메뉴 건너뛰기




Volumn 101, Issue 8, 2012, Pages 2777-2786

Naltrexone salt selection for enhanced transdermal permeation through microneedle-treated skin

Author keywords

Diffusion; In vitro models; Microneedles; Naltrexone; Permeability; Salts; Skin; Solubility; Transdermal drug delivery

Indexed keywords

NALTREXONE;

EID: 84862884589     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.23189     Document Type: Article
Times cited : (12)

References (23)
  • 1
    • 1342346643 scopus 로고    scopus 로고
    • The stratum corneum: Structure and function in health and disease
    • Harding Clive R. 2004. The stratum corneum: Structure and function in health and disease. Dermatol Ther 17(Suppl 1):6-15.
    • (2004) Dermatol Ther , vol.17 , Issue.SUPPL. 1 , pp. 6-15
    • Harding, C.R.1
  • 2
    • 0042121374 scopus 로고    scopus 로고
    • Barrier function of the skin: "La raison d'etre" of the epidermis
    • Madison KC. 2003. Barrier function of the skin: "La raison d'etre" of the epidermis. J Invest Dermatol 121(2):231-241.
    • (2003) J Invest Dermatol , vol.121 , Issue.2 , pp. 231-241
    • Madison, K.C.1
  • 3
    • 1242308254 scopus 로고    scopus 로고
    • Current status and future potential of transdermal drug delivery
    • Prausnitz MR, Mitragotri S, Langer R. 2004. Current status and future potential of transdermal drug delivery. Nat Rev Drug Discov 3(2):115-124.
    • (2004) Nat Rev Drug Discov , vol.3 , Issue.2 , pp. 115-124
    • Prausnitz, M.R.1    Mitragotri, S.2    Langer, R.3
  • 4
    • 55749108348 scopus 로고    scopus 로고
    • Transdermal drug delivery
    • Prausnitz MR, Langer R. 2008. Transdermal drug delivery. Nat Biotechnol 26(11):1261-1268.
    • (2008) Nat Biotechnol , vol.26 , Issue.11 , pp. 1261-1268
    • Prausnitz, M.R.1    Langer, R.2
  • 5
    • 55649101168 scopus 로고    scopus 로고
    • Micro-scale devices for transdermal drug delivery
    • Arora A, Prausnitz MR, Mitragotri S. 2008. Micro-scale devices for transdermal drug delivery. Int J Pharm 364(2):227-236.
    • (2008) Int J Pharm , vol.364 , Issue.2 , pp. 227-236
    • Arora, A.1    Prausnitz, M.R.2    Mitragotri, S.3
  • 8
    • 55249125056 scopus 로고    scopus 로고
    • Effect of microneedle design on pain in human volunteers
    • Gill HS, Denson DD, Burris BA, Prausnitz MR. 2008. Effect of microneedle design on pain in human volunteers. Clin J Pain 24(7):585-594.
    • (2008) Clin J Pain , vol.24 , Issue.7 , pp. 585-594
    • Gill, H.S.1    Denson, D.D.2    Burris, B.A.3    Prausnitz, M.R.4
  • 10
    • 27644450531 scopus 로고    scopus 로고
    • Transdermal delivery of naltrexone and its active metabolite 6-beta-naltrexol in human skin in vitro and guinea pigs in vivo
    • Paudel KS, Nalluri BN, Hammell DC, Valiveti S, Kiptoo P, Hamad MO, Crooks PA, Stinchcomb AL. 2005. Transdermal delivery of naltrexone and its active metabolite 6-beta-naltrexol in human skin in vitro and guinea pigs in vivo. J Pharm Sci 94(9):1965-1975.
    • (2005) J Pharm Sci , vol.94 , Issue.9 , pp. 1965-1975
    • Paudel, K.S.1    Nalluri, B.N.2    Hammell, D.C.3    Valiveti, S.4    Kiptoo, P.5    Hamad, M.O.6    Crooks, P.A.7    Stinchcomb, A.L.8
  • 11
    • 44649083690 scopus 로고    scopus 로고
    • Flux across microneedle-treated skin is increased by increasing charge of naltrexone and naltrexol in vitro
    • Banks SL, Pinninti RR, Gill HS, Crooks PA, Prausnitz MR, Stinchcomb AL. 2008. Flux across microneedle-treated skin is increased by increasing charge of naltrexone and naltrexol in vitro. Pharm Res 25(7):1677-1685.
    • (2008) Pharm Res , vol.25 , Issue.7 , pp. 1677-1685
    • Banks, S.L.1    Pinninti, R.R.2    Gill, H.S.3    Crooks, P.A.4    Prausnitz, M.R.5    Stinchcomb, A.L.6
  • 15
    • 33846492454 scopus 로고    scopus 로고
    • Coated microneedles for transdermal delivery
    • Gill HS, Prausnitz MR. 2007. Coated microneedles for transdermal delivery. In J. Control Release 117 (2): 227-237.
    • (2007) J. Control Release , vol.117 , Issue.2 , pp. 227-237
    • Gill, H.S.1    Prausnitz, M.R.2
  • 16
    • 0023264053 scopus 로고
    • Improvement of the oral bioavailability of naltrexone in dogs: A prodrug approach
    • Hussain MA, Koval CA, Myers MJ, Shami EG, Shefter E. 1987. Improvement of the oral bioavailability of naltrexone in dogs: A prodrug approach. J Pharm Sci 76(5):356-358.
    • (1987) J Pharm Sci , vol.76 , Issue.5 , pp. 356-358
    • Hussain, M.A.1    Koval, C.A.2    Myers, M.J.3    Shami, E.G.4    Shefter, E.5
  • 17
    • 78651254362 scopus 로고    scopus 로고
    • Vehicle composition influence on the microneedle-enhanced transdermal flux of naltrexone hydrochloride
    • Milewski M, Stinchcomb AL. 2010. Vehicle composition influence on the microneedle-enhanced transdermal flux of naltrexone hydrochloride. Pharm Res 28(1):124-134.
    • (2010) Pharm Res , vol.28 , Issue.1 , pp. 124-134
    • Milewski, M.1    Stinchcomb, A.L.2
  • 18
    • 0016741904 scopus 로고
    • Microelectrometric titration measurement of the pKa's and partition and drug distribution coefficients of narcotics and narcotic antagonists and their pH and temperature dependence
    • Kaufman JJ, Semo NM, Koski WS. 1975. Microelectrometric titration measurement of the pKa's and partition and drug distribution coefficients of narcotics and narcotic antagonists and their pH and temperature dependence. J Med Chem 18(7):647-655.
    • (1975) J Med Chem , vol.18 , Issue.7 , pp. 647-655
    • Kaufman, J.J.1    Semo, N.M.2    Koski, W.S.3
  • 19
    • 34548032742 scopus 로고    scopus 로고
    • Salt formation to improve drug solubility
    • Serajuddin ATM. 2007. Salt formation to improve drug solubility. Adv Drug Deliv Rev 59(7):603-616.
    • (2007) Adv Drug Deliv Rev , vol.59 , Issue.7 , pp. 603-616
    • Serajuddin, A.T.M.1
  • 20
    • 36048955468 scopus 로고    scopus 로고
    • Partitioning, diffusivity and clearance of skin permeants in mammalian dermis
    • Kretsos K, Miller MA, Zamora-Estrada G, Kasting GB. 2008. Partitioning, diffusivity and clearance of skin permeants in mammalian dermis. Int J Pharm 346(1-2):64-79.
    • (2008) Int J Pharm , vol.346 , Issue.1-2 , pp. 64-79
    • Kretsos, K.1    Miller, M.A.2    Zamora-Estrada, G.3    Kasting, G.B.4
  • 21
    • 0001813673 scopus 로고
    • Cutaneous and transdermal delivery: processes and systems of delivery
    • Banker GS, Rhodes CT, Eds. 2nd ed. New York: Marcel Dekker
    • Flynn GL. 1990. Cutaneous and transdermal delivery: processes and systems of delivery. In Modern pharmaceutics; Banker GS, Rhodes CT, Eds. 2nd ed. New York: Marcel Dekker. pp 239-298.
    • (1990) Modern pharmaceutics; , pp. 239-298
    • Flynn, G.L.1
  • 22
    • 84862860415 scopus 로고    scopus 로고
    • FDA. Alpha hydroxy acids in cosmetics. Silver Spring, Maryland: FDA
    • FDA. 2009. Alpha hydroxy acids in cosmetics. Silver Spring, Maryland: FDA
    • (2009)


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.