메뉴 건너뛰기




Volumn 77, Issue 8-9, 2012, Pages 845-849

Synthesis and bioassay of a boron-dipyrromethene derivative of estradiol for fluorescence imaging in vivo

Author keywords

BODIPY; Estrogen receptor; Uterus

Indexed keywords

ALKENE; BORON DIPYRROMETHENE DERIVATIVE; ESTRADIOL; ESTROGEN RECEPTOR; UNCLASSIFIED DRUG;

EID: 84861651774     PISSN: 0039128X     EISSN: 18785867     Source Type: Journal    
DOI: 10.1016/j.steroids.2012.04.011     Document Type: Article
Times cited : (17)

References (16)
  • 1
    • 0028919090 scopus 로고
    • Estrogen receptors in human nontarget tissues: Biological and clinical implications
    • D.R. Ciocca, and L.M. Roig Estrogen receptors in human nontarget tissues: biological and clinical implications Endocr Rev 16 1995 35 62
    • (1995) Endocr Rev , vol.16 , pp. 35-62
    • Ciocca, D.R.1    Roig, L.M.2
  • 2
    • 0028283503 scopus 로고
    • Molecular mechanisms of action of steroid/thyroid receptor superfamily members
    • M.J. Tsai, and B.W. O'Malley Molecular mechanisms of action of steroid/thyroid receptor superfamily members Annu Rev Biochem 63 1994 451 486 (Pubitemid 24218640)
    • (1994) Annual Review of Biochemistry , vol.63 , pp. 451-486
    • Tsai, M.-J.1    O'Malley, B.W.2
  • 4
    • 32144447789 scopus 로고    scopus 로고
    • High affinity 17α-substituted estradiol derivatives: Synthesis and evaluation of estrogen receptor agonist activity
    • DOI 10.1016/j.steroids.2005.10.004, PII S0039128X05002606
    • K.M. Kasiotis, C. Mendorou, S.A. Haroutounian, and M.N. Alexis High affinity 17alpha-substituted estradiol derivatives: synthesis and evaluation of estrogen receptor agonist activity Steroids 71 2006 249 255 (Pubitemid 43208961)
    • (2006) Steroids , vol.71 , Issue.3 , pp. 249-255
    • Kasiotis, K.M.1    Mendorou, C.2    Haroutounian, S.A.3    Alexis, M.N.4
  • 5
    • 0033571579 scopus 로고    scopus 로고
    • An ultrahigh-throughput screening assay for estrogen receptor ligands
    • G.F. Allan, A. Hutchins, and J. Clancy An ultrahigh-throughput screening assay for estrogen receptor ligands Anal Biochem 275 1999 243 247
    • (1999) Anal Biochem , vol.275 , pp. 243-247
    • Allan, G.F.1    Hutchins, A.2    Clancy, J.3
  • 8
    • 0345440144 scopus 로고    scopus 로고
    • Synthesis and binding affinities of novel Re-containing 7alpha-substituted estradiol complexes: Models for breast cancer imaging agents
    • M.B. Skaddan, F.R. Wust, and J.A. Katzenellenbogen Synthesis and binding affinities of novel Re-containing 7alpha-substituted estradiol complexes: models for breast cancer imaging agents J Org Chem 64 1999 8108 8121
    • (1999) J Org Chem , vol.64 , pp. 8108-8121
    • Skaddan, M.B.1    Wust, F.R.2    Katzenellenbogen, J.A.3
  • 9
    • 0027270144 scopus 로고
    • A synthesis of 7 alpha-substituted estradiols: Synthesis and biological evaluation of a 7 alpha-pentyl substituted BODIPY fluorescent conjugate and a fluorine-18-labeled 7 alpha-pentylestradiol analog
    • A.N. French, S.R. Wilson, M.J. Welch, and J.A. Katzenellenbogen A synthesis of 7 alpha-substituted estradiols: synthesis and biological evaluation of a 7 alpha-pentyl substituted BODIPY fluorescent conjugate and a fluorine-18-labeled 7 alpha-pentylestradiol analog Steroids 58 1993 157 169
    • (1993) Steroids , vol.58 , pp. 157-169
    • French, A.N.1    Wilson, S.R.2    Welch, M.J.3    Katzenellenbogen, J.A.4
  • 10
    • 36849053388 scopus 로고    scopus 로고
    • BODIPY dyes and their derivatives: Syntheses and spectroscopic properties
    • DOI 10.1021/cr078381n
    • A. Loudet, and K. Burgess BODIPY dyes and their derivatives: syntheses and spectroscopic properties Chem Rev 107 2007 4891 4932 (Pubitemid 350225866)
    • (2007) Chemical Reviews , vol.107 , Issue.11 , pp. 4891-4932
    • Loudet, A.1    Burgess, K.2
  • 11
    • 0027255941 scopus 로고
    • Surprising places of estrogenic activity
    • K.S. Korach Surprising places of estrogenic activity Endocrinology 132 1993 2277 2278
    • (1993) Endocrinology , vol.132 , pp. 2277-2278
    • Korach, K.S.1
  • 12
    • 0030498123 scopus 로고    scopus 로고
    • Assessing environmental chemicals for estrogenicity using a combination of in vitro and in vivo assays
    • M.D. Shelby, R.R. Newbold, D.B. Tully, K. Chae, and V.L. Davis Assessing environmental chemicals for estrogenicity using a combination of in vitro and in vivo assays Environ Health Perspect 104 1996 1296 1300 (Pubitemid 27065080)
    • (1996) Environmental Health Perspectives , vol.104 , Issue.12 , pp. 1296-1300
    • Shelby, M.D.1    Newbold, R.R.2    Tully, D.B.3    Chae, K.4    Davis, V.L.5
  • 14
    • 0032052810 scopus 로고    scopus 로고
    • An updated review of environmental estrogen and androgen mimics and antagonists
    • DOI 10.1016/S0960-0760(98)00027-2, PII S0960076098000272
    • C. Sonnenschein, and A.M. Soto An updated review of environmental estrogen and androgen mimics and antagonists J Steroid Biochem Mol Biol 65 1998 143 150 (Pubitemid 28335600)
    • (1998) Journal of Steroid Biochemistry and Molecular Biology , vol.65 , Issue.1-6 , pp. 143-150
    • Sonnenschein, C.1    Soto, A.M.2
  • 15
    • 33847675759 scopus 로고    scopus 로고
    • Synthesis of borondipyrromethene (BODIPY)-labeled sphingosine derivatives by cross-metathesis reaction
    • DOI 10.1021/jo062347b
    • C. Peters, A. Billich, M. Ghobrial, K. Hogenauer, T. Ullrich, and P. Nussbaumer Synthesis of borondipyrromethene (BODIPY)-labeled sphingosine derivatives by cross-metathesis reaction J Org Chem 72 2007 1842 1845 (Pubitemid 46355490)
    • (2007) Journal of Organic Chemistry , vol.72 , Issue.5 , pp. 1842-1845
    • Peters, C.1    Billich, A.2    Ghobrial, M.3    Hogenauer, K.4    Ullrich, T.5    Nussbaumer, P.6
  • 16
    • 0028818201 scopus 로고
    • The E-SCREEN assay as a tool to identify estrogens: An update on estrogenic environmental pollutants
    • A.M. Soto, C. Sonnenschein, K.L. Chung, M.F. Fernandez, N. Olea, and F.O. Serrano The E-SCREEN assay as a tool to identify estrogens: an update on estrogenic environmental pollutants Environ Health Perspect 103 Suppl. 7 1995 113 122
    • (1995) Environ Health Perspect , vol.103 , Issue.SUPPL. 7 , pp. 113-122
    • Soto, A.M.1    Sonnenschein, C.2    Chung, K.L.3    Fernandez, M.F.4    Olea, N.5    Serrano, F.O.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.