
-
-
0030555985
-
Synthesis and reactions of 2-mercaptomethyl-1,3,4-oxadiazolin-5-one
-
M. M. Hamad, S. A. Said and Y. M. El-Ekyabi, "Synthesis and reactions of 2-mercaptomethyl-1,3,4-oxadiazolin-5-one", Monastshefte für Chemie., 127, 549-555 (1996).
-
(1996)
Monastshefte für Chemie
, vol.127
, pp. 549-555
-
-
Hamad, M.M.1
Said, S.A.2
El-Ekyabi, Y.M.3
-
16
-
-
32844460667
-
Synthesis of 1-Acyl-2-alkylthio-1,2,4-triazolobenzimidazoles with Antifungal, Anti-inflammatory and Analgesic effects
-
B. G. Mohammad, M. A. Hussein, A. M. Abdel-Alim and M. Hashem, "Synthesis of 1-Acyl-2-alkylthio-1,2,4-triazolobenzimidazoles with Antifungal, Anti-inflammatory and Analgesic effects", Acta. Pharm., 56, 31-48 (2006).
-
(2006)
Acta. Pharm.
, vol.56
, pp. 31-48
-
-
Mohammad, B.G.1
Hussein, M.A.2
Abdel-Alim, A.M.3
Hashem, M.4
-
17
-
-
0037046859
-
Hydrazones of 1,2-benzisothiazole hydrazides: Synthesis, antimicrobial activity and QSAR investigations
-
P. Vicini, F. Zani, P. Cozzini and I. Doytchinova, "Hydrazones of 1,2-benzisothiazole hydrazides: synthesis, antimicrobial activity and QSAR investigations", Eur. J. Med. Chem. 37, 553-564 (2002).
-
(2002)
Eur. J. Med. Chem.
, vol.37
, pp. 553-564
-
-
Vicini, P.1
Zani, F.2
Cozzini, P.3
Doytchinova, I.4
-
18
-
-
34247581707
-
A new class of nifuroxazide analogues: Synthesis of 5-nitrothiophene derivatives with antimicrobial activity against multidrug-resistant Staphylococcus aureus
-
A. Masunari and L. C. Tavares, "A new class of nifuroxazide analogues: Synthesis of 5-nitrothiophene derivatives with antimicrobial activity against multidrug-resistant Staphylococcus aureus", Bioorg. & Med. Chem., 15, 4229-4236 (2007).
-
(2007)
Bioorg. & Med. Chem.
, vol.15
, pp. 4229-4236
-
-
Masunari, A.1
Tavares, L.C.2
-
19
-
-
0034064517
-
Synthesis and analgesic activity of novel Nacylarylhydrazones and isosters, derived from natural safrole
-
P. C. Lima, L. M. Lima, K. C. Silva, P. H. Léda, A. L. P. Miranda, C. A. M. Fraga and E. J. Barreiro, "Synthesis and analgesic activity of novel Nacylarylhydrazones and isosters, derived from natural safrole", Eur. J. Med. Chem., 35, 187-203 (2000).
-
(2000)
Eur. J. Med. Chem.
, vol.35
, pp. 187-203
-
-
Lima, P.C.1
Lima, L.M.2
Silva, K.C.3
Léda, P.H.4
Miranda, A.L.P.5
Fraga, C.A.M.6
Barreiro, E.J.7
-
20
-
-
0033800136
-
Synthesis and pharmacological evaluation of novel heterotricyclic acylhydrazone derivatives, designed as PAF antagonists
-
A. G. M. Fraga, C. R. Rodrigues, A. L. P. Miranda, E. J. Barreiro and C. A. M. Fraga, "Synthesis and pharmacological evaluation of novel heterotricyclic acylhydrazone derivatives, designed as PAF antagonists", Eur. J. Pharm. Sci., 11, 285-290 (2000).
-
(2000)
Eur. J. Pharm. Sci.
, vol.11
, pp. 285-290
-
-
Fraga, A.G.M.1
Rodrigues, C.R.2
Miranda, A.L.P.3
Barreiro, E.J.4
Fraga, C.A.M.5
-
21
-
-
0036203802
-
Synthesis, antibacterial, antifungal and genotoxic activity of bis-1,3,4-oxadiazole derivatives
-
A. O. Maslat, M. Abussaud, H. Tashtoush and M. AL-Talib, "Synthesis, antibacterial, antifungal and genotoxic activity of bis-1,3,4-oxadiazole derivatives", Pol. J. Pharmacol., 54, 55-59 (2002).
-
(2002)
Pol. J. Pharmacol.
, vol.54
, pp. 55-59
-
-
Maslat, A.O.1
Abussaud, M.2
Tashtoush, H.3
Al-Talib, M.4
-
22
-
-
70349560719
-
Synthesis, evaluation and characterization of some 1,3,4-oxadiazoles as antimicrobial agents
-
N. BhardWaj, S. K. Saraf, P. Sharma and P. Kumar, "Synthesis, evaluation and characterization of some 1,3,4-oxadiazoles as antimicrobial agents", E-Journal of Chemistry, 6 (4), 1133-1138 (2009).
-
(2009)
E-Journal of Chemistry
, vol.6
, Issue.4
, pp. 1133-1138
-
-
BhardWaj, N.1
Saraf, S.K.2
Sharma, P.3
Kumar, P.4
-
23
-
-
34548531844
-
Anti-inflammatory, analgesic, ulcerogenic activities of some new non-acidic diclofenac and 1,3,4-oxadiazole derivatives in animal models
-
M. K. Raut, S. V. Bhandari, K. G. Bothara, A. A. Patil and A. P. Sarkate, "Anti-inflammatory, analgesic, ulcerogenic activities of some new non-acidic diclofenac and 1,3,4-oxadiazole derivatives in animal models", Pharmacologyonline, 2, 172-186 (2007).
-
(2007)
Pharmacologyonline
, vol.2
, pp. 172-186
-
-
Raut, M.K.1
Bhandari, S.V.2
Bothara, K.G.3
Patil, A.A.4
Sarkate, A.P.5
-
24
-
-
84862851347
-
Synthesis and evaluation of anti-inflammatory and antimicrobial activities of 2,5-disubstituted-1,3,4-oxadiazoles
-
P. Chawla, R. Maheshwari and S. A. Saraf, "Synthesis and evaluation of anti-inflammatory and antimicrobial activities of 2,5-disubstituted-1,3,4- oxadiazoles", Der Pharma Chemica, 2 (4), 38-45 (2010).
-
(2010)
Der Pharma Chemica
, vol.2
, Issue.4
, pp. 38-45
-
-
Chawla, P.1
Maheshwari, R.2
Saraf, S.A.3
-
25
-
-
0017766654
-
Oxidation of 1,2-diaminobenzimidazole to 3-amino-1,2,4-benzotriazines
-
A. V. Zeiger and M. M. Joullié, "Oxidation of 1,2-diaminobenzimidazole to 3-amino-1,2,4-benzotriazines", J. Org. Chem., 42, 542-545 (1977).
-
(1977)
J. Org. Chem.
, vol.42
, pp. 542-545
-
-
Zeiger, A.V.1
Joullié, M.M.2
-
26
-
-
0004262889
-
-
Academic Press, New York
-
H. William, "Microbiological Assay, An Introduction to Quantitative Principles and Evaluation", Academic Press, New York, 1977, pp 1-68.
-
(1977)
Microbiological Assay, An Introduction to Quantitative Principles and Evaluation
, pp. 1-68
-
-
William, H.1
-
29
-
-
0028352765
-
Anti-inflammatory activity of substituted 1,3,4-oxadiazoles
-
L. V. Nargund, G. R. Reddy and V. Hariprasad, "Anti-inflammatory activity of substituted 1,3,4-oxadiazoles", J. Pharm. Sci., 83, 246-248 (1994).
-
(1994)
J. Pharm. Sci.
, vol.83
, pp. 246-248
-
-
Nargund, L.V.1
Reddy, G.R.2
Hariprasad, V.3
-
30
-
-
0004313709
-
-
version 2009.06. Montreal, Quebec, Canada
-
"Molecular Operating Environment (MOE)", version 2009.06. Chemical Computing Group, Inc. Montreal, Quebec, Canada, 2009, http://www.chemcomp.com.
-
(2009)
Molecular Operating Environment (MOE)
-
-
-
31
-
-
0009979056
-
-
Weissberger, A., editor, John Wiely and Sons, New York
-
D. M. Smith, "Chemistry of Heterocyclic Compounds", Vol. 40, part I, Weissberger, A., editor, John Wiely and Sons, New York, 1981, p. 331.
-
(1981)
Chemistry of Heterocyclic Compounds
, vol.40
, Issue.PART I
, pp. 331
-
-
Smith, D.M.1
-
32
-
-
60549092516
-
Synthesis of some new 1,2,4-triazoles, their Mannich and Schiff bases and evaluation of their antimicrobial activities
-
H. Bayrak, A. Demirbas, S. A. Karaoglu and N. Demirbas, "Synthesis of some new 1,2,4-triazoles, their Mannich and Schiff bases and evaluation of their antimicrobial activities", Eur. J. Med. Chem., 44, 1057-1066 (2009).
-
(2009)
Eur. J. Med. Chem.
, vol.44
, pp. 1057-1066
-
-
Bayrak, H.1
Demirbas, A.2
Karaoglu, S.A.3
Demirbas, N.4
-
33
-
-
0032583456
-
Synthesis and antimicrobial activity of N-[(α-methyl)benzylidene]- (3-substituted-1,2,4-triazol-5-yl-thio) acetohydrazides
-
S. Ersan, S. Nacak and R. Berkem, "Synthesis and antimicrobial activity of N-[(α-methyl)benzylidene]-(3-substituted-1,2,4-triazol-5-yl- thio) acetohydrazides", Il Farmaco, 53, 773-776 (1998).
-
(1998)
Il Farmaco
, vol.53
, pp. 773-776
-
-
Ersan, S.1
Nacak, S.2
Berkem, R.3
-
34
-
-
0035439443
-
Synthesis and receptor docking studies of N-substituted indole-2-carboxylic acid esters as a search for COX-2 selective enzyme inhibitors
-
S. Olgen, E. Akaho and D. Nebioglu, "Synthesis and receptor docking studies of N-substituted indole-2-carboxylic acid esters as a search for COX-2 selective enzyme inhibitors", Eur. J. Med. Chem., 36, 747-770 (2001).
-
(2001)
Eur. J. Med. Chem.
, vol.36
, pp. 747-770
-
-
Olgen, S.1
Akaho, E.2
Nebioglu, D.3
-
35
-
-
0036136418
-
Molecular modelling of the differential interaction between several non-steroidal anti-inflammatory drugs and human prostaglandin endoperoxide H synthase-2 (h-PGHS-2)
-
R. Pouplana, J. J. Lozano and J. Ruiz, "Molecular modelling of the differential interaction between several non-steroidal anti-inflammatory drugs and human prostaglandin endoperoxide H synthase-2 (h-PGHS-2)", J. Molecular Graphics and Modeling, 20, 329 (2002).
-
(2002)
J. Molecular Graphics and Modeling
, vol.20
, pp. 329
-
-
Pouplana, R.1
Lozano, J.J.2
Ruiz, J.3
|